4.8 Article

SWI/SNF catalytic subunits' switch drives resistance to EZH2 inhibitors in ARID1A-mutated cells

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Cell Biology

ARID1A-mutated ovarian cancers depend on HDAC6 activity

Benjamin G. Bitler et al.

NATURE CELL BIOLOGY (2017)

Article Multidisciplinary Sciences

PRC2-mediated repression of SMARCA2 predicts EZH2 inhibitor activity in SWI/SNF mutant tumors

Thomas Januario et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2017)

Review Cell Biology

Mammalian SWI/SNF complexes in cancer: emerging therapeutic opportunities

Roodolph St. Pierre et al.

CURRENT OPINION IN GENETICS & DEVELOPMENT (2017)

Article Multidisciplinary Sciences

EZH2 inhibition sensitizes BRG1 and EGFR mutant lung tumours to TopoII inhibitors

Christine M. Fillmore et al.

NATURE (2015)

Article Biochemistry & Molecular Biology

SWI/SNF-mutant cancers depend on catalytic and non-catalytic activity of EZH2

Kimberly H. Kim et al.

NATURE MEDICINE (2015)

Article Biochemistry & Molecular Biology

Synthetic lethality by targeting EZH2 methyltransferase activity in ARID1A-mutated cancers

Benjamin G. Bitler et al.

NATURE MEDICINE (2015)

Article Biochemistry & Molecular Biology

Residual Complexes Containing SMARCA2 (BRM) Underlie the Oncogenic Drive of SMARCA4 (BRG1) Mutation

Boris G. Wilson et al.

MOLECULAR AND CELLULAR BIOLOGY (2014)

Article Multidisciplinary Sciences

Discovery and saturation analysis of cancer genes across 21 tumour types

Michael S. Lawrence et al.

NATURE (2014)

Article Biochemistry & Molecular Biology

ARID1B is a specific vulnerability in ARID1A-mutant cancers

Katherine C. Helming et al.

NATURE MEDICINE (2014)

Article Multidisciplinary Sciences

Functional epigenetics approach identifies BRM/SMARCA2 as a critical synthetic lethal target in BRG1-deficient cancers

Gregory R. Hoffman et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2014)

Article Biochemistry & Molecular Biology

ABT-199, a potent and selective BCL-2 inhibitor, achieves antitumor activity while sparing platelets

Andrew J. Souers et al.

NATURE MEDICINE (2013)

Article Biochemistry & Molecular Biology

Mechanisms of resistance to therapies targeting BRCA-mutant cancers

Christopher J. Lord et al.

NATURE MEDICINE (2013)

Article Multidisciplinary Sciences

EZH2 inhibition as a therapeutic strategy for lymphoma with EZH2-activating mutations

Michael T. McCabe et al.

NATURE (2012)

Article Biochemistry & Molecular Biology

A selective inhibitor of EZH2 blocks H3K27 methylation and kills mutant lymphoma cells

Sarah K. Knutson et al.

NATURE CHEMICAL BIOLOGY (2012)

Article Biochemical Research Methods

Fast gapped-read alignment with Bowtie 2

Ben Langmead et al.

NATURE METHODS (2012)

Article Multidisciplinary Sciences

Selective inhibition of Ezh2 by a small molecule inhibitor blocks tumor cells proliferation

Wei Qi et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2012)

Review Oncology

SWI/SNF nucleosome remodellers and cancer

Boris G. Wilson et al.

NATURE REVIEWS CANCER (2011)

Editorial Material Obstetrics & Gynecology

Researchers find a new cancer gene and a possible link between ovarian cancer and endometriosis

[Anonymous]

WOMENS HEALTH (2010)

Article Medicine, General & Internal

ARID1A Mutations in Endometriosis-Associated Ovarian Carcinomas

Kimberly C. Wiegand et al.

NEW ENGLAND JOURNAL OF MEDICINE (2010)

Article Biochemistry & Molecular Biology

Antagonistic Roles for BRM and BRG1 SWI/SNF Complexes in Differentiation

Stephen Flowers et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2009)

Article Oncology

ABT-263: A potent and orally bioavailable Bcl-2 family inhibitor

Christin Tse et al.

CANCER RESEARCH (2008)

Article Biochemistry & Molecular Biology

Transcriptional specificity of human SWI/SNF BRG1 and BRM chromatin remodeling complexes

S Kadam et al.

MOLECULAR CELL (2003)

Article Multidisciplinary Sciences

Role of histone H3 lysine 27 methylation in polycomb-group silencing

R Cao et al.

SCIENCE (2002)