4.7 Article

Mechanism of Action of Thalassospiramides, A New Class of Calpain Inhibitors

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Biochemistry & Molecular Biology

A Coumarin- Labeled Vinyl Sulfone as Tripeptidomimetic Activity- Based Probe for Cysteine Cathepsins

Matthias D. Mertens et al.

CHEMBIOCHEM (2014)

Article Biochemistry & Molecular Biology

Enzyme Inhibition by Hydroamination: Design and Mechanism of a Hybrid Carmaphycin-Syringolin Enone Proteasome Inhibitor

Daniela B. B. Trivella et al.

CHEMISTRY & BIOLOGY (2014)

Article Chemistry, Medicinal

A Fragment-Based Method to Discover Irreversible Covalent Inhibitors of Cysteine Proteases

Stefan G. Kathman et al.

JOURNAL OF MEDICINAL CHEMISTRY (2014)

Article Chemistry, Multidisciplinary

Biosynthetic Multitasking Facilitates Thalassospiramide Structural Diversity in Marine Bacteria

Avena C. Ross et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)

Article Chemistry, Multidisciplinary

Probing the Mechanism of Cyanobacterial Aldehyde Decarbonylase Using a Cyclopropyl Aldehyde

Bishwajit Paul et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)

Article Biochemistry & Molecular Biology

Discovery of Specific Inhibitors of Human USP7/HAUSP Deubiquitinating Enzyme

Celine Reverdy et al.

CHEMISTRY & BIOLOGY (2012)

Article Chemistry, Medicinal

Kinetic Template-Guided Tethering of Fragments

Rebecca H. Nonoo et al.

CHEMMEDCHEM (2012)

Review Chemistry, Medicinal

Calpain inhibitors: a survey of compounds reported in the patent and scientific literature

Isaac O. Donkor

EXPERT OPINION ON THERAPEUTIC PATENTS (2011)

Review Pharmacology & Pharmacy

Calpains as potential anti-cancer targets

Ludovic Leloup et al.

EXPERT OPINION ON THERAPEUTIC TARGETS (2011)

Article Chemistry, Medicinal

Molecular Modeling: A Search for a Calpain Inhibitor as a New Treatment for Cataractogenesis

Blair G. Stuart et al.

JOURNAL OF MEDICINAL CHEMISTRY (2011)

Review Chemistry, Medicinal

Calpains: Attractive Targets for the Development of Synthetic Inhibitors

Markus Pietsch et al.

CURRENT TOPICS IN MEDICINAL CHEMISTRY (2010)

Review Veterinary Sciences

Expanding Members and Roles of the Calpain Superfamily and Their Genetically Modified Animals

Hiroyuki Sorimachi et al.

EXPERIMENTAL ANIMALS (2010)

Article Biochemical Research Methods

Deciphering Modifications in Swine Cardiac Troponin I by Top-Down High-Resolution Tandem Mass Spectrometry

Jiang Zhang et al.

JOURNAL OF THE AMERICAN SOCIETY FOR MASS SPECTROMETRY (2010)

Article Neurosciences

Regulation of Calpain-2 in Neurons: Implications for Synaptic Plasticity

Sohila Zadran et al.

MOLECULAR NEUROBIOLOGY (2010)

Review Clinical Neurology

Calpain as a Therapeutic Target in Traumatic Brain Injury

Kathryn E. Saatman et al.

NEUROTHERAPEUTICS (2010)

Article Chemistry, Physical

Staggered Mesh Ewald: An Extension of the Smooth Particle-Mesh Ewald Method Adding Great Versatility

David S. Cerutti et al.

JOURNAL OF CHEMICAL THEORY AND COMPUTATION (2009)

Article Chemistry, Multidisciplinary

AutoDock4 and AutoDockTools4: Automated Docking with Selective Receptor Flexibility

Garrett M. Morris et al.

JOURNAL OF COMPUTATIONAL CHEMISTRY (2009)

Article Chemistry, Medicinal

Novel Peptidomimetics Containing a Vinyl Ester Moiety as Highly Potent and Selective Falcipain-2 Inhibitors

Roberta Ettari et al.

JOURNAL OF MEDICINAL CHEMISTRY (2009)

Article Multidisciplinary Sciences

Synthetic and structural studies on syringolin A and B reveal critical determinants of selectivity and potency of proteasome inhibition

Jerome Clerc et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2009)

Article Multidisciplinary Sciences

Top-down high-resolution mass spectrometry of cardiac myosin binding protein C revealed that truncation alters protein phosphorylation state

Ying Ge et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2009)

Article Chemistry, Physical

GROMACS 4: Algorithms for highly efficient, load-balanced, and scalable molecular simulation

Berk Hess et al.

JOURNAL OF CHEMICAL THEORY AND COMPUTATION (2008)

Article Chemistry, Medicinal

Structural basis for the potent calpain inhibitory activity of peptidyl α-ketoacids

Isaac O. Donkor et al.

JOURNAL OF MEDICINAL CHEMISTRY (2008)

Review Endocrinology & Metabolism

Mechanistic role of calpains in postischemic neurodegeneration

Matthew B. Bevers et al.

JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM (2008)

Article Biochemistry & Molecular Biology

Development of calpain-specific inactivators by screening of positional scanning epoxide libraries

Dominic Cuerrier et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2007)

Review Biotechnology & Applied Microbiology

The calpains: modular designs and functional diversity

Dorothy E. Croall et al.

GENOME BIOLOGY (2007)

Article Biochemistry & Molecular Biology

Comparison of multiple amber force fields and development of improved protein backbone parameters

Viktor Hornak et al.

PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS (2006)

Review Pharmacology & Pharmacy

The therapeutic potential of the calpain family: new aspects

Maria E. Saez et al.

DRUG DISCOVERY TODAY (2006)

Article Chemistry, Medicinal

Exploration of orally available calpain inhibitors 2: Peptidyl hemiacetal derivatives

Yoshihisa Shirasaki et al.

JOURNAL OF MEDICINAL CHEMISTRY (2006)

Article Biochemistry & Molecular Biology

Calpain inhibition by α-ketoamide and cyclic hemiacetal inhibitors revealed by X-ray crystallography

D. Cuerrier et al.

BIOCHEMISTRY (2006)

Review Medicine, General & Internal

Mechanisms of disease: Calpains and disease

M Zatz et al.

NEW ENGLAND JOURNAL OF MEDICINE (2005)

Article Biochemistry & Molecular Biology

α,β-unsaturated ketone is a core moiety of natural ligands for covalent binding to peroxisome proliferator-activated receptor

T Shiraki et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2005)

Article Biochemistry & Molecular Biology

PDB2PQR: an automated pipeline for the setup of Poisson-Boltzmann electrostatics calculations

TJ Dolinsky et al.

NUCLEIC ACIDS RESEARCH (2004)

Article Biochemistry & Molecular Biology

A Ca2+ switch aligns the active site of calpain

T Moldoveanu et al.

Article Biochemical Research Methods

Reactivity of the NS2/3((907-1206))ASK(4) protein with beta-mercaptoethanol studied by electrospray ion trap mass spectrometry

L Orsatti et al.

RAPID COMMUNICATIONS IN MASS SPECTROMETRY (2002)

Review Biochemistry & Molecular Biology

A survey of calpain inhibitors

IO Donkor

CURRENT MEDICINAL CHEMISTRY (2000)