期刊
ORGANIC LETTERS
卷 14, 期 14, 页码 3760-3763出版社
AMER CHEMICAL SOC
DOI: 10.1021/ol301616w
关键词
-
资金
- EPFL (Switzerland)
- Swiss National Science Foundation (SNF)
- Swiss National Centres of Competence in Research (NCCR)
- ICSN
- CNRS (France)
- EPFL
Treatment of a DMA solution of anilide 1 with a catalytic amount of palladium acetate (0.025 equiv) and XPhos (0.05 equiv) in the presence of potassium carbonate (2.0 equiv) at 100 degrees C afforded dihydroquinolin-2-ones spiro-fused to dihydrofuranyl, indolinyl, and indanyl 2 in good to excellent yields. The reaction went through a domino sequence involving a 5-exo-trig Heck cyclization followed by an intramolecular direct C-H functionalization.
作者
我是这篇论文的作者
点击您的名字以认领此论文并将其添加到您的个人资料中。
推荐
暂无数据