4.6 Article

The Promise and Peril of Chemical Probe Negative Controls

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Medicinal

Discovery of CPI-1612: A Potent, Selective, and Orally Bioavailable EP300/CBP Histone Acetyltransferase Inhibitor

Jonathan E. Wilson et al.

ACS MEDICINAL CHEMISTRY LETTERS (2020)

Article Biochemistry & Molecular Biology

Systematic Chemogenetic Library Assembly

Stephen M. Canham et al.

CELL CHEMICAL BIOLOGY (2020)

Article Biochemistry & Molecular Biology

Objective, Quantitative, Data-Driven Assessment of Chemical Probes

Albert A. Antolin et al.

CELL CHEMICAL BIOLOGY (2018)

Article Biochemistry & Molecular Biology

The SUV4-20 inhibitor A-196 verifies a role for epigenetics in genomic integrity

Kenneth D. Bromberg et al.

NATURE CHEMICAL BIOLOGY (2017)

Letter Biochemical Research Methods

Probes & Drugs portal: an interactive, open data resource for chemical biology

Ctibor Skuta et al.

NATURE METHODS (2017)

Review Biotechnology & Applied Microbiology

Applications of chemogenomic library screening in drug discovery

Lyn H. Jones et al.

NATURE REVIEWS DRUG DISCOVERY (2017)

Article Biotechnology & Applied Microbiology

Comprehensive characterization of the Published Kinase Inhibitor Set

Jonathan M. Elkins et al.

NATURE BIOTECHNOLOGY (2016)

Article Multidisciplinary Sciences

Integrated genetic and pharmacologic interrogation of rare cancers

Andrew L. Hong et al.

NATURE COMMUNICATIONS (2016)

Article Biochemistry & Molecular Biology

Selective JAK3 Inhibitors with a Covalent Reversible Binding Mode Targeting a New Induced Fit Binding Pocket

Michael Forster et al.

CELL CHEMICAL BIOLOGY (2016)

Article Biochemistry & Molecular Biology

LLY-507, a Cell-active, Potent, and Selective Inhibitor of Protein-lysine Methyltransferase SMYD2

Hannah Nguyen et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2015)

Article Biochemistry & Molecular Biology

The promise and peril of chemical probes

Cheryl H. Arrowsmith et al.

NATURE CHEMICAL BIOLOGY (2015)

Article Multidisciplinary Sciences

Comprehensive prediction of drug-protein interactions and side effects for the human proteome

Hongyi Zhou et al.

SCIENTIFIC REPORTS (2015)

News Item Biochemistry & Molecular Biology

Follow your lead

Brian K. Shoichet

NATURE CHEMICAL BIOLOGY (2014)

Article Biochemistry & Molecular Biology

Dual kinase-bromodomain inhibitors for rationally designed polypharmacology

Pietro Ciceri et al.

NATURE CHEMICAL BIOLOGY (2014)

Article Multidisciplinary Sciences

Activation and allosteric modulation of a muscarinic acetylcholine receptor

Andrew C. Kruse et al.

NATURE (2013)

Article Biochemistry & Molecular Biology

Target validation using chemical probes

Mark E. Bunnage et al.

NATURE CHEMICAL BIOLOGY (2013)

Article Biochemistry & Molecular Biology

The art of the chemical probe

Stephen V. Frye

NATURE CHEMICAL BIOLOGY (2010)