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CURRENT PHARMACEUTICAL DESIGN (2013)
Inactivation of the Cullin (CUL)-RING E3 ligase by the NEDD8-activating enzyme inhibitor MLN4924 triggers protective autophagy in cancer cells
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CANCER RESEARCH (2012)
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CELL RESEARCH (2012)
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ENDOCRINOLOGY (2012)
Minireview: Animal Models and Mechanisms of Ovarian Cancer Development
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ENDOCRINOLOGY (2012)
Either Kras activation or Pten loss similarly enhance the dominant-stable CTNNB1-induced genetic program to promote granulosa cell tumor development in the ovary and testis
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ONCOGENE (2012)
The oncogenic phosphatase PPM1D confers cisplatin resistance in ovarian carcinoma cells by attenuating checkpoint kinase 1 and p53 activation
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ONCOGENE (2012)
Genetic Abolishment of Hepatocyte Proliferation Activates Hepatic Stem Cells
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PLOS ONE (2012)
The p21-Dependent Radiosensitization of Human Breast Cancer Cells by MLN4924, an Investigational Inhibitor of NEDD8 Activating Enzyme
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PLOS ONE (2012)
Radiosensitization of Cancer Cells by Inactivation of Cullin-RING E3 Ubiquitin Ligases
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Targeting Cullin-RING ligases by MLN4924 induces autophagy via modulating the HIF1-REDD1-TSC1-mTORC1-DEPTOR axis
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CELL DEATH & DISEASE (2012)
SCF E3 Ubiquitin Ligases as Anticancer Targets
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CURRENT CANCER DRUG TARGETS (2011)
Cul4A is essential for spermatogenesis and male fertility
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DEVELOPMENTAL BIOLOGY (2011)
The E3 ubiquitin ligase Cullin 4A regulates meiotic progression in mouse spermatogenesis
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DEVELOPMENTAL BIOLOGY (2011)
Molecular and functional characteristics of ovarian surface epithelial cells transformed by KrasG12D and loss of Pten in a mouse model in vivo
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ONCOGENE (2011)
Induction of p21-Dependent Senescence by an NAE Inhibitor, MLN4924, as a Mechanism of Growth Suppression
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NEOPLASIA (2011)
Akt promotes chemoresistance in human ovarian cancer cells by modulating cisplatin-induced, p53-dependent ubiquitination of FLICE-like inhibitory protein
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ONCOGENE (2010)
Hepatocyte-specific deletion of DDB1 induces liver regeneration and tumorigenesis
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PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2010)
ROC1/RBX1 E3 Ubiquitin Ligase Silencing Suppresses Tumor Cell Growth via Sequential Induction of G2-M Arrest, Apoptosis, and Senescence
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CANCER RESEARCH (2009)
Differential activity of UV-DDB in mouse keratinocytes and fibroblasts: Impact on DNA repair and UV-induced skin cancer
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DNA REPAIR (2009)
CUL4A Abrogation Augments DNA Damage Response and Protection against Skin Carcinogenesis
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MOLECULAR CELL (2009)
An inhibitor of NEDD8-activating enzyme as a new approach to treat cancer
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Protein kinase DYRK2 is a scaffold that facilitates assembly of an E3 ligase
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NATURE CELL BIOLOGY (2009)
CRL4s: the CUL4-RING E3 ubiquitin ligases
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TRENDS IN BIOCHEMICAL SCIENCES (2009)
RBX1/ROC1-SCF E3 ubiquitin ligase is required for mouse embryogenesis and cancer cell survival
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CELL DIVISION (2009)
Human immunodeficiency virus type 1 Vpr-binding protein VprBP, a WD40 protein associated with the DDB1-CUL4 E3 ubiquitin ligase, is essential for DNA replication and embryonic development
Chad M. McCall et al.
MOLECULAR AND CELLULAR BIOLOGY (2008)
VprBP targets Merlin to the Roc1-Cul4A-DDB1 E3 ligase complex for degradation
J. Huang et al.
ONCOGENE (2008)
DCAFs, the missing link of the CUL4-DDB1 ubiquitin ligase
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MOLECULAR CELL (2007)
DDB1 is essential for genomic stability in developing epidermis
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PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2007)
The Caenorhabditis elegans replication licensing factor CDT-1 is targeted for degradation by the CUL-4/DDB-1 complex
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MOLECULAR AND CELLULAR BIOLOGY (2007)
Deletion of DDB1 in mouse brain and lens leads to p53-dependent elimination of proliferating cells
Yong Cang et al.
CELL (2006)
Tumor-prone phenotype of the DDB2-deficient mice
T Yoon et al.
ONCOGENE (2005)
Possible role of FLICE-like inhibitory protein (FLIP) in chemoresistant ovarian cancer cells in vitro
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ONCOGENE (2004)