Journal
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
Volume 2011, Issue 2, Pages 271-279Publisher
WILEY-V C H VERLAG GMBH
DOI: 10.1002/ejoc.201000936
Keywords
Pyridine N-oxides; Boekelheide rearrangement; Cyclization; Intramolecular reactions; Nitrogen heterocycles; Synthetic methods
Categories
Funding
- GlaxoSmithKline of Verona
Ask authors/readers for more resources
Pyrrolidines and piperidines were synthesized from (aminoalkyl)pyridine N-oxides with a general and quite efficient method developed by using di-tert-butylsilyl bis(trifluoromethanesulfonate) as a new promoter for a Boekelheide-type reaction. The use of a new Boekelheide promoter, which is compatible with amino groups, opens new perspectives in view of its application in intramolecular cyclizations.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available