期刊
JOURNAL OF ORGANIC CHEMISTRY
卷 79, 期 19, 页码 9000-9008出版社
AMER CHEMICAL SOC
DOI: 10.1021/jo501250u
关键词
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资金
- National Natural Science Foundation of China [21202152]
- Zhejiang Provincial Natural Science Foundation [Y4110044]
A straightforward assembly of 1,2-disubstituted indoles has been developed through a Cu(II)-catalyzed domino coupling/cyclization process. Under aerobic conditions, a wide range of 1,2-disubstituted indole derivatives were efficiently and facilely synthesized from 2-alkynylanilines and boronic acids. 2-(2-Bromoaryl)-1-aryl-1H-indoles, which were selectively generated in one pot under the Cu catalysis, afforded the indolo[1,2-f]phenanthridines via Pd-catalyzed intramolecular direct C(sp(2))-H arylation. The one-pot tandem approaches to the polycyclic indole derivatives were also successfully achieved.
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