期刊
ORGANIC LETTERS
卷 16, 期 7, 页码 2074-2076出版社
AMER CHEMICAL SOC
DOI: 10.1021/ol500588v
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资金
- North Carolina State University
- American Chemical Society
A copper catalyzed aminobromination of Alkene tethered thiohydroximic acids is described, providing a rapid approach to unnatural thiazoline scaffolds not readily available via existing methods. Moderate to high yields of bromothiazolines are obtained with alkyl- and aryl-substituted thiohydroximic acid building blocks containing mono-, di-, and trisubstituted alkenes. The reaction provides high levels of 5-exo selectivity, and terminally monosubstituted alkenes result in predominant syn-diastereoselectivity.
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