期刊
MINI-REVIEWS IN MEDICINAL CHEMISTRY
卷 8, 期 10, 页码 996-1005出版社
BENTHAM SCIENCE PUBL LTD
DOI: 10.2174/138955708785740607
关键词
arginine-vasopressin; oxytocin; G protein-coupled receptor; structure-activity relationships; fluorescent peptide; fluorescence resonance energy transfer; fluorescence polarization; high-throughput screening assays
资金
- NIGMS NIH HHS [R01 GM025280, GM25280] Funding Source: Medline
Different series of fluorescent agonists and antagonists have been developed and characterized for argininevasopressin and oxytocin G protein-coupled receptors. Both cyclic and linear peptide analogs of the neurohypophysial hormones are useful tools for investigating receptor localization and trafficking, analysing receptor structural organization, and developing new receptor-selective high-throughput ligand screening assays.
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