4.5 Article

Discovery of novel triazolophthalazine derivatives as DNA intercalators and topoisomerase II inhibitors

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Medicinal

Synthesis, Antiproliferative Effect, and Topoisomerase II Inhibitory Activity of 3-Methyl-2-phenyl-1H-indoles

Nace Zidar et al.

ACS MEDICINAL CHEMISTRY LETTERS (2020)

Article Pharmacology & Pharmacy

Intercalating TOP2 Poisons Attenuate Topoisomerase Action at Higher Concentrations

Mandeep Atwal et al.

MOLECULAR PHARMACOLOGY (2019)

Article Chemistry, Multidisciplinary

Acid-base behaviour and binding to double stranded DNA/RNA of benzo[g]phthalazine-based ligands

E. Carbonell et al.

NEW JOURNAL OF CHEMISTRY (2019)

Article Chemistry, Medicinal

Design, Synthesis, Molecular Docking, and Anticancer Activity of Phthalazine Derivatives as VEGFR-2 Inhibitors

Abdel-Ghany A. El-Helby et al.

ARCHIV DER PHARMAZIE (2017)

Article Chemistry, Medicinal

Identification of new potent phthalazine derivatives with VEGFR-2 and EGFR kinase inhibitory activity

Kamilia M. Amin et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)

Article Chemistry, Medicinal

Design, synthesis and in vitro antitumor activity of novel N-substituted-4-phenyl/benzylphthalazin-1-ones

Wagdy M. Eldehna et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)

Article Chemistry, Medicinal

Synthesis and anticancer activities of novel 1,2,4-triazolo[3,4-a] phthalazine derivatives

Deng-Qi Xue et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)

Article Chemistry, Medicinal

[1,2,4]Triazolo[4,3-a]phthalazines: Inhibitors of Diverse Bromodomains

Oleg Fedorov et al.

JOURNAL OF MEDICINAL CHEMISTRY (2014)

Article Mathematical & Computational Biology

Molecular Docking Studies of Curcumin Natural Derivatives with DNA Topoisomerase I and II-DNA Complexes

Anil Kumar et al.

INTERDISCIPLINARY SCIENCES-COMPUTATIONAL LIFE SCIENCES (2014)

Article Biochemistry & Molecular Biology

On the structural basis and design guidelines for type II topoisomerase-targeting anticancer drugs

Chyuan-Chuan Wu et al.

NUCLEIC ACIDS RESEARCH (2013)

Review Chemistry, Multidisciplinary

Contemporary Challenges in the Design of Topoisomerase II Inhibitors for Cancer Chemotherapy

Christian Bailly

CHEMICAL REVIEWS (2012)

Review Biochemistry & Molecular Biology

DNA Topoisomerases and Their Poisoning by Anticancer and Antibacterial Drugs

Yves Pommier et al.

CHEMISTRY & BIOLOGY (2010)

Review Oncology

Targeting DNA topoisomerase II in cancer chemotherapy

John L. Nitiss

NATURE REVIEWS CANCER (2009)

Review Chemistry, Inorganic & Nuclear

Luminescent biological probes derived from ruthenium(II) estradiol polypyridine complexes

Kenneth Kam-Wing Lo et al.

INORGANIC CHEMISTRY (2008)