期刊
JOURNAL OF ORGANIC CHEMISTRY
卷 85, 期 15, 页码 10182-10188出版社
AMER CHEMICAL SOC
DOI: 10.1021/acs.joc.0c00399
关键词
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资金
- National Natural Science Foundation of China [81673288, 81473079]
- Program for Jiangsu Province Innovative Research Team
- Program for Jiangsu Province Innovative Personnel
- Program for Specially Appointed Professor of Jiangsu Province
- Funding of Double First-Rate Discipline Innovation Teams [CPU2018GY05, CPU2018GF05]
A general and efficient method for the synthesis of azabicyclo[4,3,0]nonanone and azabicyclo[5,3,0]clecanone amino acid derivatives was developed with the palladium-catalyzed coupling of intermediates 9 and 10 with BocNH(2) and Boc(2)NH and the following reduction of the C-C double bond by hydrogenation as the key steps. The exploration of the synthesis of C-6-substituted dipeptide mimetics from 9 and 10 using Suzuki coupling as the key reaction has also been performed.
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