4.8 Article

Catalytic, enantioselective synthesis of stilbene cis-diamines: A concise preparation of (-)-Nutlin-3, a potent p53/MDM2 inhibitor

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Multidisciplinary

Bifunctional Asymmetric Catalysis: Amplification of Bronsted Basicity Can Orthogonally Increase the Reactivity of a Chiral Bronsted Acid

Tyler A. Davis et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2010)

Article Multidisciplinary Sciences

Umpolung reactivity in amide and peptide synthesis

Bo Shen et al.

NATURE (2010)

Review Chemistry, Organic

Catalytic Enantioselective Aza-Henry Reactions

Eugenia Marques-Lopez et al.

EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2009)

Article Chemistry, Multidisciplinary

Metal-catalysed 1,2-diamination reactions

Francesca Cardona et al.

NATURE CHEMISTRY (2009)

Article Chemistry, Applied

A novel bis-thiourea organocatalyst for the asymmetric aza-Henry reaction

Constantinos Rampalakos et al.

ADVANCED SYNTHESIS & CATALYSIS (2008)

Article Chemistry, Multidisciplinary

A diastereo- and enantioselective synthesis of alpha-substituted anti-alpha,beta-diaminophosphonic acid derivatives

Jeremy C. Wilt et al.

CHEMICAL COMMUNICATIONS (2008)

Article Chemistry, Organic

The imino-pinacol coupling reaction

Vanessa Faugeroux et al.

CURRENT ORGANIC CHEMISTRY (2008)

Article Chemistry, Organic

The structure of polymer-supported triphenylphosphine ditriflate: A potentially useful reagent in organic synthesis

Maria J. Petersson et al.

JOURNAL OF ORGANIC CHEMISTRY (2008)

Article Chemistry, Multidisciplinary

A diastereo- and enantioselective synthesis of α-substituted syn-α,β-diamino acids

Anand Singh et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2008)

Review Chemistry, Organic

Organocatalytic asymmetric Mannich reactions: New methodology, catalyst design, and synthetic applications

Amal Ting et al.

EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2007)

Article Chemistry, Multidisciplinary

Chiral proton catalysis: Enantioselective bronsted acid catalyzed additions of nitroacetic acid derivatives as glycine equivalents

Anand Singh et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2007)

Article Chemistry, Organic

Enantioselective aza-Henry reaction using cinchona organocatalysts

L Bernardi et al.

TETRAHEDRON (2006)

Article Chemistry, Multidisciplinary

Bifunctional-thiourea-catalyzed diastereo- and enantioselective aza-Henry reaction

XN Xu et al.

CHEMISTRY-A EUROPEAN JOURNAL (2006)

Review Chemistry, Applied

Recent progress in chiral Bronsted acid catalysis

Takahiko Akiyama et al.

ADVANCED SYNTHESIS & CATALYSIS (2006)

Article Chemistry, Multidisciplinary

Catalytic enantioselective aza-Henry reaction with broad substrate scope

C Palomo et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2005)

Review Oncology

MDM2 is a central node in the p53 pathway: 12 years and counting

GL Bond et al.

CURRENT CANCER DRUG TARGETS (2005)

Article Chemistry, Multidisciplinary

Phase-transfer-catalyzed asymmetric aza-Henry reaction using N-carbamoyl imines generated in situ from alpha-amido sulfones

F Fini et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2005)

Article Chemistry, Multidisciplinary

Chiral proton catalysis: A catalytic enantioselective direct aza-Henry reaction

BM Nugent et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2004)

Article Chemistry, Organic

Enantioselective Aza-Henry reaction catalyzed by a bifunctional organocatalyst

T Okino et al.

ORGANIC LETTERS (2004)

Article Multidisciplinary Sciences

In vivo activation of the p53 pathway by small-molecule antagonists of MDM2

LT Vassilev et al.

SCIENCE (2004)

Article Pharmacology & Pharmacy

Small-molecule inhibitors of the p53 suppressor HDM2: have protein-protein interactions come of age as drug targets?

PM Fischer et al.

TRENDS IN PHARMACOLOGICAL SCIENCES (2004)

Article Multidisciplinary Sciences

Intrinsic tumour suppression

SW Lowe et al.

NATURE (2004)

Article Chemistry, Multidisciplinary

A biomimetic synthesis of thiazolines using hexaphenyloxodiphosphonium trifluoromethanesulfonate

SL You et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2003)

Article Chemistry, Multidisciplinary

Asymmetric catalytic aza-Henry reactions leading to 1,2-diamines and 1-,2-diaminocarboxylic acids

B Westermann

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2003)