期刊
JOURNAL OF ORGANIC CHEMISTRY
卷 85, 期 12, 页码 7772-7780出版社
AMER CHEMICAL SOC
DOI: 10.1021/acs.joc.0c00279
关键词
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资金
- SERB, DST, New Delhi [IFA12-CH-61]
- JNU [217]
- UGC [23/06/2013(i)EU-V]
The aza-Diels-Alder reaction of various alkenes and in situ formed 1-aza-1,3-dienes from the reaction of furan/pyrrole/thiophene and PhINTs for the regioselective synthesis of tetrahydropyridine (THP) derivatives was realized. The reaction was catalyzed by Tp(Me2)Cu as a catalyst under very mild reaction conditions. Structurally different alkenes, along with an alkyne, have been utilized as dienophiles to afford a wide range of different THP derivatives up to 70% yield. The potential application of the envisaged method was also investigated by a gram-scale synthesis.
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