相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Design, Synthesis, and Biological Evaluation of Newer Arylidene Incorporated 4-Thiazolidinones Derivatives as Potential Antimicrobial Agents
Pravin S. Kulkarni et al.
POLYCYCLIC AROMATIC COMPOUNDS (2022)
Design, Synthesis, and Antimicrobial Activities of 1,2,3-Triazole Glycoside Clickamers
Tamer El Malah et al.
MOLECULES (2020)
Synthesis, Biological Activity, and Molecular Modeling Studies of Pyrazole and Triazole Derivatives as Selective COX-2 Inhibitors
Mohyeddin Assali et al.
JOURNAL OF CHEMISTRY (2020)
Pyridine- and Thiazole-Based Hydrazides with Promising Anti-inflammatory and Antimicrobial Activities along with Their In Silico Studies
Vinuta Kamat et al.
ACS OMEGA (2020)
Design, synthesis, modeling studies and biological evaluation of thiazolidine derivatives containing pyrazole core as potential anti-diabetic PPAR-γ agonists and anti-inflammatory COX-2 selective inhibitors
Khaled R. A. Abdellatif et al.
BIOORGANIC CHEMISTRY (2019)
Design and synthesis of novel xanthone-triazole derivatives as potential antidiabetic agents: α-Glucosidase inhibition and glucose uptake promotion
Gao-Jie Ye et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
New Series of Thiazole Derivatives: Synthesis, Structural Elucidation, Antimicrobial Activity, Molecular Modeling and MOE Docking
Ismail Althagafi et al.
MOLECULES (2019)
Novel Thiazolidin-4-ones as Potential Non-Nucleoside Inhibitors of HIV-1 Reverse Transcriptase
Anthi Petrou et al.
MOLECULES (2019)
1,2,3-Triazole-containing hybrids as potential anticancer agents: Current developments, action mechanisms and structure-activity relationships
Zhi Xu et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
1,2-Annulated Adamantane Heterocyclic Derivatives as Anti-Influenza A Virus Agents
Vasiliki Pardali et al.
CROATICA CHEMICA ACTA (2019)
Molecular mechanisms underlying prostaglandin E2-exacerbated inflammation and immune diseases
Kyoshiro Tsuge et al.
INTERNATIONAL IMMUNOLOGY (2019)
Synthesis, antibacterial activity and molecular docking study of vanillin derived 1,4-disubstituted 1,2,3-triazoles as inhibitors of bacterial DNA synthesis
Mumtaz Hussain et al.
HELIYON (2019)
Microwave-assisted synthesis, antioxidant and antimicrobial evaluation of 2-indolinone-based bis-1,2,3-triazole derivatives
Dongamanti Ashok et al.
MOLECULAR DIVERSITY (2018)
Design, synthesis and biological evaluation of novel pyridine-thiazolidinone derivatives as anticancer agents: Targeting human carbonic anhydrase IX
Mohammad Fawad Ansari et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
[1,3]Thiazolo[3,2-b][1,2,4]triazol-7-ium salts: synthesis, properties and structural studies
Mikhailo Slivka et al.
HETEROCYCLIC COMMUNICATIONS (2018)
Novel anti-inflammatory and analgesic agents: synthesis, molecular docking and in vivo studies
David Izuchukwu Ugwu et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2018)
Docking assisted design of novel 4-adamantanyl-2-thiazolylimino-5-arylidene-4-thiazolidinones as potent NSAIDs
O. Kouatly et al.
SAR AND QSAR IN ENVIRONMENTAL RESEARCH (2018)
Design, synthesis and biological evaluation of new substituted 5-benzylideno-2-adamantylthiazol[3,2-b][1,2,4]triazol-6(5H)ones. Pharmacophore models for antifungal activity
C. Tratrat et al.
ARABIAN JOURNAL OF CHEMISTRY (2018)
Synthesis of a Series of Substituted Thiazole Derivatives: New COX-2 Enzyme Inhibitors for Colon Cancer and Inflammation Treatment
Reham F. Barghash et al.
CHEMISTRYSELECT (2018)
Effects of NSAIDs on the Release of Calcitonin Gene-Related Peptide and Prostaglandin E-2 from Rat Trigeminal Ganglia
Vittorio Vellani et al.
MEDIATORS OF INFLAMMATION (2017)
Synthesis of 2-phenylamino-thiazole derivatives as antimicrobial agents
Dominique Serge Ngono Bikobo et al.
JOURNAL OF SAUDI CHEMICAL SOCIETY (2017)
Anti-inflammatory and Anti-ulcer Activities of New Fused Thiazole Derivatives Derived from 2-(2-Oxo-2H-chromen-3-yl) thiazol-4(5H)-one
Rafat M. Mohareb et al.
ACTA CHIMICA SLOVENICA (2017)
Study of novel anticancer 4-thiazolidinone derivatives
Konrad A. Szychowski et al.
CHEMICO-BIOLOGICAL INTERACTIONS (2017)
Synthesis and in silico investigation of thiazoles bearing pyrazoles derivatives as anti-inflammatory agents
Rahul D. Kamble et al.
COMPUTATIONAL BIOLOGY AND CHEMISTRY (2016)
Molecular modeling and synthesis of some new 2-imino-4-thiazolidinone derivatives with promising TNF-α inhibitory activity
Yakub Ali et al.
NEW JOURNAL OF CHEMISTRY (2016)
Novel 4-Thiazolidinone Derivatives as Anti-Infective Agents: Synthesis, Characterization, and Antimicrobial Evaluation
Amit Gupta et al.
BIOCHEMISTRY RESEARCH INTERNATIONAL (2016)
Novel thiazolo[3,2-b]-1,2,4-triazoles derived from naproxen with analgesic/anti-inflammatory properties: Synthesis, biological evaluation and molecular modeling studies
Deniz Sarigol et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2015)
Synthesis and biological evaluation of phenyl-1H-1,2,3-triazole derivatives as anti-inflammatory agents
Tae Woo Kim et al.
BIOORGANIC CHEMISTRY (2015)
Novel tetrahydropyrimidine-adamantane hybrids as anti-inflammatory agents: synthesis, structure and biological evaluation
Utpalparna Kalita et al.
MEDICINAL CHEMISTRY RESEARCH (2015)
Prediction of enzyme inhibition and mode of inhibitory action based on calculation of distances between hydrogen bond donor/acceptor groups of the molecule and docking analysis: An application on the discovery of novel effective PTP1B inhibitors
P. Eleftheriou et al.
SAR AND QSAR IN ENVIRONMENTAL RESEARCH (2015)
New small-molecule drug design strategies for fighting resistant influenza A
Zuyuan Shen et al.
ACTA PHARMACEUTICA SINICA B (2015)
TACHYKININS AND THEIR RECEPTORS: CONTRIBUTIONS TO PHYSIOLOGICAL CONTROL AND THE MECHANISMS OF DISEASE
Martin S. Steinhoff et al.
PHYSIOLOGICAL REVIEWS (2014)
Synthesis and biological evaluation of some 5-arylidene-2-(1,3-thiazol-2-ylimino)-1,3-thiazolidin-4-ones as dual anti-inflammatory/antimicrobial agents
I. Apostolidis et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2013)
Synthesis and HIV-1 RT inhibitory action of novel (4/6-substituted benzo[d]thiazol-2-yl)thiazolidin-4-ones. Divergence from the non-competitive inhibition mechanism
Eleni Pitta et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2013)
Inflammation 2010: New Adventures of an Old Flame
Ruslan Medzhitov
CELL (2010)
Novel Thiazolidinone Derivatives with an Uncommon Mechanism of Inhibition Towards HIV-1 Reverse Transcriptase
Eleni Pitta et al.
LETTERS IN DRUG DESIGN & DISCOVERY (2010)
Synthesis and anti-HIV studies of 2-and 3-adamantyl-substituted thiazolidin-4-ones
Jan Balzarini et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2009)
Evaluation of the local anaesthetic activity of 3-aminobenzo[d]isothiazole derivatives using the rat sciatic nerve model
Athina Geronikaki et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2009)
AutoDock4 and AutoDockTools4: Automated Docking with Selective Receptor Flexibility
Garrett M. Morris et al.
JOURNAL OF COMPUTATIONAL CHEMISTRY (2009)
Computer-aided discovery of anti-inflammatory thiazolidinones with dual cyclooxygenase/lipoxygenase inhibition
Athina A. Geronikaki et al.
JOURNAL OF MEDICINAL CHEMISTRY (2008)
Analgesic, antiinflammatory, and ulcerogenic studies of meloxicam solid dispersion prepared with polyethylene glycol 6000
S. G. Vijaya Kumar et al.
METHODS AND FINDINGS IN EXPERIMENTAL AND CLINICAL PHARMACOLOGY (2006)
A novel mechanism of cyclooxygenase-2 inhibition involving interactions with Ser-530 and Tyr-385
SW Rowlinson et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
Prediction of biological activity spectra for substances: Evaluation on the diverse sets of drug-like structures
A Stepanchikova et al.
CURRENT MEDICINAL CHEMISTRY (2003)
Advances in atypical antipsychotics for the treatment of schizophrenia - New formulations and new agents
JP Kelleher et al.
CNS DRUGS (2002)
Structural analysis of NSAID binding by prostaglandin H2 synthase:: Time-dependent and time-independent inhibitors elicit identical enzyme conformations
BS Selinsky et al.
BIOCHEMISTRY (2001)
Interactions between leukotrienes and other inflammatory mediators/modulators in the microvasculature
P Hedqvist et al.
AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE (2000)