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Suri Babu Madasu et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2012)
Antileishmanial activity of benzocycloalkyl azole oximino ethers: The conformationally constraint analogues of oxiconazole
Aditya Verma et al.
ACTA TROPICA (2011)
Clinical and Molecular Pharmacology of Etomidate
Stuart A. Forman
ANESTHESIOLOGY (2011)
HPV episome levels are potently decreased by pyrrole-imidazole polyamides
Terri G. Edwards et al.
ANTIVIRAL RESEARCH (2011)
An overview of the key routes to the best selling 5-membered ring heterocyclic pharmaceuticals
Marcus Baumann et al.
BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY (2011)
Synthesis and evaluation of novel 2-butyl-4-chloro-1-methylimidazole embedded chalcones and pyrazoles as angiotensin converting enzyme (ACE) inhibitors
Srinivas Kantevari et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2011)
Discovery of novel hepatoselective HMG-CoA reductase inhibitors for treating hypercholesterolemia: A bench-to-bedside case study on tissue selective drug distribution
Jeffrey A. Pfefferkorn et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Substituted imidazole derivatives as novel cardiovascular agents
Vineet Malhotra et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Pharmacophore Design of p38α MAP Kinase Inhibitors with Either 2,4,5-Trisubstituted or 1,2,4,5-Tetrasubstituted Imidazole Scaffold
T. Scior et al.
CURRENT MEDICINAL CHEMISTRY (2011)
mGluR5 Negative Allosteric Modulators Overview: A Medicinal Chemistry Approach Towards a Series of Novel Therapeutic Agents
Jean-Philippe Rocher et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2011)
Inhibition of α-glucosidase and α-amylase by diaryl derivatives of imidazole-thione and 1,2,4-triazole-thiol
Mahmoud Balba et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Synthesis and evaluation of new furanyl and thiophenyl azoles as antileishmanial agents
Vijay K. Marrapu et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Novel 3-hydroxy-3-methylglutaryl-coenzyme A reductase inhibitors: a patent review
Jeffrey A. Pfefferkorn
EXPERT OPINION ON THERAPEUTIC PATENTS (2011)
Urease inhibitors as potential drugs for gastric and urinary tract infections: a patent review
Paulina Kosikowska et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2011)
Recent advances in leishmaniasis treatment
Tatiana S. Tiuman et al.
INTERNATIONAL JOURNAL OF INFECTIOUS DISEASES (2011)
JNK3 as a Therapeutic Target for Neurodegenerative Diseases
Xanthi Antoniou et al.
JOURNAL OF ALZHEIMERS DISEASE (2011)
Synthesis of Angiotensin II Receptor Blockers by Means of a Catalytic System for C-H Activation
Masahiko Seki et al.
JOURNAL OF ORGANIC CHEMISTRY (2011)
Structure and synthesis of 2-aminoimidazole alkaloids from Leucetta and Clathrina sponges
Panduka B. Koswatta et al.
NATURAL PRODUCT REPORTS (2011)
Allosteric modulation of metabotropic glutamate receptors: Structural insights and therapeutic potential
Karen J. Gregory et al.
NEUROPHARMACOLOGY (2011)
Silver-Mediated Palladium-Catalyzed Direct C-H Arylation of 3-Bromoisothiazole-4-carbonitrile
Heraklidia A. Ioannidou et al.
ORGANIC LETTERS (2011)
Indole synthesis: a review and proposed classification
Douglass F. Taber et al.
TETRAHEDRON (2011)
CTEP: A Novel, Potent, Long-Acting, and Orally Bioavailable Metabotropic Glutamate Receptor 5 Inhibitor
Lothar Lindemann et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2011)
Synthesis and anthelmintic activity of some novel 2-substituted-4,5-diphenyl imidazoles
Satyajit Dutta
ACTA PHARMACEUTICA (2010)
Regioselective Functionalization of the Imidazole Ring via Transition Metal-Catalyzed C-N and C-C Bond Forming Reactions
Fabio Bellina et al.
ADVANCED SYNTHESIS & CATALYSIS (2010)
Review article: anti-fibrotic agents for the treatment of Crohn's disease - lessons learnt from other diseases
H. Szabo et al.
ALIMENTARY PHARMACOLOGY & THERAPEUTICS (2010)
Concise and Diversity-Oriented Route toward Polysubstituted 2-Aminoimidazole Alkaloids and Their Analogues
Denis S. Ermolat'ev et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2010)
Adverse effects of non-steroidal anti-inflammatory drugs (NSAIDs, aspirin and coxibs) on upper gastrointestinal tract
Carlos Sostres et al.
BEST PRACTICE & RESEARCH CLINICAL GASTROENTEROLOGY (2010)
Angiotensin II receptor type 1 (AT1) selective nonpeptidic antagonists-A perspective
Prashant Naik et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2010)
Synthesis and SAR of novel imidazoles as potent and selective cannabinoid CB2 receptor antagonists with high binding efficiencies
Jos H. M. Lange et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Synthesis and biological activity of a series of tetrasubstituted-imidazoles as P2X7 antagonists
Robert J. Gleave et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Tri- and tetrasubstituted imidazoles as p38α mitogen-activated protein kinase inhibitors
Stefan Laufer et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Design of a series of bicyclic HIV-1 integrase inhibitors. Part 2: Azoles: Effective metal chelators
Giang Le et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Synthesis and structure-activity relationships of a series of (1H-pyrazol-4-yl)acetamide antagonists of the P2X7 receptor
Laura J. Chambers et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Synthesis of substituted aryloxy alkyl and aryloxy aryl alkyl imidazoles as antileishmanial agents
Kalpana Bhandari et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Use of the GTPγS ([35S]GTPγS and Eu-GTPγS) binding assay for analysis of ligand potency and efficacy at G protein-coupled receptors
Philip G. Strange
BRITISH JOURNAL OF PHARMACOLOGY (2010)
IRTKS suppresses p53 activity through promoting MDM2 mediated p53 monoubiquitination
Xin Zhang et al.
CANCER RESEARCH (2010)
Concise total synthesis of naamine G and naamidine H
Panduka B. Koswatta et al.
CHEMICAL COMMUNICATIONS (2010)
Tacrine Derivatives and Alzheimer's Disease
V. Tumiatti et al.
CURRENT MEDICINAL CHEMISTRY (2010)
Targeted covalent drugs of the kinase family
Juswinder Singh et al.
CURRENT OPINION IN CHEMICAL BIOLOGY (2010)
Synthesis of 2-substituted-N-[4-(1-methyl-4,5-diphenyl-1H-imidazole-2-yl) phenyl]acetamide derivatives and evaluation of their anticancer activity
Yusuf Ozkay et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
Targeting kinases for the treatment of inflammatory diseases
Susanne Mueller et al.
EXPERT OPINION ON DRUG DISCOVERY (2010)
Hydrogen peroxide is the major oxidant product of xanthine oxidase
Eric E. Kelley et al.
FREE RADICAL BIOLOGY AND MEDICINE (2010)
Strategies for discovering and derisking covalent, irreversible enzyme inhibitors
Douglas S. Johnson et al.
FUTURE MEDICINAL CHEMISTRY (2010)
Small Molecule JNK (c-Jun N-Terminal Kinase) Inhibitors
M. Arshad Siddiqui et al.
JOURNAL OF MEDICINAL CHEMISTRY (2010)
New World cutaneous leishmaniasis: Updated review of current and future diagnosis and treatment
Panagiotis Mitropoulos et al.
JOURNAL OF THE AMERICAN ACADEMY OF DERMATOLOGY (2010)
Synthesis of 5-Amino-3-methylimidazolidine-2,4-dione and 1,3,5-Triazine Derivatives as Analogues of the Alkaloids Naamidine A and G
Helen M. Witchard et al.
SYNTHESIS-STUTTGART (2010)
Total syntheses of naamidine G and 14-methoxynaamidine G
Panduka B. Koswatta et al.
TETRAHEDRON LETTERS (2010)
TR-FRET Biochemical Assays for Detecting Posttranslational Modifications of p53
Jeanne M. Dudek et al.
JOURNAL OF BIOMOLECULAR SCREENING (2010)
Synthesis of related substances of olmesartan medoxomil, anti-hypertensive drug
Karrothu Srihari Babu et al.
ARKIVOC (2010)
Methoxycarbonyl-etomidate A Novel Rapidly Metabolized and Ultra-short-acting Etomidate Analogue that Does Not Produce Prolonged Adrenocortical Suppression
Joseph F. Cotten et al.
ANESTHESIOLOGY (2009)
The marine alkaloid naamidine A promotes caspase-dependent apoptosis in tumor cells
Daniel V. LaBarbera et al.
ANTI-CANCER DRUGS (2009)
TGF-β and fibrosis in different organs - molecular pathway imprints
Dirk Pohlers et al.
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR BASIS OF DISEASE (2009)
Synthesis and biological evaluation of imidazole thioacetanilides as novel non-nucleoside HIV-1 reverse transcriptase inhibitors
Peng Zhan et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2009)
Aryloxy cyclohexyl imidazoles: A novel class of antileishmanial agents
Nagarapu Srinivas et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
2-Acylaminopyridin-4-ylimidazoles as p38 MAP Kinase Inhibitors: Design, Synthesis, and Biological and Metabolic Evaluations
Katharina Ziegler et al.
CHEMMEDCHEM (2009)
Cardiovascular Effects of Losartan and Its Relevant Clinical Application
Feichao Xu et al.
CURRENT MEDICINAL CHEMISTRY (2009)
Statins and Cardiovascular Diseases: From Cholesterol Lowering to Pleiotropy
Qian Zhou et al.
CURRENT PHARMACEUTICAL DESIGN (2009)
Nitroimidazolyl-1,3,4-thiadiazole-based anti-leishmanial agents: Synthesis and in vitro biological evaluation
Fatemeh Poorrajab et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2009)
Targeting Liver Fibrosis: Strategies for Development and Validation of Antifibrotic Therapies
Yury Popov et al.
HEPATOLOGY (2009)
The Membrane-Bound Bile Acid Receptor TGR5 Is Localized in the Epithelium of Human Gallbladders
Verena Keitel et al.
HEPATOLOGY (2009)
Post-translational modifications of tubulin in the nervous system
Nobuyuki Fukushima et al.
JOURNAL OF NEUROCHEMISTRY (2009)
Interaction between Helicobacter pylori, diet, and genetic polymorphisms as related to non-cancer diseases
Alberto Izzotti et al.
MUTATION RESEARCH-FUNDAMENTAL AND MOLECULAR MECHANISMS OF MUTAGENESIS (2009)
Nickel-Catalyzed Direct Alkynylation of Azoles with Alkynyl Bromides
Naoto Matsuyama et al.
ORGANIC LETTERS (2009)
Total Synthesis of the Putative Structure of Nagelamide D
Manojkumar R. Bhandari et al.
ORGANIC LETTERS (2009)
Imidazole derivatives and their antitumor activity (review)
M. A. Iradyan et al.
PHARMACEUTICAL CHEMISTRY JOURNAL (2009)
Selective P2X7 receptor antagonists for chronic inflammation and pain
William A. Carroll et al.
PURINERGIC SIGNALLING (2009)
Efficient Synthesis of Olmesartan Medoxomil, an Antihypertensive Drug
Karrothu Srihari Babu et al.
SYNTHETIC COMMUNICATIONS (2009)
Expedient total syntheses of preclathridine A and clathridine A
Panduka B. Koswatta et al.
TETRAHEDRON LETTERS (2009)
Advances in antifibrotic therapy
Zahra Ghiassi-Nejad et al.
Expert Review of Gastroenterology & Hepatology (2009)
Biology and therapeutic potential of cannabinoid CB2 receptor inverse agonists
C. A. Lunn et al.
BRITISH JOURNAL OF PHARMACOLOGY (2008)
Mitogen-activated protein kinases as therapeutic targets in osteoarthritis
Richard F. Loeser et al.
CURRENT OPINION IN RHEUMATOLOGY (2008)
Olmesartan medoxomil - A review of its use in the management of hypertension
Lesley J. Scott et al.
DRUGS (2008)
Synthesis, Spectral and Anthelmintic Activity Studies on Some Novel Imidazole Derivatives
Rajiv Dahiya et al.
E-JOURNAL OF CHEMISTRY (2008)
Regioselective Synthesis of 4,5-Diaryl-1-methyl-1H-imidazoles Including Highly Cytotoxic Derivatives by Pd-Catalyzed Direct C-5 Arylation of 1-Methyl-1H-imidazole with Aryl Bromides
Fabio Bellina et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2008)
The P2X7 receptor as a therapeutic target
Romeo Romagnoli et al.
EXPERT OPINION ON THERAPEUTIC TARGETS (2008)
Thermodynamic and structure guided design of statin based inhibitors of 3-hydroxy-3-methylglutaryl coenzyme a reductase
Ronald W. Sarver et al.
JOURNAL OF MEDICINAL CHEMISTRY (2008)
Design, synthesis, and biological evaluation of novel tri- and tetrasubstituted imidazoles as highly potent and specific ATP-mimetic inhibitors of p38 MAP kinase: Focus on optimized interactions with the enzyme's surface-exposed front region
Stefan A. Laufer et al.
JOURNAL OF MEDICINAL CHEMISTRY (2008)
Preparation of a HMG-CoA Reductase Inhibitor via an Optimized Imidazole-Forming Condensation Reaction
Daniel M. Bowles et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2008)
Convenient access to bis-indole alkaloids.: Application to the synthesis of topsentins
Sajal K. Mal et al.
TETRAHEDRON (2008)
The Role of Leukotriene B4 in Allergic Diseases
Hiroshi Ohnishi et al.
ALLERGOLOGY INTERNATIONAL (2008)
High-throughput screening-based identification of paramyxovirus inhibitors
Jeong-Joong Yoon et al.
JOURNAL OF BIOMOLECULAR SCREENING (2008)
Synthesis and evaluation of new difluoromethyl azoles as antileishmanial agents
Sabrina B. Ferreira et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2007)
Naamidines H and I, cytotoxic imidazole alkaloids from the Indonesian marine sponge Leucetta chagosensis
Sachiko Tsukamoto et al.
JOURNAL OF NATURAL PRODUCTS (2007)
A chemical route to stem cells?
John Bonner
CHEMISTRY WORLD (2007)
Synthetic small molecules that induce neurogenesis in skeletal muscle
Darren R. Williams et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2007)
P38 MAP-Kinases pathway regulation, function and role in human diseases
Ana Cuenda et al.
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR CELL RESEARCH (2007)
Synthesis and biological evaluation of analogues of the anti-tumor alkaloid naamidine A
Nicholas Aberle et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)
Transforming growth factor-β and fibrosis
Franck Verrecchia et al.
WORLD JOURNAL OF GASTROENTEROLOGY (2007)
The cannabinoid CB2 receptor as a target for inflammation-dependent neurodegeneration
John C. Ashton et al.
CURRENT NEUROPHARMACOLOGY (2007)
Synthesis and biological activity of vicinal diaryl-substituted 1H-imidazoles
Fabio Bellina et al.
TETRAHEDRON (2007)
Optimization of imidazole amide derivatives as cannabinoid-1 receptor antagonists for the treatment of obesity
Roger A. Smith et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)
Preparation and Diels-Alder chemistry of 4-vinylimidazoles
Carl J. Lovely et al.
JOURNAL OF ORGANIC CHEMISTRY (2007)
NSAIDs and Alzheimer disease: Epidemiological, animal model and clinical studies
Patrick L. McGeer et al.
NEUROBIOLOGY OF AGING (2007)
Efficient synthesis of 1,5-disubstituted tetrazoles
Alan R. Katritzky et al.
SYNTHESIS-STUTTGART (2007)
Synthesis of 2,4,5-triaryl-imidazoles catalyzed by NiCl2•6H2O under heterogeneous system
Majid M. Heravi et al.
JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL (2007)
Angiotensin II type 1 receptor blockade attenuates TGF-β-induced failure of muscle regeneration in multiple myopathic states
Ronald D. Cohn et al.
NATURE MEDICINE (2007)
Impact of losartan on stroke risk in hypertensive patients in primary care
K. Bestehorn et al.
CLINICAL DRUG INVESTIGATION (2007)
Nitroimidazoies, Part 4:: Synthesis and anti-HIV activity of new 5-alkylsulfanyl and 5-(4′-arylsulfonyl)piperazinyl-4-nitroimidazole derivatives
Yaseen A. Al-Soud et al.
HETEROATOM CHEMISTRY (2007)
Intramolecular amidation: Synthesis of novel thiazole-fused diazepinones
Rajesh S. Koti et al.
SYNTHETIC COMMUNICATIONS (2007)
Recent progress in the catalysis synthesis in imidazoles
Shin Kamijo et al.
CHEMISTRY-AN ASIAN JOURNAL (2007)
p38 pathway kinases as anti-inflammatory drug targets
J. F. Schindler et al.
JOURNAL OF DENTAL RESEARCH (2007)
Direct palladium-catalyzed ortho-arylation of benzylamines
Anna Lazareva et al.
ORGANIC LETTERS (2006)
How the antihypertensive losartan was discovered
Gaurab Bhardwaj
EXPERT OPINION ON DRUG DISCOVERY (2006)
Olmesartan is an angiotensin II receptor blocker with an inhibitory effect on angiotensin-converting enzyme
Jun Agata et al.
HYPERTENSION RESEARCH (2006)
IN-1130, a novel transforming growth factor-β type I receptor kinase (ALK5) inhibitor, suppresses renal fibrosis in obstructive nephropathy
J-A Moon et al.
KIDNEY INTERNATIONAL (2006)
Losartan, an AT1 antagonist, prevents aortic aneurysm in a mouse model of Marfan syndrome
JP Habashi et al.
SCIENCE (2006)
The P2X7 receptor:: A key player in IL-1 processing and release
Davide Ferrari et al.
JOURNAL OF IMMUNOLOGY (2006)
Unmet medical needs in antibacterial therapy
LB Rice
BIOCHEMICAL PHARMACOLOGY (2006)
Design and synthesis of new tetrazolyl- and carboxy-biphenylylmethyl-quinazolin-4-one derivatives as angiotensin II AT1 receptor antagonists
MAH Ismail et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Therapeutic effects of xanthine oxidase inhibitors: Renaissance half a century after the discovery of allopurinol
P Pacher et al.
PHARMACOLOGICAL REVIEWS (2006)
A concise total synthesis of naamidine A
NS Aberle et al.
ORGANIC LETTERS (2006)
Targeting acetylcholinesterase and butyrylcholinesterase in dementia
RM Lane et al.
INTERNATIONAL JOURNAL OF NEUROPSYCHOPHARMACOLOGY (2006)
Prostaglandin E-2 synthesis and secretion: The role of PGE(2) synthases
Jean Y. Park et al.
CLINICAL IMMUNOLOGY (2006)
Drug resistance in leishmaniasis
SL Croft et al.
CLINICAL MICROBIOLOGY REVIEWS (2006)
Adult neurogenesis and neurodegenerative disease
Barbara Steiner et al.
REGENERATIVE MEDICINE (2006)
Febuxostat: a non-purine, selective inhibitor of xanthine oxidase for the management of hyperuricaemia in patients with gout
HR Schumacher
EXPERT OPINION ON INVESTIGATIONAL DRUGS (2005)
Synthesis of 2-(aminocarbonylmethylthio)-1H-imidazoles as novel Capravirine analogues
YM Loksha et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2005)
Inhibition of gene markers of fibrosis with a novel inhibitor of transforming growth factor-β type I receptor kinase in puromycin-induced nephritis
ET Grygielko et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2005)
Chemical synthesis of (S)-4,5-dihydroxy-2,3-pentanedione, a bacterial signal molecule precursor, and validation of its activity in Salmonella typhimurium
SCJ De Keersmaecker et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2005)
Cannabinoid CB1 receptor antagonists as promising new medications for drug dependence
B Le Foll et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2005)
Small molecule inhibitors of p53/MDM2 interaction
N Fotouhi et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2005)
Anilide ortho-arylation by using C-H activation methodology
O Daugulis et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2005)
Mechanisms of caspase-1 activation by P2X7 receptor-mediated K+ release
JM Kahlenberg et al.
AMERICAN JOURNAL OF PHYSIOLOGY-CELL PHYSIOLOGY (2004)
New imidazole alkaloids from the Indonesian sponge Leucetta chagosensis
W Hassan et al.
JOURNAL OF NATURAL PRODUCTS (2004)
Adverse drug reactions to anthelmintics
H Bagheri et al.
ANNALS OF PHARMACOTHERAPY (2004)
Leishmaniasis: current situation and new perspectives
P Desjeux
COMPARATIVE IMMUNOLOGY MICROBIOLOGY AND INFECTIOUS DISEASES (2004)
Tetrasubstituted imidazole inhibitors of cytokine release: Probing substituents in the N-1 position
SA Laufer et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
Targeting JNK3 for the treatment of neurodegenerative disorders
L Resnick et al.
DRUG DISCOVERY TODAY (2004)
The growing impact of click chemistry on drug discovery
HC Kolb et al.
DRUG DISCOVERY TODAY (2003)
p38 map kinases: Key signalling molecules as therapeutic targets for inflammatory diseases
S Kumar et al.
NATURE REVIEWS DRUG DISCOVERY (2003)
An angiotensin II type 1 receptor antagonist, olmesartan medoxomil, improves experimental liver fibrosis by suppression of proliferation and collagen synthesis in activated hepatic stellate cells
N Kurikawa et al.
BRITISH JOURNAL OF PHARMACOLOGY (2003)
Induction of CB2 receptor expression in the rat spinal cord of neuropathic but not inflammatory chronic pain models
J Zhang et al.
EUROPEAN JOURNAL OF NEUROSCIENCE (2003)
N-aminoimidazole derivatives inhibiting retroviral replication via a yet unidentified mode of action
IM Lagoja et al.
JOURNAL OF MEDICINAL CHEMISTRY (2003)
Cholinesterase inhibitors for the treatment of Alzheimer's disease: Getting on and staying on
GT Grossberg
CURRENT THERAPEUTIC RESEARCH-CLINICAL AND EXPERIMENTAL (2003)
A G protein-coupled receptor responsive to bile acids
Y Kawamata et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
The reaction mechanism of xanthine oxidase: Evidence for two-electron chemistry rather than sequential one-electron steps
AL Stockert et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2002)
Purine and pyrimidine (P2) receptors as drug targets
KA Jacobson et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Chemistry and mechanism of urease inhibition
Z Amtul et al.
CURRENT MEDICINAL CHEMISTRY (2002)
Review article: natural history and epidemiology of Helicobacter pylori injection
MF Go
ALIMENTARY PHARMACOLOGY & THERAPEUTICS (2002)
Advances in the treatment of Alzheimer's disease: Benefits of dual cholinesterase inhibition
CG Ballard
EUROPEAN NEUROLOGY (2002)
Renoprotective effects of blockade of angiotensin II AT1 receptors in an animal model of type 2 diabetes
M Mizuno et al.
HYPERTENSION RESEARCH (2002)
Developments in local anaesthetic drugs
JB Whiteside et al.
BRITISH JOURNAL OF ANAESTHESIA (2001)
Comparison of upper gastrointestinal toxicity of rofecoxib and naproxen in patients with rheumatoid arthritis.
C Bombardier et al.
NEW ENGLAND JOURNAL OF MEDICINE (2000)
IC261, a specific inhibitor of the protein kinases casein kinase 1-delta and -epsilon, triggers the mitotic checkpoint and induces p53-dependent postmitotic effects
L Behrend et al.
ONCOGENE (2000)
Gastrointestinal toxicity with celecoxib vs nonsteroidal anti-inflammatory drugs for osteoarthritis and rheumatoid arthritis - The CLASS study: A randomized controlled trial
FE Silverstein et al.
JAMA-JOURNAL OF THE AMERICAN MEDICAL ASSOCIATION (2000)
Inhibition of p38 MAP kinase as a therapeutic strategy
JC Lee et al.
IMMUNOPHARMACOLOGY (2000)
Total syntheses of naamine A and naamidine A, marine imidazole alkaloids
S Ohta et al.
HETEROCYCLES (2000)
Losartan - A review of its use, with special focus on elderly patients
KL Simpson et al.
DRUGS & AGING (2000)
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