期刊
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
卷 136, 期 9, 页码 3354-3357出版社
AMER CHEMICAL SOC
DOI: 10.1021/ja412880r
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资金
- Shanghai Institute of Organic Chemistry
- Chinese Academy of Sciences
- CAS/SAFEA International Partnership Program for Creative Research Teams
- Recruitment Program of Global Experts
A Cu(OAc)(2)-mediated C-H amidation and amination of arenes and heteroarenes has been developed using a readily removable directing group. A wide range of sulfonamides, amides, and anilines function as amine donors in this reaction. Heterocycles present in both reactants are tolerated, making this a broadly applicable method for the synthesis of a family of inhibitors including 2-benzamidobenzoic acids and N-phenylaminobenzoates.
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