4.6 Article

Bromodomain Drug Discovery - the Past, the Present, and the Future

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Multidisciplinary

Discovery of a PCAF Bromodomain Chemical Probe

Moses Moustakim et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2017)

Article Chemistry, Medicinal

Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains

Lea Bouche et al.

JOURNAL OF MEDICINAL CHEMISTRY (2017)

Review Microbiology

Bromodomains in Protozoan Parasites: Evolution, Function, and Opportunities for Drug Development

Victoria Jeffers et al.

MICROBIOLOGY AND MOLECULAR BIOLOGY REVIEWS (2017)

Article Biochemistry & Molecular Biology

Structural basis of PROTAC cooperative recognition for selective protein degradation

Morgan S. Gadd et al.

NATURE CHEMICAL BIOLOGY (2017)

Article Biochemistry & Molecular Biology

Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action

Amaury E. Fernandez-Montalvan et al.

ACS CHEMICAL BIOLOGY (2017)

Article Biochemistry & Molecular Biology

Selective Targeting of Bromodomains of the Bromodomain-PHD Fingers Family Impairs Osteoclast Differentiation

Julia C. Meier et al.

ACS CHEMICAL BIOLOGY (2017)

Article Chemistry, Multidisciplinary

Beyond the BET Family: Targeting CBP/p300 with 4-Acyl Pyrroles

Martin Huegle et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2017)

Article Biochemistry & Molecular Biology

Synthesis and evaluation of novel dual BRD4/HDAC inhibitors

Seika Amemiya et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2017)

Article Chemistry, Medicinal

Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B

Peiling Chen et al.

JOURNAL OF MEDICINAL CHEMISTRY (2016)

Article Oncology

BRD4 Regulates Breast Cancer Dissemination through Jagged1/Notch1 Signaling

Guillaume Andrieu et al.

CANCER RESEARCH (2016)

Article Chemistry, Medicinal

Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor

Laetitia J. Martin et al.

JOURNAL OF MEDICINAL CHEMISTRY (2016)

Article Multidisciplinary Sciences

PROTAC-induced BET protein degradation as a therapy for castration-resistant prostate cancer

Kanak Raina et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2016)

Article Microbiology

A Plasmodium Falciparum Bromodomain Protein Regulates Invasion Gene Expression

Gabrielle A. Josling et al.

CELL HOST & MICROBE (2015)

Article Gastroenterology & Hepatology

ATAD2 Overexpression Identifies Colorectal Cancer Patients with Poor Prognosis and Drives Proliferation of Cancer Cells

Yang Luo et al.

GASTROENTEROLOGY RESEARCH AND PRACTICE (2015)

Article Oncology

BET Bromodomain Inhibition of MYC-Amplified Medulloblastoma

Pratiti Bandopadhayay et al.

CLINICAL CANCER RESEARCH (2014)

Article Biochemistry & Molecular Biology

BET bromodomain proteins are required for glioblastoma cell proliferation

Chiara Pastori et al.

EPIGENETICS (2014)

Article Dermatology

The Epigenetic Regulator I-BET151 Induces BIM-Dependent Apoptosis and Cell Cycle Arrest of Human Melanoma Cells

Stuart J. Gallagher et al.

JOURNAL OF INVESTIGATIVE DERMATOLOGY (2014)

Article Chemistry, Multidisciplinary

Discovery and Optimization of Small-Molecule Ligands for the CBP/p300 Bromodomains

Duncan A. Hay et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)

Article Biochemistry & Molecular Biology

Dual kinase-bromodomain inhibitors for rationally designed polypharmacology

Pietro Ciceri et al.

NATURE CHEMICAL BIOLOGY (2014)

Article Multidisciplinary Sciences

BET and HDAC inhibitors induce similar genes and biological effects and synergize to kill in Myc-induced murine lymphoma

Joydeep Bhadury et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2014)

Article Immunology

BET bromodomain inhibition suppresses TH17-mediated pathology

Deanna A. Mele et al.

JOURNAL OF EXPERIMENTAL MEDICINE (2013)

Article Cardiac & Cardiovascular Systems

BET acetyl-lysine binding proteins control pathological cardiac hypertrophy

Jessica I. Spiltoir et al.

JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY (2013)

Article Oncology

Targeting MYCN in Neuroblastoma by BET Bromodomain Inhibition

Alexandre Puissant et al.

CANCER DISCOVERY (2013)

Article Biochemical Research Methods

ChromoHub: a data hub for navigators of chromatin-mediated signalling

Lihua Liu et al.

BIOINFORMATICS (2012)

Article Biochemistry & Molecular Biology

Small-Molecule Inhibition of BRDT for Male Contraception

Martin M. Matzuk et al.

Article Cell Biology

BET bromodomain inhibition as a novel strategy for reactivation of HIV-1

Camellia Banerjee et al.

JOURNAL OF LEUKOCYTE BIOLOGY (2012)

Article Multidisciplinary Sciences

Sensitivity of human lung adenocarcinoma cell lines to targeted inhibition of BET epigenetic signaling proteins

William W. Lockwood et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2012)

Article Biochemistry & Molecular Biology

BET Bromodomain Inhibition as a Therapeutic Strategy to Target c-Myc

Jake E. Delmore et al.

Article Multidisciplinary Sciences

Targeting MYC dependence in cancer by inhibiting BET bromodomains

Jennifer A. Mertz et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2011)

Article Multidisciplinary Sciences

Selective inhibition of BET bromodomains

Panagis Filippakopoulos et al.

NATURE (2010)

Article Multidisciplinary Sciences

Regulation of Cellular Metabolism by Protein Lysine Acetylation

Shimin Zhao et al.

SCIENCE (2010)

Article Biochemistry & Molecular Biology

Regulation of Aurora B Expression by the Bromodomain Protein Brd4

Jianxin You et al.

MOLECULAR AND CELLULAR BIOLOGY (2009)

Article Biochemistry & Molecular Biology

Mammalian ASH1L is a histone methyl transferase that occupies the transcribed region of active genes

Gregory D. Gregory et al.

MOLECULAR AND CELLULAR BIOLOGY (2007)

Article Genetics & Heredity

Mutations in the BRWD3 gene cause X-linked mental retardation associated with macrocephaly

Michael Field et al.

AMERICAN JOURNAL OF HUMAN GENETICS (2007)

Article Chemistry, Multidisciplinary

Selective small molecules blocking HIV-1 Tat and coactivator PCAF association

L Zeng et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2005)