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Mechanism-based profiling of enzyme families
Michael J. Evans et al.
CHEMICAL REVIEWS (2006)
Novel selective inhibitors of neutral endopeptidase for the treatment of female sexual arousal disorder. Synthesis and activity of functionalized glutaramides
David C. Pryde et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Click chemistry in a supramolecular environment:: Stabilization of organogels by copper(I)-catalyzed azide-alkyne [3+2] cycloaddition
David D. Diaz et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
A click approach to unprotected glycodendrimers
E Fernandez-Megia et al.
MACROMOLECULES (2006)
Catalytic click rotaxanes:: A substoichiometric metal-template pathway to mechanically interlocked architectures
V Aucagne et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
Rapid synthesis of triazole-modified resveratrol analogues via click chemistry
F Pagliai et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Syntheses and biological activity of bisdaunorubicins
GS Zhang et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2006)
Rationally designed nucleoside antibiotics that inhibit siderophore biosynthesis of Mycobacterium tuberculosis
RV Somu et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Cu-I-catalyzed alkyne-azide click cycloadditions from a mechanistic and synthetic perspective
VD Bock et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2006)
Microtiter plate based chemistry and in situ screening: a useful approach for rapid inhibitor discovery
A Brik et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2006)
Click chemistry: a new facile and efficient strategy for preparation of functionalized HPLC packings
Zhimou Guo et al.
CHEMICAL COMMUNICATIONS (2006)
The chemical modification of liposome surfaces via a copper-mediated [3+2] azide-alkyne cycloaddition monitored by a colorimetric assay
Silvia Cavalli et al.
CHEMICAL COMMUNICATIONS (2006)
Click chemistry by microcontact printing
Dorota I. Rozkiewicz et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2006)
Advances in cycloaddition polymerizations
GW Goodall et al.
CHEMICAL SOCIETY REVIEWS (2006)
Azide/alkyne-click reactions: Applications in material science and organic synthesis
Wolfgang H. Binder et al.
CURRENT ORGANIC CHEMISTRY (2006)
New prospects for the grafting of functional groups onto aliphatic polyesters. Ring-opening polymerization of alpha- or gamma-substituted epsilon-caprolactone followed by chemical derivatization of the substituents
Philippe Lecomte et al.
MACROMOLECULAR SYMPOSIA (2006)
Protein semi-synthesis: New proteins for functional and structural studies
T Durek et al.
BIOMOLECULAR ENGINEERING (2005)
Accelerated bioorthogonal conjugation: A practical method for the Ligation of diverse functional molecules to a polyvalent virus scaffold
S Sen Gupta et al.
BIOCONJUGATE CHEMISTRY (2005)
Synthesis, characterization and antimicrobial activity of some substituted 1,2,3-triazoles
BS Holla et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2005)
4-Aryl-1,2,3-triazole: A novel template for a reversible methionine aminopeptidase 2 inhibitor, optimized to inhibit angiogenesis in vivo
LS Kallander et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
The convergence of synthetic organic and polymer chemistries
CJ Hawker et al.
SCIENCE (2005)
High-yielding microwave-assisted synthesis of triazole-linked glycodendrimers by copper-catalyzed [3+2] cycloaddition
JAF Joosten et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2005)
Benzoyl and/or benzyl substituted 1,2,3-triazoles as potassium channel activators. VIII
V Calderone et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2005)
Toward semisynthetic lipoproteins by convergent strategies based on click and Ligation chemistry
HJ Musiol et al.
CHEMBIOCHEM (2005)
Identification of 4-substituted 1,2,3-triazoles as novel oxazolidinone antibacterial agents with reduced activity against monoamine oxidase A
F Reck et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
Synthetic applications of aliphatic unsaturated alpha-H-alpha-amino acids
J Kaiser et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2005)
Virus-glycopolymer conjugates by copper(I) catalysis of atom transfer radical polymerization and azide-alkyne cycloaddition
S Sen Gupta et al.
CHEMICAL COMMUNICATIONS (2005)
Discovery of novel heteroarylazoles that are metabotropic glutamate subtype 5 receptor antagonists with anxiolytic activity
J Roppe et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
Presentation and detection of azide functionality in bacterial cell surface proteins
AJ Link et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2004)
Discovery and characterization of catalysts for azide-alkyne cycloaddition by fluorescence quenching
WG Lewis et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2004)
A fluorogenic probe for the copper(I)-catalyzed azide-alkyne ligation reaction:: Modulation of the fluorescence emission via 3(n,π*)-1(π,π*) inversion
Z Zhou et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2004)
Heterocyclic peptide backbone modifications in an α-helical coiled coil
WS Horne et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2004)
A fluorogenic 1,3-dipolar cycloaddition reaction of 3-azidocoumarins and acetylenes
K Sivakumar et al.
ORGANIC LETTERS (2004)
The Staudinger ligation - A gift to chemical biology'
M Kohn et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2004)
Expanded utility of the native chemical ligation reaction
DSY Yeo et al.
CHEMISTRY-A EUROPEAN JOURNAL (2004)
Pseudoamide-type pyrrolidine and pyrrolizidine glycomimetics and their inhibitory activities against glycosidases
MI García-Moreno et al.
JOURNAL OF ORGANIC CHEMISTRY (2004)
Combinatorial library of peptidotriazoles:: Identification of [1,2,3]-triazole inhibitors against a recombinant Leishmania mexicana cysteine protease
CW Tornoe et al.
JOURNAL OF COMBINATORIAL CHEMISTRY (2004)
The growing impact of click chemistry on drug discovery
HC Kolb et al.
DRUG DISCOVERY TODAY (2003)
Azide-alkyne coupling:: A powerful reaction for bioconjugate chemistry
R Breinbauer et al.
CHEMBIOCHEM (2003)
Synthesis of 1,2,3-triazolo-carbanucleoside analogues of ribavirin targeting an HCV in replicon
Y Saito et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2003)
Mechanism and dynamics of azobenzene photoisomerization
T Schultz et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2003)
Bioconjugation by copper(I)-catalyzed azide-alkyne [3+2] cycloaddition
Q Wang et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2003)
Synthesis and investigation of tuberculosis inhibition activities of some 1,2,3-triazole derivatives
K Dabak et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2003)
Synthesis and structure-affinity relationship investigations of 5-heteroaryl-substituted analogues of the antipsychotic sertindole.: A new class of highly selective α1 adrenoceptor antagonists
T Balle et al.
JOURNAL OF MEDICINAL CHEMISTRY (2003)
Peptidotriazoles on solid phase: [1,2,3]-triazoles by regiospecific copper(I)-catalyzed 1,3-dipolar cycloadditions of terminal alkynes to azides
CW Tornoe et al.
JOURNAL OF ORGANIC CHEMISTRY (2002)
Incorporation of azides into recombinant proteins for chemoselective modification by the Staudinger ligation
KL Kiick et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2002)
Novel 1-hydroxyazole bioisosteres of glutamic acid.: Synthesis, protolytic properties, and pharmacology
TB Stensbol et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Biotransformation reactions of five-membered aromatic heterocyclic rings
DK Dalvie et al.
CHEMICAL RESEARCH IN TOXICOLOGY (2002)
An orally active, water-soluble neurokinin-1 receptor antagonist suitable for both intravenous and oral clinical administration
T Harrison et al.
JOURNAL OF MEDICINAL CHEMISTRY (2001)
Structure-activity relationships of 1,4-dihydro-(1H,4H)-quinoxaline-2,3-diones as N-methyl-D-aspartate (glycine site) receptor antagonists.: 1.: Heterocyclic substituted 5-alkyl derivatives
MJ Fray et al.
JOURNAL OF MEDICINAL CHEMISTRY (2001)
Human β3-adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides
LL Brockunier et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2000)
Cell surface engineering by a modified Staudinger reaction
E Saxon et al.
SCIENCE (2000)