期刊
JOURNAL OF HETEROCYCLIC CHEMISTRY
卷 46, 期 6, 页码 1420-1424出版社
WILEY-BLACKWELL PUBLISHING, INC
DOI: 10.1002/jhet.230
关键词
-
资金
- European Commission [HEALTH-F3-2008-201032]
We herein report conventional and microwave-assisted methods for the synthesis of a series of compounds containing some bivalent ion chelating requirements useful to exert potential HIV-1 integrase (IN) enzyme inhibition activity. The biological screening highlighted that only derivative 5 proved to be a strand-transfer step inhibitor of the virus integration process at micromolar concentration.
作者
我是这篇论文的作者
点击您的名字以认领此论文并将其添加到您的个人资料中。
推荐
暂无数据