4.3 Article

Evaluation of the endothelin receptor antagonists ambrisentan, darusentan, bosentan, and sitaxsentan as substrates and inhibitors of hepatobiliary transporters in sandwich-cultured human hepatocytes

Related references

Note: Only part of the references are listed.
Article Pharmacology & Pharmacy

Effect of Ketoconazole on the Pharmacokinetic Profile of Ambrisentan

Duncan B. Richards et al.

JOURNAL OF CLINICAL PHARMACOLOGY (2009)

Article Respiratory System

Endothelin receptor antagonists in pulmonary arterial hypertension

J. Dupuis et al.

EUROPEAN RESPIRATORY JOURNAL (2008)

Article Respiratory System

Results of European post-marketing surveillance of bosentan in pulmonary hypertension

M. Humbert et al.

EUROPEAN RESPIRATORY JOURNAL (2007)

Article Pharmacology & Pharmacy

In vitro-in vivo correlation of hepatobiliary drug clearance in humans

G. Ghibellini et al.

CLINICAL PHARMACOLOGY & THERAPEUTICS (2007)

Meeting Abstract Critical Care Medicine

No clinically relevant pharmacokinetic interaction between ambrisentan and sildenafil

Christopher Dufton et al.

CHEST (2006)

Article Cardiac & Cardiovascular Systems

Treatment of pulmonary arterial hypertension with the selective endothelin-A receptor antagonist sitaxsentan

Robyn J. Barst et al.

JOURNAL OF THE AMERICAN COLLEGE OF CARDIOLOGY (2006)

Review Medicine, Research & Experimental

Methods to evaluate biliary excretion of drugs in humans: An updated review

Giulia Ghibellini et al.

MOLECULAR PHARMACEUTICS (2006)

Review Cardiac & Cardiovascular Systems

Ambrisentan, a non-peptide endothelin receptor antagonist

Hartmut Vatter et al.

CARDIOVASCULAR DRUG REVIEWS (2006)

Article Cardiac & Cardiovascular Systems

Ambrisentan therapy for pulmonary arterial hypertension

N Galié et al.

JOURNAL OF THE AMERICAN COLLEGE OF CARDIOLOGY (2005)

Article Respiratory System

Survival with first-line bosentan in patients with primary pulmonary hypertension

VV McLaughlin et al.

EUROPEAN RESPIRATORY JOURNAL (2005)

Article Critical Care Medicine

Sitaxsentan therapy for pulmonary arterial hypertension

RJ Barst et al.

AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE (2004)

Article Gastroenterology & Hepatology

Contribution of mrp2 in alterations of canalicular bile formation by the endothelin antagonist bosentan

L Fouassier et al.

JOURNAL OF HEPATOLOGY (2002)

Article Pharmacology & Pharmacy

Single- and multiple-dose pharmacokinetics of bosentan and its interaction with ketoconazole

PLM van Giersbergen et al.

BRITISH JOURNAL OF CLINICAL PHARMACOLOGY (2002)

Article Medicine, General & Internal

Bosentan therapy for pulmonary arterial hypertension

LJ Rubin et al.

NEW ENGLAND JOURNAL OF MEDICINE (2002)

Article Urology & Nephrology

Renal hemodynamics and pharmacokinetics of bosentan with and without cyclosporine A

I Binet et al.

KIDNEY INTERNATIONAL (2000)