4.8 Article

Discovery of drug-like inhibitors of an essential RNA-editing ligase in Trypanosoma brucei

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Chemistry, Medicinal

Ensemble-based virtual screening reveals potential novel antiviral compounds for avian influenza neuraminidase

Lily S. Cheng et al.

JOURNAL OF MEDICINAL CHEMISTRY (2008)

Article Biochemistry & Molecular Biology

RNA editing in Trypanosoma brucei requires three different editosomes

Jason Carnes et al.

MOLECULAR AND CELLULAR BIOLOGY (2008)

Review Pharmacology & Pharmacy

Human African trypanosomiasis: pharmacological re-engagement with a neglected disease

M. P. Barrett et al.

BRITISH JOURNAL OF PHARMACOLOGY (2007)

Article Chemistry, Multidisciplinary

A semiempirical free energy force field with charge-based desolvation

Ruth Huey et al.

JOURNAL OF COMPUTATIONAL CHEMISTRY (2007)

Review Chemistry, Multidisciplinary

DNA ligases: Structure, reaction mechanism, and function

AE Tomkinson et al.

CHEMICAL REVIEWS (2006)

Article Chemistry, Medicinal

Novel procedure for modeling ligand/receptor induced fit effects

W Sherman et al.

JOURNAL OF MEDICINAL CHEMISTRY (2006)

Review Parasitology

Chemotherapy of trypanosomiases and leishmaniasis

SL Croft et al.

TRENDS IN PARASITOLOGY (2005)

Review Biochemistry & Molecular Biology

Complex management: RNA editing in trypanosomes

KD Stuart et al.

TRENDS IN BIOCHEMICAL SCIENCES (2005)

Article Chemistry, Medicinal

Discovery of a novel binding trench in HIV integrase

JR Schames et al.

JOURNAL OF MEDICINAL CHEMISTRY (2004)

Article Biochemistry & Molecular Biology

Protein flexibility in ligand docking and virtual screening to protein kinases

CN Cavasotto et al.

JOURNAL OF MOLECULAR BIOLOGY (2004)

Article Biochemistry & Molecular Biology

Structure and mechanism of RNA ligase

CK Ho et al.

STRUCTURE (2004)

Article Multidisciplinary Sciences

A naphthyridine carboxamide provides evidence for discordant resistance between mechanistically identical inhibitors of HIV-1 integrase

DJ Hazuda et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2004)

Review Biochemistry & Molecular Biology

Integrating virtual screening in lead discovery

TI Oprea et al.

CURRENT OPINION IN CHEMICAL BIOLOGY (2004)

Article Biochemistry & Molecular Biology

PDB2PQR: an automated pipeline for the setup of Poisson-Boltzmann electrostatics calculations

TJ Dolinsky et al.

NUCLEIC ACIDS RESEARCH (2004)

Article Biochemistry & Molecular Biology

High resolution crystal structure of a key editosome enzyme from Trypanosoma brucei:: RNA editing ligase 1

JP Deng et al.

JOURNAL OF MOLECULAR BIOLOGY (2004)

Article Multidisciplinary Sciences

Nonlinear elasticity, proteinquakes, and the energy landscapes of functional transitions in proteins

O Miyashita et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2003)

Review Pharmacology & Pharmacy

Drug transport and drug resistance in African trypanosomes

P Mäser et al.

DRUG RESISTANCE UPDATES (2003)

Article Chemistry, Medicinal

A specific mechanism of nonspecific inhibition

SL McGovern et al.

JOURNAL OF MEDICINAL CHEMISTRY (2003)

Article Biochemistry & Molecular Biology

Separate insertion and deletion subcomplexes of the Trypanosoma brucei RNA editing complex

A Schnaufer et al.

MOLECULAR CELL (2003)

Article Chemistry, Medicinal

Effect of detergent on promiscuous inhibitors

AJ Ryan et al.

JOURNAL OF MEDICINAL CHEMISTRY (2003)

Article Biochemistry & Molecular Biology

Structure-function analysis of T4 RNA ligase 2

SM Yin et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2003)

Review Microbiology

Evolution of structure in aminoacyl-tRNA synthetases

P O'Donoghue et al.

MICROBIOLOGY AND MOLECULAR BIOLOGY REVIEWS (2003)

Review Biochemistry & Molecular Biology

Protein flexibility and drug design: how to hit a moving target

HA Carlson

CURRENT OPINION IN CHEMICAL BIOLOGY (2002)

Review Parasitology

Natural and induced dyskinetoplastic trypanosomatids: how to live without mitochondrial DNA

A Schnaufer et al.

INTERNATIONAL JOURNAL FOR PARASITOLOGY (2002)

Article Chemistry, Multidisciplinary

Computational drug design accommodating receptor flexibility: The relaxed complex scheme

JH Lin et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2002)

Article Chemistry, Multidisciplinary

Comparison of the NCI open database with seven large chemical structural databases

JH Voigt et al.

JOURNAL OF CHEMICAL INFORMATION AND COMPUTER SCIENCES (2001)

Article Biochemistry & Molecular Biology

FlexE: Efficient molecular docking considering protein structure variations

H Claussen et al.

JOURNAL OF MOLECULAR BIOLOGY (2001)

Article Chemistry, Multidisciplinary

Mining and visualizing large anticancer drug discovery databases

LM Shi et al.

JOURNAL OF CHEMICAL INFORMATION AND COMPUTER SCIENCES (2000)