期刊
ORGANIC LETTERS
卷 13, 期 16, 页码 4220-4223出版社
AMER CHEMICAL SOC
DOI: 10.1021/ol201555z
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资金
- Natural Science Foundation of Zhejiang Province [Y4100201]
- Foundation of Science and Technology Department of Zhejiang Province [2011R09002-09]
- Opening Foundation of Zhejiang Provincial Top Key Discipline
A mild and efficient protocol for the synthesis of fluorinated pyrazoles has been developed via gold(I)-catalyzed tandem aminofluorination of alkynes in the presence of Selectfluor. This method offers a broad substrate scope.
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