期刊
ORGANIC LETTERS
卷 17, 期 19, 页码 4710-4713出版社
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.5b02173
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资金
- Universite Francois Rabelais de Tours
- Labex SynOrg [ANR-11-LABX-0029]
- ANR-LABEX SynOrg [ANR-11-LABX-0029]
A simple and efficient procedure for the Pd-catalyzed amination of N-free 2-chloro-7-azaindole is described, using either primary or secondary amines. An optimized combination of Brettphos, a Brettphos precatalyst, and LiHMDS in THF led us to a novel methodology, applied to various functionalized amines to study the scope of the reaction. This is the first report of cross-coupling amination on N-free 2-chloro-7-azaindole.
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