期刊
ORGANIC LETTERS
卷 22, 期 21, 页码 8658-8664出版社
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.0c03252
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资金
- JSPS KAKENHI [19K07000]
- Grants-in-Aid for Scientific Research [19K07000] Funding Source: KAKEN
We report the catalytic direct peptide bond formations via dehydrative condensation of beta-hydroxy-alpha-amino acids, affording the serine, threonine, or beta-hydroxyvaline-derived peptides in high to excellent yields with high functional group tolerance, minimum epimerization, and excellent chemoselectivity. The key to the success of these atom-economical transformations is the use of diboronic acid anhydride catalyst for the hydroxy-directed reactions.
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