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NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY (2015)
Copper-Catalyzed Oxidative C(sp3)-H Functionalization for Facile Synthesis of 1,2,4-Triazoles and 1,3,5-Triazines from Amidines
Huawen Huang et al.
ORGANIC LETTERS (2015)
One-Pot Synthesis of 3,4,5-Trisubstituted 1,2,4-Triazoles via the Addition of Hydrazides to Activated Secondary Amides
William S. Bechara et al.
ORGANIC LETTERS (2015)
Glycogen synthase kinase-3 (GSK3): Regulation, actions, and diseases
Eleonore Beurel et al.
PHARMACOLOGY & THERAPEUTICS (2015)
Microwave-Assisted Catalyst-Free Synthesis of Substituted 1,2,4-Triazoles
Ganesh M. Shelke et al.
SYNLETT (2015)
Divergent and concise total syntheses of dihydrochalcones and 5-deoxyflavones recently isolated from Tacca species and Mimosa diplotricha
Tze Han Sum et al.
TETRAHEDRON (2015)
Organogelators based on iodo 1,2,3-triazole functionalized with coumarin: properties and gelator-solvent interaction
Yaodong Huang et al.
TETRAHEDRON (2015)
FDA-approved small-molecule kinase inhibitors
Peng Wu et al.
TRENDS IN PHARMACOLOGICAL SCIENCES (2015)
Design, synthesis and antifungal activity of novel paeonol derivatives linked with 1,2,3-triazole moiety by the click reaction
Yuqin Jiang et al.
JOURNAL OF CHEMICAL RESEARCH (2015)
Investigational drugs for visceral leishmaniasis
Shyam Sundar et al.
EXPERT OPINION ON INVESTIGATIONAL DRUGS (2015)
The Discovery of Polo-Like Kinase 4 Inhibitors: Design and Optimization of Spiro[cyclopropane-1,3′[3H]indol]-2′(1′H)-ones as Orally Bioavailable Antitumor Agents
Peter B. Sampson et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
On the investigation of hybrid quinones: synthesis, electrochemical studies and evaluation of trypanocidal activity
Guilherme A. M. Jardim et al.
RSC ADVANCES (2015)
In Vitro and In Vivo Efficacy of Novel Flavonoid Dimers against Cutaneous Leishmaniasis
Iris L. K. Wong et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2014)
1,2,3-Triazole-, arylamino- and thio-substituted 1,4-naphthoquinones: Potent antitumor activity, electrochemical aspects, and bioisosteric replacement of C-ring-modified lapachones
Eduardo H. G. da Cruz et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2014)
Synthesis, cytotoxicity, antimicrobial and anti-biofilm activities of novel pyrazolo[3,4-b]pyridine and pyrimidine functionalized 1,2,3-triazole derivatives
P. Nagender et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Synthesis and biological evaluation of novel isoxazoles and triazoles linked 6-hydroxycoumarin as potent cytotoxic agents
Shakeel-u-Rehman et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Anti-cancer activity of carbamate derivatives of melampomagnolide B
Venumadhav Janganati et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Design and synthesis of novel 2H-chromen-2-one derivatives bearing 1,2,3-triazole moiety as lead antimicrobials
Khushbu Kushwaha et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Heck products of parthenolide and melampomagnolide-B as anticancer modulators that modify cell cycle progression
Narsimha R. Penthala et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Sequential synthesis of amino-1,4-naphthoquinone-appended triazoles and triazole-chromene hybrids and their antimycobacterial evaluation
Balasubramanian Devi Bala et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
7-Chloroquinolinotriazoles: Synthesis by the azide-alkyne cycloaddition click chemistry, antimalarial activity, cytotoxicity and SAR studies
Guilherme R. Pereira et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Development of quinone analogues as dynamin GTPase inhibitors
Kylie A. MacGregor et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Synthesis, biological evaluation and molecular docking of novel chalcone-coumarin hybrids as anticancer and antimalarial agents
Ratchanok Pingaew et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Access to a new class of biologically active quinoline based 1,2,4-triazoles
Rahul V. Patel et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Novel benzopsoralen analogues: Synthesis, biological activity and molecular docking studies
Carla S. Francisco et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Synthesis and evaluation of the cytotoxic activity of 1,2-furanonaphthoquinones tethered to 1,2,3-1H-triazoles in myeloid and lymphoid leukemia cell lines
Mariana F. C. Cardoso et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Synthesis and preliminary biological evaluation of 1,2,3-triazole-Jaspine B hybrids as potential cytotoxic agents
Jin-Mei Xu et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Design, economical synthesis and antiplasmodial evaluation of vanillin derived allylated chalcones and their marked synergism with artemisinin against chloroquine resistant strains of Plasmodium falciparum
Nandini Sharma et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Antibacterial Inhibitors of Gram-Positive Thymidylate Kinase: Structure-Activity Relationships and Chiral Preference of a New Hydrophobic Binding Region
Sameer P. Kawatkar et al.
JOURNAL OF MEDICINAL CHEMISTRY (2014)
Nature of Electrogenerated Intermediates in Nitro-Substituted Nor-β-lapachones: The Structure of Radical Species during Successive Electron Transfer in Multiredox Centers
Georgina Armendariz-Vidales et al.
JOURNAL OF ORGANIC CHEMISTRY (2014)
IN VIVO ANTILEISHMANIAL EFFICACY OF MILTEFOSINE AGAINST LEISHMANIA (LEISHMANIA) AMAZONENSIS
Maria F. Garcia Bustos et al.
JOURNAL OF PARASITOLOGY (2014)
Eugenol enhances the resistance of tomato against tomato yellow leaf curl virus
Chunmei Wang et al.
JOURNAL OF THE SCIENCE OF FOOD AND AGRICULTURE (2014)
Chemo-Enzymatic Synthesis of Silybin and 2,3-Dehydrosilybin Dimers
Eva Vavrikova et al.
MOLECULES (2014)
Synthesis and anticancer activity evaluation of new 1,2,3-triazole-4-carboxamide derivatives
Nazariy Pokhodylo et al.
MEDICINAL CHEMISTRY RESEARCH (2014)
Rare biscoumarin derivatives and flavonoids from Hypericum riparium
Serge Alain Fobofou Tanemossu et al.
PHYTOCHEMISTRY (2014)
The Natural Antimicrobial Carvacrol Inhibits Quorum Sensing in Chromobacterium violaceum and Reduces Bacterial Biofilm Formation at Sub-Lethal Concentrations
Sara A. Burt et al.
PLOS ONE (2014)
Tetrabutyl ammonium bromide-mediated benzylation of phenols in water under mild condition
Hailei Wang et al.
TETRAHEDRON (2014)
Total synthesis of agomelatine via Friedel-Crafts acylation followed by Willgerodt-Kindler reaction
Satish Kumar Vujjini et al.
TETRAHEDRON LETTERS (2014)
In Vitro Phytochemical, Antibacterial, and Antifungal Activities of Leaf, Stem, and Root Extracts of Adiantum capillus veneris
Muhammad Saqib Ishaq et al.
SCIENTIFIC WORLD JOURNAL (2014)
Synthesis and anticancer activity evaluation of resveratrol-chalcone conjugates
Deepak Kumar et al.
MEDCHEMCOMM (2014)
Structural modification of berberine alkaloid and their hypoglycemic activity
Yangping Ding et al.
JOURNAL OF FUNCTIONAL FOODS (2014)
Phytochemical Evaluation, Antimicrobial Activity, and Determination of Bioactive Components from Leaves of Aegle marmelos
Farina Mujeeb et al.
BIOMED RESEARCH INTERNATIONAL (2014)
Synthesis of novel psoralen analogues and their in vitro antitumor activity
Carla S. Francisco et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2013)
Synthesis and anti-Trypanosoma cruzi activity of naphthoquinone-containing triazoles: Electrochemical studies on the effects of the quinoidal moiety
Emilay B. T. Diogo et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2013)
Synthesis, antimalarial activity and cytotoxic potential of new monocarbonyl analogues of curcumin
Sunny Manohar et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)
Microtubule Affinity-Regulating Kinase 4: Structure, Function, and Regulation
Farha Naz et al.
CELL BIOCHEMISTRY AND BIOPHYSICS (2013)
Parthenolide: from plant shoots to cancer roots
Akram Ghantous et al.
DRUG DISCOVERY TODAY (2013)
Afatinib: First Global Approval
Rosselle T. Dungo et al.
DRUGS (2013)
β-Ionone derived chalcones as potent antiproliferative agents
Vishal Sharma et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Synthesis of quinoidal molecules: Strategies towards bioactive compounds with an emphasis on lapachones
Solange L. de Castro et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Multifunctional tacrine flavonoid hybrids with cholinergic, β-amyloid-reducing, and metal chelating properties for the treatment of Alzheimer's disease
Su-Yi Li et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Acetylcholinesterase inhibitors as Alzheimer therapy: From nerve toxins to neuroprotection
Manjinder Singh et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Design, synthesis and antiproliferative activity studies of novel 1,2,3-triazole-dithiocarbamate-urea hybrids
Ying-Chao Duan et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Potent naphthoquinones against antimony-sensitive and -resistant Leishmania parasites: Synthesis of novel α- and nor-α-lapachone-based 1,2,3-triazoles by copper-catalyzed azide-alkyne cycloaddition
Tiago T. Guimaraes et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Recent development on naphthoquinone derivatives and their therapeutic applications as anticancer agents
Vishnu Kumar Tandon et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2013)
The apoptotic effect of hesperetin on human cervical cancer cells is mediated through cell cycle arrest, death receptor, and mitochondrial pathways
Ali A. Alshatwi et al.
FUNDAMENTAL & CLINICAL PHARMACOLOGY (2013)
Sesquiterpenoids Lactones: Benefits to Plants and People
Martin Chadwick et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2013)
Targeting Aberrant Glutathione Metabolism to Eradicate Human Acute Myelogenous Leukemia Cells
Shanshan Pei et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2013)
Pyranoflavones: A Group of Small-Molecule Probes for Exploring the Active Site Cavities of Cytochrome P450 Enzymes 1A1, 1A2, and 1B1
Jiawang Liu et al.
JOURNAL OF MEDICINAL CHEMISTRY (2013)
Synthesis and Phytotoxic Activity of 1,2,3-Triazole Derivatives
Thiago F. Borgati et al.
JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY (2013)
Synthesis of Novel Isatin-Type 5'-(4-Alkyl/Aryl-1H-1,2,3-triazoles) via 1,3-Dipolar Cycloaddition Reactions
Bianca N. M. Silva et al.
JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY (2013)
Synthesis of 1H-1,2,3-triazoles and Study of their Antifungal and Cytotoxicity Activities
Iara da Silva et al.
Medicinal Chemistry (2013)
Metal-Catalyzed Cascade Rearrangements of 3-Alkynyl Flavone Ethers
Yuan Xiong et al.
ORGANIC LETTERS (2013)
The Antifungal Eugenol Perturbs Dual Aromatic and Branched-Chain Amino Acid Permeases in the Cytoplasmic Membrane of Yeast
Emad Darvishi et al.
PLOS ONE (2013)
Synthesis and Cytotoxicity of Chalcones and 5-Deoxyflavonoids
Jing Zhang et al.
SCIENTIFIC WORLD JOURNAL (2013)
Cellular and molecular mechanisms activating the cell death processes by chalcones: Critical structural effects
Pierre Champelovier et al.
TOXICOLOGY IN VITRO (2013)
Amino-derivatives of the sesquiterpene lactone class of natural products as prodrugs
James R. Woods et al.
MEDCHEMCOMM (2013)
Indole-triazole conjugates are selective inhibitors and inducers of bacterial biofilms
Marine J. Minvielle et al.
MEDCHEMCOMM (2013)
Synthesis, Characterization, and Biological Activity of Novel Schiff and Mannich Bases of 4-Amino-3-(N-phthalimidomethyl)-1,2,4-triazole-5-thione
Uzma Yunus et al.
JOURNAL OF CHEMISTRY (2013)
Inhibition of Dengue virus and West Nile virus proteases by click chemistry-derived benz[d]isothiazol-3(2H)-one derivatives
Kok-Chuan Tiew et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2012)
Cancer Stem Cells: Impact, Heterogeneity, and Uncertainty
Jeffrey A. Magee et al.
CANCER CELL (2012)
Chemical Synthesis of the Cardiotonic Steroid Glycosides and Related Natural Products
Brian Heasley
CHEMISTRY-A EUROPEAN JOURNAL (2012)
Cancer risk and the complexity of the interactions between environmental and host factors: HENVINET interactive diagrams as simple tools for exploring and understanding the scientific evidence
Domenico F. Merlo et al.
ENVIRONMENTAL HEALTH (2012)
1,2,3-Triazole tethered β-lactam-Chalcone bifunctional hybrids: Synthesis and anticancer evaluation
Pardeep Singh et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
On the search for potential anti-Trypanosoma cruzi drugs: Synthesis and biological evaluation of 2-hydroxy-3-methylamino and 1,2,3-triazolic naphthoquinoidal compounds obtained by click chemistry reactions
Eufranio N. da Silva Junior et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Activity of novel quinoxaline-derived chalcones on in vitro glioma cell proliferation
Tania R. Mielcke et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Design, synthesis and anticancer activity of nitric oxide donating/chalcone hybrids
Mai A. E. Mourad et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Synthesis, biological evaluation and molecular docking studies of 3-(triazolyl)coumarin derivatives: Effect on inducible nitric oxide synthase
Helio A. Stefani et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Design, Synthesis, and Structure-Activity Correlations of Novel Dibenzo[b,d]furan, Dibenzo[b,d]thiophene, and N-Methylcarbazole Clubbed 1,2,3-Triazoles as Potent Inhibitors of Mycobacterium tuberculosis
Santhosh Reddy Patpi et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Amine Linked Flavonoid Dimers as Modulators for P-Glycoprotein-Based Multidrug Resistance: Structure-Activity Relationship and Mechanism of Modulation
Kin-Fai Chan et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Guaianolide Sesquiterpene Lactones, a Source To Discover Agents That Selectively Inhibit Acute Myelogenous Leukemia Stern and Progenitor Cells
Quan Zhang et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Silica and zirconia supported olefin metathesis pre-catalysts: Synthesis, catalytic activity and multiple-use in dimethyl carbonate
Adel Keraani et al.
JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL (2012)
Synthesis of N-Substituted Phthalimidoalkyl 1H-1,2,3-Triazoles: a Molecular Diversity Combining Click Chemistry and Ultrasound Irradiation
Moara T. da Silva et al.
JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY (2012)
Synthesis of Chalcones with Anticancer Activities
Suvitha Syam et al.
MOLECULES (2012)
Synthesis of 9-O-glycosyl-berberine derivatives and bioavailability evaluation
Zhu Chen et al.
MEDICINAL CHEMISTRY RESEARCH (2012)
Sterols with antileishmanial activity isolated from the roots of Pentalinon andrieuxii
Li Pan et al.
PHYTOCHEMISTRY (2012)
Investigating Phenotypic Variability in Colletotrichum lindemuthianum Populations
J. M. A. Pinto et al.
PHYTOPATHOLOGY (2012)
Exploring the Versatility of Cycloplatinated Thiosemicarbazones as Antitumor and Antiparasitic Agents
Prinessa Chellan et al.
ORGANOMETALLICS (2012)
Leishmaniasis Worldwide and Global Estimates of Its Incidence
Jorge Alvar et al.
PLOS ONE (2012)
Synthetic diversification of natural products: semi-synthesis and evaluation of triazole jadomycins
Stephanie N. Dupuis et al.
CHEMICAL SCIENCE (2012)
Cholinesterase inhibitors and memantine for symptomatic treatment of dementia
Joanne Rodda et al.
BMJ-BRITISH MEDICAL JOURNAL (2012)
Berberine in type 2 diabetes therapy: a new perspective for an old antidiarrheal drug?
Ming Zhang et al.
ACTA PHARMACEUTICA SINICA B (2012)
Cancer stem cells: an evolving concept
Long V. Nguyen et al.
NATURE REVIEWS CANCER (2012)
Berberine exerts anti-adipogenic activity through up-regulation of C/EBP inhibitors, CHOP and DEC2
Truc P. T. Pham et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2011)
Determining the binding mode and binding affinity constant of tyrosine kinase inhibitor PD153035 to DNA using optical tweezers
Chih-Ming Cheng et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2011)
Geraniol inhibits prostate cancer growth by targeting cell cycle and apoptosis pathways
Su-Hwa Kim et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2011)
Synthesis and anti-HSV-1 activity of new 1,2,3-triazole derivatives
Alessandro K. Jordao et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2011)
Synthesis and in vitro cytotoxic evaluation of N-alkylbromo and N-alkylphthalimido-isatins
Pardeep Singh et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Inhibition of the M. tuberculosis 3β-hydroxysteroid dehydrogenase by azasteroids
Suzanne T. Thomas et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Isatin 1,2,3-triazoles as potent inhibitors against caspase-3
Yang Jiang et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Designing 2-aminoimidazole alkaloids analogs with anti-biofilm activities: Structure-activities relationships of polysubstituted triazoles
D. Linares et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
In vitro efficacy of 7-benzylamino-1-isoquinolinamines against Plasmodium falciparum related to the efficacy of chalcones
Clare E. Gutteridge et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Potent antiprotozoal activity of a novel semi-synthetic berberine derivative
Mark Bahar et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Synthesis and evaluation of a class of new coumarin triazole derivatives as potential antimicrobial agents
Yuan Shi et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Click Chemistry: 1,2,3-Triazoles as Pharmacophores
Sandip G. Agalave et al.
CHEMISTRY-AN ASIAN JOURNAL (2011)
New Insights into Chemistry and Anti-Infective Potential of Triazole Scaffold
R. Kharb et al.
CURRENT MEDICINAL CHEMISTRY (2011)
Pharmacokinetic-pharmacodynamic optimization of triazole antifungal therapy
Russell E. Lewis
CURRENT OPINION IN INFECTIOUS DISEASES (2011)
The novel anti-tumor agents of 4-triazol-1,8-naphthalimides: Synthesis, cytotoxicity, DNA intercalation and photocleavage
Xiaolian Li et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Antifungal activity of natural and enzymatically-modified flavonoids isolated from citrus species
Maria Paula Salas et al.
FOOD CHEMISTRY (2011)
Dietary chalcones with chemopreventive and chemotherapeutic potential
Barbora Orlikova et al.
GENES AND NUTRITION (2011)
Aromatic Small Molecules Remodel Toxic Soluble Oligomers of Amyloid β through Three Independent Pathways
Ali Reza A. Ladiwala et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2011)
Pharmacological significance of triazole scaffold
Rajeev Kharb et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2011)
Structure-Based Discovery of Inhibitors of Microsomal Prostaglandin E2 Synthase-1, 5-Lipoxygenase and 5-Lipoxygenase-Activating Protein: Promising Hits for the Development of New Anti-inflammatory Agents
Rosa De Simone et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Novel 1,2,3-Triazole Derivatives for Use against Mycobacterium tuberculosis H37Rv (ATCC 27294) Strain
Nubia Boechat et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Concise Synthesis of 5-Methoxy-6-hydroxy-2-methyichromone-7-O- and 5-Hydroxy-2-methyichromone-7-O-rutinosides. Investigation of Their Cytotoxic Activities against Several Human Tumor Cell Lines
Baolin Wu et al.
JOURNAL OF ORGANIC CHEMISTRY (2011)
Rapid Synthesis of 1,3,5-Substituted 1,2,4-Triazoles from Carboxylic Acids, Amidines, and Hydrazines
Georgette M. Castanedo et al.
JOURNAL OF ORGANIC CHEMISTRY (2011)
Cancer stem cells: problems for therapy?
Malcolm R. Alison et al.
JOURNAL OF PATHOLOGY (2011)
An Efficient Synthesis of Mono and Bis-1,2,3-triazole AZT Derivatives via Copper(I)-catalyzed Cycloaddition
Jin-Wei Yuan et al.
JOURNAL OF THE CHINESE CHEMICAL SOCIETY (2011)
Berberine Improves Glucose Metabolism in Diabetic Rats by Inhibition of Hepatic Gluconeogenesis
Xuan Xia et al.
PLOS ONE (2011)
A reação "click" na síntese de 1,2,3-triazóis: aspectos químicos e aplicações
Luiza Baptista de Oliveira Freitas et al.
QUIMICA NOVA (2011)
Synthesis and biological evaluation of simple methoxylated chalcones as anticancer, anti-inflammatory and antioxidant agents
Babasaheb P. Bandgar et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2010)
A boronic acid chalcone analog of combretastatin A-4 as a potent anti-proliferation agent
Yali Kong et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2010)
Design, synthesis and in vitro antimalarial evaluation of triazole-linked chalcone and dienone hybrid compounds
Eric M. Guantai et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2010)
Synthesis, antimalarial and antitubercular activity of acetylenic chalcones
Renate H. Hans et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Synthesis and in vitro evaluation of novel coumarin-chalcone hybrids as potential anticancer agents
Koneni V. Sashidhara et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Identification of aryl 2-aminoimidazoles as biofilm inhibitors in Gram-negative bacteria
Cynthia A. Bunders et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
The NF (Nuclear factor)-κB inhibitor parthenolide interacts with histone deacetylase inhibitors to induce MKK7/JNK1-dependent apoptosis in human acute myeloid leukaemia cells
Yun Dai et al.
BRITISH JOURNAL OF HAEMATOLOGY (2010)
Preparation of Cyclonucleosides
Adam Mieczkowski et al.
CHEMICAL REVIEWS (2010)
Copper-catalyzed azide-alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(I) acetylides
Jason E. Hein et al.
CHEMICAL SOCIETY REVIEWS (2010)
What made sesquiterpene lactones reach cancer clinical trials?
Akram Ghantous et al.
DRUG DISCOVERY TODAY (2010)
Synthesis and antimicrobial activity evaluation of new 1,2,4-triazoles and 1,3,4-thiadiazoles bearing imidazo[2,1-b]thiazole moiety
Nuray Ulusoy Guzeldemirci et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
A Graphical Journey of Innovative Organic Architectures That Have Improved Our Lives
Nicholas A. McGrath et al.
JOURNAL OF CHEMICAL EDUCATION (2010)
N-((1-Benzyl-1H-1,2,3-triazol-4-yl)methyl)arylamide as a New Scaffold that Provides Rapid Access to Antimicrotubule Agents: Synthesis and Evaluation of Antiproliferative Activity Against Select Cancer Cell Lines
Jonathan A. Stefely et al.
JOURNAL OF MEDICINAL CHEMISTRY (2010)
Gene Expression Enabling Synthetic Diversification of Natural Products: Chemogenetic Generation of Pacidamycin Analogs
Abhijeet Deb Roy et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2010)
Butein Sensitizes Human Hepatoma Cells to TRAIL-Induced Apoptosis via Extracellular Signal-Regulated Kinase/Sp1-Dependent DR5 Upregulation and NF-KB Inactivation
Dong-Oh Moon et al.
MOLECULAR CANCER THERAPEUTICS (2010)
Steroids: partial synthesis in medicinal chemistry
James R. Hanson
NATURAL PRODUCT REPORTS (2010)
Post-PKS tailoring steps in natural product-producing actinomycetes from the perspective of combinatorial biosynthesis
Carlos Olano et al.
NATURAL PRODUCT REPORTS (2010)
Alzheimer's disease: strategies for disease modification
Martin Citron
NATURE REVIEWS DRUG DISCOVERY (2010)
MECHANISMS OF DISEASE Alzheimer's Disease
Henry W. Querfurth et al.
NEW ENGLAND JOURNAL OF MEDICINE (2010)
Diverse DNA-Cleaving Capacities of the Jadomycins through Precursor-Directed Biosynthesis
Kristal M. Cottreau et al.
ORGANIC LETTERS (2010)
Application of copper(I)-catalysed azide/alkyne cycloaddition (CuAAC) 'click chemistry' in carbohydrate drug and neoglycopolymer synthesis
Valquiria Aragao-Leoneti et al.
TETRAHEDRON (2010)
'Click' chemistry as a tool for the facile synthesis of fullerene glycoconjugate derivatives
Guilherme Rocha Pereira et al.
TETRAHEDRON LETTERS (2010)
Acute Fatal Liver Toxicity under Erlotinib
Sabina Schacher-Kaufmann et al.
CASE REPORTS IN ONCOLOGY (2010)
Copper(I)-Catalyzed Cycloaddition of Organic Azides and 1-Iodoalkynes
Jason E. Hein et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2009)
Antimicrobial Activities of Jadomycin B and Structurally Related Analogues
David L. Jakeman et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2009)
Exploration and synthesis of curcumin analogues with improved structural stability both in vitro and in vivo as cytotoxic agents
Guang Liang et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2009)
Combretastatin-like chalcones as inhibitors of microtubule polymerization. Part 1: Synthesis and biological evaluation of antivascular activity
Sylvie Ducki et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2009)
Natural and synthetic 2′-hydroxy-chalcones and aurones: Synthesis, characterization and evaluation of the antioxidant and soybean lipoxygenase inhibitory activity
Anastasia Detsi et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2009)
Hybrid α-bromoacryloylamido chalcones. Design, synthesis and biological evaluation
Romeo Romagnoli et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
Synthesis and antifungal activity of 1,2,3-triazole containing fluconazole analogues
Nilkanth G. Aher et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
Cu(I)-Catalyzed Huisgen Azide-Alkyne 1,3-Dipolar Cycloaddition Reaction in Nucleoside, Nucleotide, and Oligonucleotide Chemistry
Franck Amblard et al.
CHEMICAL REVIEWS (2009)
Synthesis and antibacterial activity of novel 5-(4-methyl-1H-1,2,3-triazole) methyl oxazolidinones
Oludotun A. Phillips et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2009)
Novel Flavonoids in Dragon's Blood of Daemonorops draco
Ken-ichi Nakashima et al.
HELVETICA CHIMICA ACTA (2009)
Diosgenin targets Akt-mediated prosurvival signaling in human breast cancer cells
Sowmyalakshmi Srinivasan et al.
INTERNATIONAL JOURNAL OF CANCER (2009)
Antioxidant Activity of the Dihydrochalcones Aspalathin and Nothofagin and Their Corresponding Flavones in Relation to Other Rooibos (Aspalathus linearis) Flavonoids, Epigallocatechin Gallate, and Trolox
Petra W. Snijman et al.
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY (2009)
Facile Synthesis of 1,2,4-Triazoles via a Copper-Catalyzed Tandem Addition-Oxidative Cyclization
Satoshi Ueda et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2009)
Pentavalent Antimonials: New Perspectives for Old Drugs
Frederic Frezard et al.
MOLECULES (2009)
Recent Developments in Anti-Inflammatory Natural Products
Raju Gautam et al.
MEDICINAL RESEARCH REVIEWS (2009)
Inhibition of Acinetobacter baumannii, Staphylococcus aureus and Pseudomonas aeruginosa biofilm formation with a class of TAGE-triazole conjugates
Robert W. Huigens et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2009)
Isolation and characterization of jadomycin L from Streptomyces venezuelae ISP5230 for solid tumor efficacy studies
David L. Jakeman et al.
PURE AND APPLIED CHEMISTRY (2009)
Synthesis of a polyprenyl-type library containing 1,4-disubstituted-1,2,3-triazoles with anti-biofilm activities against Pseudoalteromonas sp.
Annie Praud-Tabaries et al.
TETRAHEDRON LETTERS (2009)
Plant derived antioxidants - Geraniol and camphene protect rat alveolar macrophages against t-BHP induced oxidative stress
M. Tiwari et al.
TOXICOLOGY IN VITRO (2009)
Construction and screening of a 2-aminoimidazole library identifies a small molecule capable of inhibiting and dispersing bacterial biofilms across order, class, and phylum
Steven A. Rogers et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2008)
Natural-Product Sugar Biosynthesis and Enzymatic Glycodiversification
Christopher J. Thibodeaux et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2008)
Nucleosides and oligonucleotides containing 1,2,3-triazole residues with nucleobase tethers: Synthesis via the azide-alkyne 'click' reaction
Padmaja Chittepu et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2008)
Synthesis and SAR studies of biaryloxy-substituted triazoles as antifungal agents
Ping Liu et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)
Synthesis of triazole-oxazolidinones via a one-pot reaction and evaluation of their antimicrobial activity
Jeffrey A. Demaray et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)
Synthesis and anti-bacterial properties of mono-carbonyl analogues of curcumin
Guang Liang et al.
CHEMICAL & PHARMACEUTICAL BULLETIN (2008)
Cu-catalyzed azide-alkyne cycloaddition
Morten Meldal et al.
CHEMICAL REVIEWS (2008)
Synthesis and Antibiofilm Activity of a Second-Generation Reverse-Amide Oroidin Library: A Structure-Activity Relationship Study
T. Eric Ballard et al.
CHEMISTRY-A EUROPEAN JOURNAL (2008)
Luteolin, a Flavonoid with Potential for Cancer Prevention and Therapy
Yong Lin et al.
CURRENT CANCER DRUG TARGETS (2008)
The impact of enzyme engineering upon natural product glycodiversification
Gavin J. Williams et al.
CURRENT OPINION IN CHEMICAL BIOLOGY (2008)
Berberine and its more biologically available derivative, dihydroberberine, inhibit mitochondrial respiratory complex I: A mechanism for the action of berberine to activate AMP-Activated protein kinase and improve insulin action
Nigel Turner et al.
DIABETES (2008)
Naphthoquinoidal [1,2,3]-triazole, a new structural moiety active against Trypanosoma cruzi
Eufranio N. da Silva et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2008)
Biological effects of essential oils - A review
F. Bakkali et al.
FOOD AND CHEMICAL TOXICOLOGY (2008)
Design, Synthesis and antiHIV activity of Novel Isatine-Sulphonamides
P. Selvam et al.
INDIAN JOURNAL OF PHARMACEUTICAL SCIENCES (2008)
A Copper(I)-Catalyzed 1,2,3-Triazole Azide-Alkyne Click Compound Is a Potent Inhibitor of a Multidrug-Resistant HIV-1 Protease Variant
Michael J. Giffin et al.
JOURNAL OF MEDICINAL CHEMISTRY (2008)
Synthesis, thermal stabilities, and anisotropic properties of some new isoflavone-based esters 7-decanoyloxy-3-(4'-substitutedphenyl)-4H-1-benzopyran-4-ones
Guan-Yeow Yeap et al.
LIQUID CRYSTALS (2008)
Mutasynthesis, chemobiosynthesis, and back to semi-synthesis: combining synthetic chemistry and biosynthetic engineering for diversifying natural products
Jonathan Kennedy
NATURAL PRODUCT REPORTS (2008)
Natural products to drugs: natural product-derived compounds in clinical trials
Mark S. Butler
NATURAL PRODUCT REPORTS (2008)
Inner reorganization during the radical-biradical transition in a nor-β-lapachone derivative possessing two redox centers
Dulce Maria Hernandez et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2008)
An evaluation of the effects of gatifloxacin on glucose homeostasis
Ahunna J. Onyenwenyi et al.
PHARMACY WORLD & SCIENCE (2008)
Malaria: Historical aspects and chemoterapy
Tanos C. C. Franca et al.
QUIMICA NOVA (2008)
An orally bioavailable parthenolide analog selectively eradicates acute myelogenous leukemia stem and progenitor cells
Monica L. Guzman et al.
BLOOD (2007)
Synthesis of furo[2,3-b]pyrazine nucleoside analogues with 1,2,3-triazole linkage
Denis S. Ermolat'ev et al.
QSAR & COMBINATORIAL SCIENCE (2007)
The influence of drug-like concepts on decision-making in medicinal chemistry
Paul D. Leeson et al.
NATURE REVIEWS DRUG DISCOVERY (2007)
Diosgenin, a naturally occurring furostanol saponin suppresses 3-hydroxy-3-methylglutaryl CoA reductase expression and induces apoptosis in HCT-116 human colon carcinoma cells
Jayadev Raju et al.
CANCER LETTERS (2007)
Sesquiterpene compounds from Inula viscosa
Gianfranco Fontana et al.
NATURAL PRODUCT RESEARCH (2007)
Stereochemical integrity of oxazolone ring-containing jadomycins
Charles N. Borissow et al.
CHEMBIOCHEM (2007)
Sesquiterpene lactone parthenolide suppresses tumor growth in a xenograft model of renal cell carcinoma by inhibiting the activation of NF-κB
Daizo Oka et al.
INTERNATIONAL JOURNAL OF CANCER (2007)
Synthesis of novel steroidal heterocyclic derivatives as antibacterial agents
Mervat M. Abdelhalim et al.
STEROIDS (2007)
Sterol biosynthesis inhibitors: Potential for transition state analogs and mechanism-based Inactivators targeted at sterol methyltransferase
Zhihong Song et al.
LIPIDS (2007)
Quaternary protoberberine alkaloids
Lenka Grycova et al.
PHYTOCHEMISTRY (2007)
Total synthesis approaches to natural product derivatives based on the combination of chemical synthesis and metabolic engineering
Andreas Kirschning et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2007)
The Dioscorea genus: a review of bioactive steroid saponins
Marc Sautour et al.
JOURNAL OF NATURAL MEDICINES (2007)
Multi-component syntheses of heterocycles by transition-metal catalysis
Daniel M. D'Souza et al.
CHEMICAL SOCIETY REVIEWS (2007)
Adipocyte differentiation from the inside out
Evan D. Rosen et al.
NATURE REVIEWS MOLECULAR CELL BIOLOGY (2006)
Culture conditions improving the production of jadomycin B
David L. Jakeman et al.
JOURNAL OF INDUSTRIAL MICROBIOLOGY & BIOTECHNOLOGY (2006)
Antioxidant and neuroprotective effects of hesperidin and its aglycone hesperetin
Jungsook Cho
ARCHIVES OF PHARMACAL RESEARCH (2006)
1.2.3-triazolic heterocycles: History, preparations, applications and pharmacological activities.
Julio O. F. Melo et al.
QUIMICA NOVA (2006)
Structure-based optimization of azole antifungal agents by CoMFA, CoMSIA, and molecular docking
CQ Sheng et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Synthesis and biological activity of (+)-hedychilactone A and its analogs from (+)-sclareolide
S Oh et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2006)
Synthesis and antihyperglycemic evaluation of various protoberberine derivatives
XL Bian et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2006)
Cu-I-catalyzed alkyne-azide click cycloadditions from a mechanistic and synthetic perspective
VD Bock et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2006)
Inhibitors of HIV-1 protease by using in situ click chemistry
M Whiting et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2006)
Antileishmanial activity of Eugenol-rich essential oil from Ocimum gratissimum
Tania Ueda-Nakamura et al.
PARASITOLOGY INTERNATIONAL (2006)
New 1,2,3,4-tetrahydro-1-aza-anthraquinones and 2-aminoalkyl compounds from norlapachol with molluscicidal activity
TP Barbosa et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2005)
Apoptosis: a basic biological phenomenon with wide-ranging implications in human disease
B Fadeel et al.
JOURNAL OF INTERNAL MEDICINE (2005)
4-Aryl-1,2,3-triazole: A novel template for a reversible methionine aminopeptidase 2 inhibitor, optimized to inhibit angiogenesis in vivo
LS Kallander et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
FDA drug approval summary:: Erlotinib (Tarceva®) tablets
MH Cohen et al.
ONCOLOGIST (2005)
Cytotoxic activities of new jadomycin derivatives
JT Zheng et al.
JOURNAL OF ANTIBIOTICS (2005)
The sesquiterpene lactone parthenolide induces apoptosis of human acute myelogenous leukemia stem and progenitor cells
ML Guzman et al.
BLOOD (2005)
A highly enantio- and diastereoselective catalytic intramolecular stetter reaction
JR de Alaniz et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2005)
Aromatase inhibitors in the treatment of breast cancer
RW Brueggemeier et al.
ENDOCRINE REVIEWS (2005)
The final catalytic step of cytochrome P450 aromatase: A density functional theory study
JC Hackett et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2005)
Molecular chameleons. Design and synthesis of a second series of flexible nucleosides
KL Seley et al.
JOURNAL OF ORGANIC CHEMISTRY (2005)
Dietary polyphenols and the prevention of diseases
A Scalbert et al.
CRITICAL REVIEWS IN FOOD SCIENCE AND NUTRITION (2005)
Copper(I)-catalyzed synthesis of azoles. DFT study predicts unprecedented reactivity and intermediates
F Himo et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2005)
Molecular mechanisms of drug resistance
DB Longley et al.
JOURNAL OF PATHOLOGY (2005)
Treatment of infections caused by metronidazole-resistant Trichomonas vaginalis
SL Cudmore et al.
CLINICAL MICROBIOLOGY REVIEWS (2004)
Leishmaniasis: drugs in the clinic, resistance and new developments
M Ouellette et al.
DRUG RESISTANCE UPDATES (2004)
Privileged structures: Applications in drug discovery
RW DeSimone et al.
COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING (2004)
Heterocyclic peptide backbone modifications in an α-helical coiled coil
WS Horne et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2004)
Compound library development guided by protein structure similarity clustering and natural product structure
MA Koch et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2004)
A microwave-assisted click chemistry synthesis of 1,4-disubstituted 1,2,3-triazoles via a copper(I)-catalyzed three-component reaction
P Appukkuttan et al.
ORGANIC LETTERS (2004)
Selective anti-Toxoplasma gondii activities of azasterols
L Dantas-Leite et al.
INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS (2004)
Large-scale synthesis of the anti-cancer marine natural product (+)-discodermolide. Part 1: Synthetic strategy and preparation of a common precursor
SJ Mickel et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2004)
The growing impact of click chemistry on drug discovery
HC Kolb et al.
DRUG DISCOVERY TODAY (2003)
Leishmaniasis - current chemotherapy and recent advances in the search for novel drugs
SL Croft et al.
TRENDS IN PARASITOLOGY (2003)
Azasterols as inhibitors of sterol 24-methyltransferase in leishmania species and Trypanosoma cruzi
F Magaraci et al.
JOURNAL OF MEDICINAL CHEMISTRY (2003)
Potent anti-amyloidogenic and fibril-destabilizing effects of polyphenols in vitro:: implications for the prevention and therapeutics of Alzheimer's disease
K Ono et al.
JOURNAL OF NEUROCHEMISTRY (2003)
Epidermal growth factor receptor (EGFR) as a target in cancer therapy: understanding the role of receptor expression and other molecular determinants that could influence the response to anti-EGFR drugs
F Ciardiello et al.
EUROPEAN JOURNAL OF CANCER (2003)
Synthesis of α-amino γ-butyrolactone derivatives by aziridination of α-ylidene γ-butyrolactones
T Gasperi et al.
TETRAHEDRON LETTERS (2003)
Pharmaceutical profiling in drug discovery
EH Kerns et al.
DRUG DISCOVERY TODAY (2003)
Fatty acid and sterol metabolism: potential antimicrobial targets in apicomplexan and trypanosomatid parasitic protozoa
CW Roberts et al.
MOLECULAR AND BIOCHEMICAL PARASITOLOGY (2003)
FDA drug approval summary: Gefitinib (ZD1839) (Iressa (R)) tablets
MH Cohen et al.
ONCOLOGIST (2003)
Solid-phase synthesis and bioevaluation of lupeol-based libraries as antimalarial agents
T Srinivasan et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2002)
Glutathione catabolism as a signaling mechanism
A Paolicchi et al.
BIOCHEMICAL PHARMACOLOGY (2002)
Peptidotriazoles on solid phase: [1,2,3]-triazoles by regiospecific copper(I)-catalyzed 1,3-dipolar cycloadditions of terminal alkynes to azides
CW Tornoe et al.
JOURNAL OF ORGANIC CHEMISTRY (2002)
NF-κB in cancer:: From innocent bystander to major culprit
M Karin et al.
NATURE REVIEWS CANCER (2002)
Synthesis and anti-inflammatory activity of 1-acylthiosemicarbazides, 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazole-3-thiones
E Palaska et al.
FARMACO (2002)
Chiral amino ether-controlled catalytic enantioselective arylthiol conjugate additions to α,β-unsaturated esters and ketones:: Scope, structural requirements, and mechanistic implications
K Nishimura et al.
JOURNAL OF ORGANIC CHEMISTRY (2002)
Antioxidant activity of anti-inflammatory plant extracts
GR Schinella et al.
LIFE SCIENCES (2002)
Multidrug resistance in cancer: Role of ATP-dependent transporters
MM Gottesman et al.
NATURE REVIEWS CANCER (2002)
Biotransformation reactions of five-membered aromatic heterocyclic rings
DK Dalvie et al.
CHEMICAL RESEARCH IN TOXICOLOGY (2002)
A mechanistic approach to the in vivo anti-inflammatory activity of sesquiterpenoid compounds isolated from Inula viscosa
V Hernández et al.
PLANTA MEDICA (2001)
Synthesis of spiropyrrolidines and spiropyrrolizidines by 1,3-dipolar cycloadditions of azomethine ylides to substituted α-methylene-γ-lactones
J Castulík et al.
TETRAHEDRON (2001)
Potent and selective nonpeptide inhibitors of caspases 3 and 7
D Lee et al.
JOURNAL OF MEDICINAL CHEMISTRY (2001)
Total synthesis of antitumor depsipeptide (-)-doliculide
AK Ghosh et al.
ORGANIC LETTERS (2001)
Synthesis and anti-HIV activity of new modified 1,2,3-triazole acyclonucleosides
HB Lazrek et al.
NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS (2001)
beta-Phenylethylamines and the isoquinoline alkaloids
KW Bentley
NATURAL PRODUCT REPORTS (2001)
Isolation of a novel human gene, MARKL1, homologous to MARK3 and its involvement in hepatocellular carcinogenesis
T Kato et al.
NEOPLASIA (2001)
The endogenous oxindoles 5-hydroxyoxindole and isatin are antiproliferative and proapoptotic
A Cane et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2000)
The influence of natural products upon drug discovery
DJ Newman et al.
NATURAL PRODUCT REPORTS (2000)
Palladium-catalyzed arylation of alpha-methylene-gamma-butyrolactone: 3-benzylfuran-2(5H)-ones vs (Z)-benzylidene-gamma-butyrolactones and their reduction to 3-benzyl-gamma butyrolactones
A Arcadi et al.
ORGANIC LETTERS (2000)
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