Journal
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
Volume 2014, Issue 22, Pages 4837-4843Publisher
WILEY-V C H VERLAG GMBH
DOI: 10.1002/ejoc.201402456
Keywords
Synthetic methods; Nitrogen heterocycles; C-H functionalization; Amination; Iodine
Categories
Funding
- National Natural Science Foundation of China (NSFC) [21272149]
- Shanghai Municipal Education Commission [14ZZ094]
- Science and Technology Commission of Shanghai Municipality [13ZR1416400]
Ask authors/readers for more resources
An efficient and mild synthesis of imidazo[1,2-a]pyrimidine derivatives has been developed from readily available pyrimidyl arylamines or enamines through a hypervalent iodine-promoted intramolecular C-H bond cycloamination reaction. This protocol allows for the facile construction of biologically active bicyclic imidazo[1,2-alpha]pyrimidine skeletons as well as other imidazo[1,2-alpha]-type fused heterocycles.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available
Share Paper
