相关参考文献
注意：仅列出部分参考文献，下载原文获取全部文献信息。Thiosemicarbazones as Potent Anticancer Agents and their Modes of Action
Bhushan Shakya et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2020)
Imidazo[2,1-b] [1,3,4]thiadiazoles with antiproliferative activity against primary and gemcitabine-resistant pancreatic cancer cells
Stella Cascioferro et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Thiazole-containing compounds as therapeutic targets for cancer therapy
Prabodh Chander Sharma et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Synthesis, Characterization, Antibacterial Activity, and Computer-Aided Design of Novel Quinazolin-2,4-dione Derivatives as Potential Inhibitors Against Vibrio cholerae
Mohamed El-Naggar et al.
EVOLUTIONARY BIOINFORMATICS (2020)
Synthesis, in vitro biological evaluation and in silico docking studies of new quinazolin-2,4-dione analogues as possible anticarcinoma agents
Aboubakr H. Abdelmonsef et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2020)
3-(6-Phenylimidazo [2,1-b][1,3,4]thiadiazol-2-yl)-1H-Indole Derivatives as New Anticancer Agents in the Treatment of Pancreatic Ductal Adenocarcinoma
Stella Cascioferro et al.
MOLECULES (2020)
A perspective on environmentally benign protocols of thiazole synthesis
Arnab Chowdhury et al.
CHEMISTRY OF HETEROCYCLIC COMPOUNDS (2020)
Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance
Stella Cascioferro et al.
JOURNAL OF MEDICINAL CHEMISTRY (2020)
One-Pot Synthesis of Novel Thiazoles as Potential Anti-Cancer Agents
Abdelwahed R. Sayed et al.
DRUG DESIGN DEVELOPMENT AND THERAPY (2020)
Thiophene-based derivatives as anticancer agents: An overview on decade's work
Archna et al.
BIOORGANIC CHEMISTRY (2020)
Novel Quinazolin-2,4-Dione Hybrid Molecules as Possible Inhibitors Against Malaria: Synthesis andin silicoMolecular Docking Studies
Aboubakr Haredi Abdelmonsef et al.
FRONTIERS IN MOLECULAR BIOSCIENCES (2020)
Knockdown of Rab7a suppresses the proliferation, migration, and xenograft tumor growth of breast cancer cells
Jiming Xie et al.
BIOSCIENCE REPORTS (2019)
Homology modeling in drug discovery: Overview, current applications, and future perspectives
Muhammed Tilahun Muhammed et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2019)
Synthesis and Biological Evaluation of Some Novel Thiazole-Based Heterocycles as Potential Anticancer and Antimicrobial Agents
Sraa Abu-Melha et al.
MOLECULES (2019)
In silico ADMET study, docking, synthesis and antimalarial evaluation of thiazole-1,3,5-triazine derivatives as Pf-DHFR inhibitor
Supriya Sahu et al.
PHARMACOLOGICAL REPORTS (2019)
Design, efficient synthesis and molecular docking of some novel thiazolyl-pyrazole derivatives as anticancer agents
Abdelwahed R. Sayed et al.
BMC CHEMISTRY (2019)
Study of the impact of consanguinity on abortion and mortality in the population of Beni Abbes (southwestern Algeria)
Said Bachir et al.
EGYPTIAN JOURNAL OF MEDICAL HUMAN GENETICS (2019)
New anticancer drug candidates sulfonamides as selective hCA IX or hCA XII inhibitors
Halise Inci Gul et al.
BIOORGANIC CHEMISTRY (2018)
Surmounting the resistance against EGFR inhibitors through the development of thieno[2,3-d]pyrimidine-based dual EGFR/HER2 inhibitors
Sandra N. Milik et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
One-Pot Synthesis of New Thiadiazolyl-Pyridines as Anticancer and Antioxidant Agents
Sobhi M. Gomha et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2018)
Synthesis and Molecular Docking of Some Novel Thiazoles and Thiadiazoles Incorporating Pyranochromene Moiety as Potent Anticancer Agents
Sobhi M. Gomha et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2018)
CASTp 3.0: computed atlas of surface topography of proteins
Wei Tian et al.
NUCLEIC ACIDS RESEARCH (2018)
5-(Thiophen-2-yl)-1,3,4-thiadiazole derivatives: synthesis, molecular docking and in vitro cytotoxicity evaluation as potential anticancer agents
Sobhi M. Gomha et al.
DRUG DESIGN DEVELOPMENT AND THERAPY (2018)
Eco-friendly one-pot synthesis of some new pyrazolo[1,2-b]phthalazinediones with antiproliferative efficacy on human hepatic cancer cell lines
Huda R. M. Rashdan et al.
GREEN CHEMISTRY LETTERS AND REVIEWS (2018)
TBC1D5 controls the GTPase cycle of Rab7b
Marita Borg Distefano et al.
JOURNAL OF CELL SCIENCE (2018)
Eco-Friendly Synthesis, Characterization and Biological Evaluation of Some Novel Pyrazolines Containing Thiazole Moiety as Potential Anticancer and Antimicrobial Agents
Mastoura M. Edrees et al.
MOLECULES (2018)
Design of novel lead molecules against RhoG protein as cancer target - a computational study
Thirupathi Dasari et al.
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS (2017)
Design and synthesis of imidazo[2,1-b]thiazole linked triazole conjugates: Microtubule-destabilizing agents
Siddiq Pasha Shaik et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Synthesis, characterization, antimicrobial activity and theoretical studies of new thiophene-based tripodal ligands
Tank Harit et al.
JOURNAL OF MOLECULAR STRUCTURE (2017)
Synthesis and cytotoxicity evaluation of thiazole derivatives obtained from 2-amino-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carbonitrile
Rafat M. Mohareb et al.
ACTA PHARMACEUTICA (2017)
A facile access and evaluation of some novel thiazole and 1,3,4-thiadiazole derivatives incorporating thiazole moiety as potent anticancer agents
Sobhi M. Gomha et al.
CHEMISTRY CENTRAL JOURNAL (2017)
Design, synthesis, in silico and in vitro evaluation of thiophene derivatives: A potent tyrosine phosphatase 1B inhibitor and anticancer activity
Kali Charan Gulipalli et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2017)
A facile synthesis and anticancer activity of some novel thiazoles carrying 1,3,4-thiadiazole moiety
Sobhi M. Gomha et al.
CHEMISTRY CENTRAL JOURNAL (2017)
Synthesis and cytotoxicity evaluation of thiosemicarbazones and their thiazole derivatives
Saulo Feheiberg Pinto Braga et al.
BRAZILIAN JOURNAL OF PHARMACEUTICAL SCIENCES (2016)
Identification of Novel Antagonists for Rab38 Protein by Homology Modeling and Virtual Screening
Aboubakr Haredi Abdelmonsef et al.
COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING (2016)
Recent developments of 2-aminothiazoles in medicinal chemistry
Debasis Das et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
SYNTHESIS OF SOME NOVEL THIAZOLE, THIADIAZOLE AND 1,4-PHENYLENE-BIS-THIAZOLE DERIVATIVES AS POTENT ANTITUMOR AGENTS
Sobhi M. Gomha et al.
HETEROCYCLES (2016)
Synthesis of New 3-Heteroarylindoles as Potential Anticancer Agents
Abdou O. Abdelhamid et al.
MOLECULES (2016)
Synthesis and Characterization of Some New Bis-Pyrazolyl-Thiazoles Incorporating the Thiophene Moiety as Potent Anti-Tumor Agents
Sobhi M. Gomha et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2016)
Synthesis, biological evaluation and 3D-QSAR study of novel 4,5-dihydro-1H-pyrazole thiazole derivatives as BRAF(V600E) inhibitors
Meng-Yue Zhao et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2015)
Cancer Statistics, 2015
Rebecca L. Siegel et al.
CA-A CANCER JOURNAL FOR CLINICIANS (2015)
Synthesis and anticancer activity of arylazothiazoles and 1,3,4-thiadiazoles using chitosan-grafted-poly(4-vinylpyridine) as a novel copolymer basic catalyst
Sobhi M. Gomha et al.
CHEMISTRY OF HETEROCYCLIC COMPOUNDS (2015)
Recent applications of 1,3-thiazole core structure in the identification of new lead compounds and drug discovery
Adile Ayati et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
SYNTHESIS AND ANTICANCER ACTIVITIES OF THIAZOLES, 1,3-THIAZINES, AND THIAZOLIDINE USING CHITOSAN-GRAFTEDPOLY(VINYLPYRIDINE) AS BASIC CATALYST
Sobhi M. Gomha et al.
HETEROCYCLES (2015)
Cellular functions of Rab GTPases at a glance
Yan Zhen et al.
JOURNAL OF CELL SCIENCE (2015)
In silico ADME/T modelling for rational drug design
Yulan Wang et al.
QUARTERLY REVIEWS OF BIOPHYSICS (2015)
In vitro and in silico antimalarial activity of 2-(2-hydrazinyl)thiazole derivatives
Parameshwar Makam et al.
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES (2014)
Cisplatin in cancer therapy: Molecular mechanisms of action
Shaloam Dasari et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2014)
5-FU and ixabepilone modify the microRNA expression profiles in MDA-MB-453 triple-negative breast cancer cells
Yongshan Yao et al.
ONCOLOGY LETTERS (2014)
Synthesis and biological evaluation of thieno [2′,3′:4,5]pyrimido[1,2-b][1,2,4]triazines and thieno[2,3-d][1,2,4]triazolo[1,5-a]pyrimidines as anti-inflammatory and analgesic agents
Hayam M. Ashour et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
admetSAR: A Comprehensive Source and Free Tool for Assessment of Chemical ADMET Properties
Feixiong Cheng et al.
JOURNAL OF CHEMICAL INFORMATION AND MODELING (2012)
Immune regulation of Rab proteins expression and intracellular transport
Gang Pei et al.
JOURNAL OF LEUKOCYTE BIOLOGY (2012)
Dynamics of Rab7b-Dependent Transport of Sorting Receptors
Cinzia Progida et al.
TRAFFIC (2012)
Design, Synthesis, and SAR Studies of 4-Substituted Methoxylbenzoyl-aryl-thiazoles Analogues as Potent and Orally Bioavailable Anticancer Agents
Yan Lu et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Challenges and advances in computational docking: 2009 in review
Elizabeth Yuriev et al.
JOURNAL OF MOLECULAR RECOGNITION (2011)
Novel Synthesis of Hydrazide-Hydrazone Derivatives and Their Utilization in the Synthesis of Coumarin, Pyridine, Thiazole and Thiophene Derivatives with Antitumor Activity
Rafat M. Mohareb et al.
MOLECULES (2011)
Open Babel: An open chemical toolbox
Noel M. O'Boyle et al.
JOURNAL OF CHEMINFORMATICS (2011)
Rab7b controls trafficking from endosomes to the TGN
Cinzia Progida et al.
JOURNAL OF CELL SCIENCE (2010)
Comparative binding energy analysis for binding affinity and target selectivity prediction
Stefan Henrich et al.
PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS (2010)
Characterization of Dasatinib and Its Structural Analogs as CYP3A4 Mechanism-Based Inactivators and the Proposed Bioactivation Pathways
Xiaohai Li et al.
DRUG METABOLISM AND DISPOSITION (2009)
Potential Antitumor Agents.: 42.: New antitumor imidazo[2,1-b]thiazole guanylhydrazones and analogues'
Aldo Andreani et al.
JOURNAL OF MEDICINAL CHEMISTRY (2008)
2,4-dimethoxyphenylsemicarbazones with anticonvulsant activity against three animal models of seizures: Synthesis and pharmacological evaluation
R Thirumurugan et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2006)
Discovery and structure-activity relationship of 3-aryl-5-aryl-1,2,4-oxadiazoles as a new series of apoptosis inducers and potential anticancer agents
HZ Zhang et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
Biomarkers for prediction of sensitivity to EGFR inhibitors in non-small cell lung cancer
FR Hirsch et al.
CURRENT OPINION IN ONCOLOGY (2005)
Epothilone B and its Analogs - A New Family of Anticancer Agents
Karl-Heinz Altmann
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2003)
PDBsum: summaries and analyses of PDB structures
RA Laskowski
NUCLEIC ACIDS RESEARCH (2001)
分享论文
