Related references
Note: Only part of the references are listed.Advances in Imaging Target Delineation
Klaudia U. Hunter et al.
CANCER JOURNAL (2011)
A Glimpse of the Future Where Will New Combinations of Diagnostics and Therapies Take Us?
Michelle Alonso-Basanta et al.
CANCER JOURNAL (2011)
Integrin alpha(v)beta(3)-targeted gold nanoshells augment tumor vasculature-specific imaging and therapy
Huan Xie et al.
INTERNATIONAL JOURNAL OF NANOMEDICINE (2011)
Integrin α5β1 facilitates cancer cell invasion through enhanced contractile forces
Claudia Tanja Mierke et al.
JOURNAL OF CELL SCIENCE (2011)
PET of αvβ3-Integrin and αvβ5-Integrin Expression with 18F-Fluciclatide for Assessment of Response to Targeted Therapy: Ready for Prime Time?
Ambros J. Beer et al.
JOURNAL OF NUCLEAR MEDICINE (2011)
Towards novel paradigms for cancer therapy
V. Pavet et al.
ONCOGENE (2011)
The tail of integrin activation
Nicholas J. Anthis et al.
TRENDS IN BIOCHEMICAL SCIENCES (2011)
Inhibition of HIV-1 Replication by Isoxazolidine and Isoxazole Sulfonamides
Belinda Loh et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2010)
Total Syntheses of Tubulysins
Taku Shibue et al.
CHEMISTRY-A EUROPEAN JOURNAL (2010)
Small Molecule Antagonists of Integrin Receptors
A. Perdih et al.
CURRENT MEDICINAL CHEMISTRY (2010)
Click-Chemistry-Derived Triazole Ligands of Arginine-Glycine-Aspartate (RGD) Integrins with a Broad Capacity To Inhibit Adhesion of Melanoma Cells and Both in Vitro and in Vivo Angiogenesis
Andrea Trabocchi et al.
JOURNAL OF MEDICINAL CHEMISTRY (2010)
A New View of Carcinogenesis and an Alternative Approach to Cancer Therapy
Miguel Lopez-Lazaro
MOLECULAR MEDICINE (2010)
Ligands for Mapping αvβ3-Integrin Expression in Vivo
Margret Schottelius et al.
ACCOUNTS OF CHEMICAL RESEARCH (2009)
Mapping the ligand-binding pocket of integrin α5β1 using a gain-of-function approach
A. Paul Mould et al.
BIOCHEMICAL JOURNAL (2009)
Expanding the repertoire of small molecule transcriptional activation domains
Ryan J. Casey et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2009)
Cyclic RGD-Containing Functionalized Azabicycloalkane Peptides as Potent Integrin Antagonists for Tumor Targeting
Leonardo Manzoni et al.
CHEMMEDCHEM (2009)
α5β1-Integrin controls ebolavirus entry by regulating endosomal cathepsins
Kathryn L. Schornberg et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2009)
A convenient synthesis of functionalized isoxazolines and related 5-hydroxyisoxazolidine-4-carboxylates
Fides Benfatti et al.
TETRAHEDRON (2009)
Investigations on synthesis of indole based constrained mimetic scaffolds through 1,3-dipolar cycloadditions of the C-(3-indolyl)-N-phenylnitrone with a variety of olefinic and allenic dipolarophiles under microwave irradiation
Surinderjit Singh Bhella et al.
TETRAHEDRON (2009)
Rational design of highly active and selective ligands for the α5β1 integrin receptor
Dominik Heckmann et al.
CHEMBIOCHEM (2008)
ANTI-ADHESION evolves to a promising therapeutic concept in oncology
R. Schmidmaier et al.
CURRENT MEDICINAL CHEMISTRY (2008)
Synthesis of Ethyl 5-Hydroxyisoxazolidine-4-carboxylates via Michael Addition/Intramolecular Hemiketalisation
Fides Benfatti et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2008)
Integrin-associated proteins as potential therapeutic targets
Joseph M. Cantor et al.
IMMUNOLOGICAL REVIEWS (2008)
Multi-target-directed ligands to combat neurodegenerative diseases
Andrea Cavalli et al.
JOURNAL OF MEDICINAL CHEMISTRY (2008)
Transcriptional activation of human mu-opioid receptor gene by insulin-like growth factor-I in neuronal cells is modulated by the transcription factor REST
Andrea Bedini et al.
JOURNAL OF NEUROCHEMISTRY (2008)
Molecular imaging in drug development
Juergen K. Willmann et al.
NATURE REVIEWS DRUG DISCOVERY (2008)
Lewis Acid Induced Highly Regioselective Synthesis of a New Class of Substituted Isoxazolidines
Fides Benfatti et al.
SYNLETT (2008)
Diastereoselective synthesis of D-xylo-isoxazolidinyl nucleosides
Eva Hyrosova et al.
TETRAHEDRON (2008)
Integrins in angiogenesis and lymphangiogenesis
Christie J. Avraamides et al.
NATURE REVIEWS CANCER (2008)
Cell adhesion molecules: Potential therapeutic & diagnostic implications
Shaker A. Mousa
MOLECULAR BIOTECHNOLOGY (2008)
Anti-cancer therapies targeting the tumor stroma
Valeska Hofmeister et al.
CANCER IMMUNOLOGY IMMUNOTHERAPY (2008)
Synthesis and biological evaluation of non-peptide αvβ3/α5β1 integrin dual antagonists containing 5,6-dihydropyridin-2-one scaffolds
Fides Benfatti et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2007)
Alpha-v integrins as therapeutic targets in oncology
Jeffrey A. Nemeth et al.
CANCER INVESTIGATION (2007)
Transcriptional up-regulation in cells mediated by a small molecule
Steven P. Rowe et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2007)
Enantioselectively organocatalytic Michael addition of ketones to alkylidene malonates
Chun-Li Cao et al.
JOURNAL OF ORGANIC CHEMISTRY (2007)
Use of antibody as carrier of oligomers of peptidomimetic αvβ3 antagonist to target tumor-induced neovasculature
In Soo Shin et al.
BIOCONJUGATE CHEMISTRY (2007)
Fragments, network biology and designing multiple ligands
Richard Morphy et al.
DRUG DISCOVERY TODAY (2007)
Nonpeptide integrin antagonists: RGD mimetics incorporating substituted azabicycloalkanes as amino acid replacements
Leonardo Manzoni et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2007)
The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands
Sylwia Urman et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2007)
Probing integrin selectivity: Rational design of highly active and selective ligands for the alpha 5 beta 1 and alpha v beta 3 integrin receptor
Dominik Heckmann et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2007)
The scaffold tree - Visualization of the scaffold universe by hierarchical scaffold classification
Ansgar Schuffenhauer et al.
JOURNAL OF CHEMICAL INFORMATION AND MODELING (2007)
New concepts regarding focal promotion of cell migration adhesion kinase and proliferation
Braden D. Cox et al.
JOURNAL OF CELLULAR BIOCHEMISTRY (2006)
Ligand binding analysis for human α5β1 integrin:: Strategies for designing new α5β1 integrin antagonists
L Marinelli et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
Heterocyclic and phenyl double-bond-locked combretastatin analogues possessing potent apoptosis-inducing activity in HL60 and in MDR cell lines
D Simoni et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
The integrin α5β1 regulates αvβ3-mediated extracellular signal-regulated kinase activation
DP Ly et al.
JOURNAL OF SURGICAL RESEARCH (2005)
Dual antagonists of integrins
K Nadrah et al.
CURRENT MEDICINAL CHEMISTRY (2005)
Non peptidic alpha(V)beta(3) antagonists: Recent developments
B Cacciari et al.
CURRENT MEDICINAL CHEMISTRY (2005)
A catalytic and iterative route to β-substituted esters via highly enantioselective conjugate addition of dimethylzinc to unsaturated malonates
J Schuppan et al.
CHEMICAL COMMUNICATIONS (2004)
Synthesis and biological evaluation of nonpeptide integrin antagonists containing spirocyclic scaffolds
JM Smallheer et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)
A concise approach to structurally diverse β-amino acids
AR Minter et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2003)
A novel RGD antagonist that targets both αvβ3 and α5β1 induces apoptosis of angiogenic endothelial cells on type I collagen
K Meerovitch et al.
VASCULAR PHARMACOLOGY (2003)
Enantioselective synthesis of aziridine 2,2-dicarboxylates. Part 1: Copper(II)-bisoxazoline complex-catalysed Michael reaction on alkylidene malonates
G Cardillo et al.
TETRAHEDRON-ASYMMETRY (2002)
Latent production of angiotensin I-converting enzyme inhibitors from buckwheat protein
CH Li et al.
JOURNAL OF PEPTIDE SCIENCE (2002)
Crystal structure of the extracellular segment of integrin αVβ3 in complex with an Arg-Gly-Asp ligand
JP Xiong et al.
SCIENCE (2002)
Non-peptide αvβ3 antagonists.: Part 3:: Identification of potent RGD mimetics incorporating novel β-amino acids as aspartic acid replacements
PJ Coleman et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2002)
Integrin activation controls metastasis in human breast cancer
B Felding-Habermann et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2001)
Catalytic enantioselective alkylation of heteroaromatic compounds using alkylidene malonates
W Zhuang et al.
CHEMICAL COMMUNICATIONS (2001)
Regulation of integrin αvβ3-mediated endothelial cell migration and angiogenesis by integrin α5β1 and protein kinase A
S Kim et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2000)
Enantioselective Lewis acid catalyzed Michael reactions of alkylidene malonates.: Catalysis by C2-symmetric bis(oxazoline) copper(II) complexes in the synthesis of chiral, differentiated glutarate esters
DA Evans et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2000)
Stereodivergent approaches to the synthesis of isoxazolidine analogues of α-amino acid nucleosides.: Total synthesis of isoxazolidinyl deoxypolyoxin C and uracil polyoxin C
P Merino et al.
JOURNAL OF ORGANIC CHEMISTRY (2000)
Regulation of angiogenesis in vivo by ligation of integrin α5β1 with the central cell-binding domain of fibronectin
S Kim et al.
AMERICAN JOURNAL OF PATHOLOGY (2000)