相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。Structure-Function of the G Protein-Coupled Receptor Superfamily
Vsevolod Katritch et al.
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, VOL 53, 2013 (2013)
Structural Basis for Molecular Recognition at Serotonin Receptors
Chong Wang et al.
SCIENCE (2013)
A Simple Method for Quantifying Functional Selectivity and Agonist Bias
Terry Kenakin et al.
ACS CHEMICAL NEUROSCIENCE (2012)
Molecular Mechanism of beta-Arrestin-Biased Agonism at Seven-Transmembrane Receptors
Eric Reiter et al.
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, VOL 52 (2012)
OPM database and PPM web server: resources for positioning of proteins in membranes
Mikhail A. Lomize et al.
NUCLEIC ACIDS RESEARCH (2012)
Structural insights into biased G protein-coupled receptor signaling revealed by fluorescence spectroscopy
Rita Rahmeh et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2012)
Biased Signaling Pathways in β2-Adrenergic Receptor Characterized by 19F-NMR
Jeffrey J. Liu et al.
SCIENCE (2012)
Crystal Structures of a Stabilized β1-Adrenoceptor Bound to the Biased Agonists Bucindolol and Carvedilol
Tony Warne et al.
STRUCTURE (2012)
Strategies to Discover Unexpected Targets for Drugs Active at G Protein-Coupled Receptors
John A. Allen et al.
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, VOL 51, 2011 (2011)
Development of an Automated High Throughput LCP-FRAP Assay to Guide Membrane Protein Crystallization in Lipid Mesophases
Fei Xu et al.
CRYSTAL GROWTH & DESIGN (2011)
Functional Selectivity and Biased Receptor Signaling
Terry Kenakin
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2011)
Structure of a nanobody-stabilized active state of the β2 adrenoceptor
Soren G. F. Rasmussen et al.
NATURE (2011)
Crystal structure of the β2 adrenergic receptor-Gs protein complex
Soren G. F. Rasmussen et al.
NATURE (2011)
Ligand discovery from a dopamine D3 receptor homology model and crystal structure
Jens Carlsson et al.
NATURE CHEMICAL BIOLOGY (2011)
Discovery of β-Arrestin-Biased Dopamine D2 Ligands for Probing Signal Transduction Pathways Essential for Antipsychotic Efficacy
John A. Allen et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2011)
Structure of an Agonist-Bound Human A2A Adenosine Receptor
Fei Xu et al.
SCIENCE (2011)
Features and development of Coot
P. Emsley et al.
ACTA CRYSTALLOGRAPHICA SECTION D-BIOLOGICAL CRYSTALLOGRAPHY (2010)
PHENIX: a comprehensive Python-based system for macromolecular structure solution
Paul D. Adams et al.
ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY (2010)
Conserved Binding Mode of Human β2 Adrenergic Receptor Inverse Agonists and Antagonist Revealed by X-ray Crystallography
Daniel Wacker et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2010)
The Expanded Biology of Serotonin
Miles Berger et al.
ANNUAL REVIEW OF MEDICINE (2009)
β-Arrestin-2 Mediates Anti-apoptotic Signaling through Regulation of BAD Phosphorylation
Seungkirl Ahn et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2009)
Rastering strategy for screening and centring of microcrystal samples of human membrane proteins with a sub-10 μm size X-ray synchrotron beam
Vadim Cherezov et al.
JOURNAL OF THE ROYAL SOCIETY INTERFACE (2009)
Parallel Functional Activity Profiling Reveals Valvulopathogens Are Potent 5-Hydroxytryptamine2B Receptor Agonists: Implications for Drug Safety Assessment
Xi-Ping Huang et al.
MOLECULAR PHARMACOLOGY (2009)
Crystallizing membrane proteins using lipidic mesophases
Martin Caffrey et al.
NATURE PROTOCOLS (2009)
Ligand binding and micro-switches in 7TM receptor structures
Rie Nygaard et al.
TRENDS IN PHARMACOLOGICAL SCIENCES (2009)
Stabilization of the human β2-adrenergic receptor TM4-TM3-TM5 helix interface by mutagenesis of Glu1223.41, a critical residue in GPCR structure
Christopher B. Roth et al.
JOURNAL OF MOLECULAR BIOLOGY (2008)
Crystal structure of opsin in its G-protein-interacting conformation
Patrick Scheerer et al.
NATURE (2008)
The genetic design of signaling cascades to record receptor activation
Gilad Barnea et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2008)
High-resolution crystal structure of an engineered human β2-adrenergic G protein-coupled receptor
Vadim Cherezov et al.
SCIENCE (2007)
Profiling of membrane protein variants in a baculovirus system by coupling cell-surface detection with small-scale parallel expression
Michael A. Hanson et al.
PROTEIN EXPRESSION AND PURIFICATION (2007)
Phaser crystallographic software
Airlie J. McCoy et al.
JOURNAL OF APPLIED CRYSTALLOGRAPHY (2007)
Functional selectivity and classical concepts of quantitative pharmacology
Jonathan D. Urban et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2007)
HKL-3000:: the integration of data reduction and structure solution -: from diffraction images to an initial model in minutes
Wladek Minor et al.
ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY (2006)
Identification of β-arrestin2 as a G protein-coupled receptor-stimulated regulator of NF-κB pathways
H Gao et al.
MOLECULAR CELL (2004)
Redesign of a four-helix bundle protein by phage display coupled with proteolysis and structural characterization by NMR and X-ray crystallography
R Chu et al.
JOURNAL OF MOLECULAR BIOLOGY (2002)
Endocytosis of the mu opioid receptor reduces tolerance and a cellular hallmark of opiate withdrawal
AK Finn et al.
NEURON (2001)
Light-induced conformational changes of rhodopsin probed by fluorescent Alexa594 immobilized on the cytoplasmic surface
Y Imamoto et al.
BIOCHEMISTRY (2000)