相关参考文献
注意：仅列出部分参考文献，下载原文获取全部文献信息。Correlating Drug-Target Residence Time and Post-antibiotic Effect: Insight into Target Vulnerability
Shabnam Davoodi et al.
ACS INFECTIOUS DISEASES (2020)
Targeting drugs for tuberculosis
Trever C. Smith et al.
SCIENCE (2019)
Drug permeation and metabolism in Mycobacterium tuberculosis: Prioritising local exposure as essential criterion in new TB drug development
Lloyd Tanner et al.
IUBMB LIFE (2018)
Kinetics of drug-ribosome interactions defines the cidality of macrolide antibiotics
Maxim S. Svetlov et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2017)
Insights into the slow-onset tight-binding inhibition of Escherichia coli dihydrofolate reductase: detailed mechanistic characterization of pyrrolo [3,2-f] quinazoline-1,3-diamine and its derivatives as novel tight-binding inhibitors
Bharath Srinivasan et al.
FEBS JOURNAL (2015)
Translating slow-binding inhibition kinetics into cellular and in vivo effects
Grant K. Walkup et al.
NATURE CHEMICAL BIOLOGY (2015)
Lipoamide Channel-Binding Sulfonamides Selectively Inhibit Mycobacterial Lipoamide Dehydrogenase
Ruslana Bryk et al.
BIOCHEMISTRY (2013)
Virulence of Mycobacterium tuberculosis Depends on Lipoamide Dehydrogenase, a Member of Three Multienzyme Complexes
Aditya Venugopal et al.
CELL HOST & MICROBE (2011)
MolProbity: all-atom structure validation for macromolecular crystallography
Vincent B. Chen et al.
ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY (2010)
PHENIX: a comprehensive Python-based system for macromolecular structure solution
Paul D. Adams et al.
ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY (2010)
Triazaspirodimethoxybenzoyls as Selective Inhibitors of Mycobacterial Lipoamide Dehydrogenase
Ruslana Bryk et al.
BIOCHEMISTRY (2010)
Casuarine-6-O-alpha-D-glucoside and its analogues are tight binding inhibitors of insect and bacterial trehalases
Francesca Cardona et al.
CHEMICAL COMMUNICATIONS (2010)
Biochemical characterization of GSK1070916, a potent and selective inhibitor of Aurora B and Aurora C kinases with an extremely long residence time
Kelly Anderson et al.
BIOCHEMICAL JOURNAL (2009)
Selective killing of nonreplicating mycobacteria
Ruslana Bryk et al.
CELL HOST & MICROBE (2008)
Biosynthesis and recycling of nicotinamide cofactors in Mycobacterium tuberculosis -: An essential role for NAD in nonreplicating bacilli
Helena I. M. Boshoff et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2008)
The protonmotive force is required for maintaining ATP homeostasis and viability of hypoxic, nonreplicating Mycobacterium tuberculosis
Srinivasa P. S. Rao et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2008)
New method for fast and accurate binding-site identification and analysis
Tom Halgren
CHEMICAL BIOLOGY & DRUG DESIGN (2007)
Opinion - Drug-target residence time and its implications for lead optimization
Robert A. Copeland et al.
NATURE REVIEWS DRUG DISCOVERY (2006)
A slow, tight-binding inhibitor of the zinc-dependent deacetylase LpxC of lipid a biosynthesis with antibiotic activity comparable to ciprofloxacin
AL McClerren et al.
BIOCHEMISTRY (2005)
Crystal structure and functional analysis of lipoamide dehydrogenase from Mycobacterium tuberculosis
KR Rajashankar et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2005)
Mycobacterium tuberculosis appears to lack α-ketoglutarate dehydrogenase and encodes pyruvate dehydrogenase in widely separated genes
J Tian et al.
MOLECULAR MICROBIOLOGY (2005)
Glide: A new approach for rapid, accurate docking and scoring. 1. Method and assessment of docking accuracy
RA Friesner et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
Coot:: model-building tools for molecular graphics
P Emsley et al.
ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY (2004)
Metabolic enzymes of mycobacteria linked to antioxidant defense by a thioredoxin-like protein
R Bryk et al.
SCIENCE (2002)
Peroxynitrite reductase activity of bacterial peroxiredoxins
R Bryk et al.
NATURE (2000)
分享论文
