4.2 Article

A stable meta-carborane enables the generation of boron-rich peptide agonists targeting the ghrelin receptor

相关参考文献

注意:仅列出部分参考文献,下载原文获取全部文献信息。
Article Biochemistry & Molecular Biology

Direct carborane-peptide conjugates: Synthesis and evaluation as non natural lipopeptide mimetics

Tamara Luetzenburg et al.

CHEMISTRY AND PHYSICS OF LIPIDS (2018)

Review Pharmacology & Pharmacy

Towards carborane-functionalised structures for the treatment of brain cancer

Gianpiero Calabrese et al.

DRUG DISCOVERY TODAY (2018)

Article Biochemistry & Molecular Biology

High metabolic in vivo stability and bioavailability of a palmitoylated ghrelin receptor ligand assessed by mass spectrometry

Katja B. Kostelnik et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2015)

Review Chemistry, Multidisciplinary

Advancements in Tumor Targeting Strategies for Boron Neutron Capture Therapy

Micah John Luderer et al.

PHARMACEUTICAL RESEARCH (2015)

Review Endocrinology & Metabolism

MECHANISMS IN ENDOCRINOLOGY Regulation of glucose metabolism by the ghrelin system: multiple players and multiple actions

Kristy M. Heppner et al.

EUROPEAN JOURNAL OF ENDOCRINOLOGY (2014)

Review Chemistry, Medicinal

N3-substituted thymidine bioconjugates for cancer therapy and imaging

Ahmed Khalil et al.

FUTURE MEDICINAL CHEMISTRY (2013)

Article Chemistry, Medicinal

An Aromatic Region To Induce a Switch between Agonism and Inverse Agonism at the Ghrelin Receptor

Sylvia Els et al.

JOURNAL OF MEDICINAL CHEMISTRY (2012)

Review Chemistry, Multidisciplinary

Carbaboranes as Pharmacophores: Properties, Synthesis, and Application Strategies

Matthias Scholz et al.

CHEMICAL REVIEWS (2011)

Article Biochemistry & Molecular Biology

Unique Interaction Pattern for a Functionally Biased Ghrelin Receptor Agonist

Bjorn Sivertsen et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2011)

Article Chemistry, Medicinal

Incorporation of ortho-Carbaboranyl-Nε-Modified L-Lysine into Neuropeptide Y Receptor Y1- and Y2-Selective Analogues

Verena M. Ahrens et al.

JOURNAL OF MEDICINAL CHEMISTRY (2011)

Article Chemistry, Multidisciplinary

Structure-Activity Relationships of GHRP-6 Azapeptide Ligands of the CD36 Scavenger Receptor by Solid-Phase Submonomer Azapeptide Synthesis

David Sabatino et al.

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2011)

Review Endocrinology & Metabolism

Ghrelin: A potential therapeutic target for cancer

Dimitrios Nikolopoulos et al.

REGULATORY PEPTIDES (2010)

Article Chemistry, Inorganic & Nuclear

Biological evaluation of boronated unnatural amino acids as new boron carriers

G. W. Kabalka et al.

APPLIED RADIATION AND ISOTOPES (2009)

Article Biochemistry & Molecular Biology

Identification of an efficacy switch region in the ghrelin receptor responsible for interchange between agonism and inverse agonism

Birgitte Holst et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2007)

Article Biochemistry & Molecular Biology

Ghrelin and the growth hormone secretagogue receptor constitute a novel autocrine pathway in astrocytoma motility

Vishwa Deep Dixit et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2006)

Article Chemistry, Multidisciplinary

Targeting normal and neoplastic tissues in the rat jejunum and colon with boronated, cationic acrylamide copolymers

AK Azab et al.

JOURNAL OF CONTROLLED RELEASE (2005)

Review Oncology

Boron neutron capture therapy of cancer: Current status and future prospects

RF Barth et al.

CLINICAL CANCER RESEARCH (2005)

Article Chemistry, Inorganic & Nuclear

Conjugation of the closo-borane mereaptoundecahydrododecaborate (BSH) to a tumour selective peptide

W Mier et al.

ZEITSCHRIFT FUR ANORGANISCHE UND ALLGEMEINE CHEMIE (2004)

Review Endocrinology & Metabolism

Peptide receptors as molecular targets for cancer diagnosis and therapy

JC Reubi

ENDOCRINE REVIEWS (2003)

Article Endocrinology & Metabolism

High constitutive signaling of the ghrelin receptor - Identification of a potent inverse agonist

B Holst et al.

MOLECULAR ENDOCRINOLOGY (2003)

Review Chemistry, Inorganic & Nuclear

The medicinal chemistry of carboranes

JF Valliant et al.

COORDINATION CHEMISTRY REVIEWS (2002)

Article Cardiac & Cardiovascular Systems

CD36 mediates the cardiovascular action of growth hormone-releasing peptides in the heart

V Bodart et al.

CIRCULATION RESEARCH (2002)