期刊
TETRAHEDRON LETTERS
卷 52, 期 43, 页码 5643-5647出版社
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tetlet.2011.08.088
关键词
Thiazole-4-carboxylate; C-H bond activation; Oxidative Heck-coupling; Alkenylation; Direct arylation
资金
- Ministry of Education of China [NCET 2008]
- Fok Ying Tong Education Foundation [121040]
- Fundamental Research Funds for the Central Universities [JKZ2009002]
Oxidative Heck coupling of thiazole-4-carboxylates via palladium(II)-catalyzed C-H bond activation has been achieved in moderate to good yields. No ligand, and no acidic additive were used in the reaction. The results showed that this protocol tolerated a series of substitutions on the thiazole ring. A preliminary attempt of direct arylation with p-xylene via Pd(II)-catalyzed C-H bond activation has also been done. (C) 2011 Elsevier Ltd. All rights reserved.
作者
我是这篇论文的作者
点击您的名字以认领此论文并将其添加到您的个人资料中。
推荐
暂无数据