4.7 Article

Carfilzomib can induce tumor cell death through selective inhibition of the chymotrypsin-like activity of the proteasome

Related references

Note: Only part of the references are listed.
Article Biophysics

Selective apoptosis of monocytes and monocyte-derived DCs induced by bortezomib (Velcade)

M. Arpinati et al.

BONE MARROW TRANSPLANTATION (2009)

Article Chemistry, Medicinal

Design and Synthesis of an Orally Bioavailable and Selective Peptide Epoxyketone Proteasome Inhibitor (PR-047)

Han-Jie Zhou et al.

JOURNAL OF MEDICINAL CHEMISTRY (2009)

Review Pharmacology & Pharmacy

Mechanisms of proteasome inhibitor action and resistance in cancer

David J. McConkey et al.

DRUG RESISTANCE UPDATES (2008)

Article Biochemical Research Methods

Immunological methods to quantify and characterize proteasome complexes: Development and application

Matthias Majetschak et al.

JOURNAL OF IMMUNOLOGICAL METHODS (2008)

Article Biochemistry & Molecular Biology

Intermediate-type 20 S proteasomes in HeLa cells: Asymmetric subunit composition, diversity and adaptation

Nicola Klare et al.

JOURNAL OF MOLECULAR BIOLOGY (2007)

Article Multidisciplinary Sciences

Effects of aneuploidy on cellular physiology and cell division in haploid yeast

Eduardo M. Torres et al.

SCIENCE (2007)

Article Biochemistry & Molecular Biology

Importance of the different proteolytic sites of the proteasome and the efficacy of inhibitors varies with the protein substrate

AF Kisselev et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2006)

Article Medicine, General & Internal

Bortezomib or high-dose dexamethasone for relapsed multiple myeloma

PG Richardson et al.

NEW ENGLAND JOURNAL OF MEDICINE (2005)

Article Biochemical Research Methods

Activity probe for in vivo profiling of the specificity of proteasome inhibitor bortezomib

CR Berkers et al.

NATURE METHODS (2005)

Article Biochemistry & Molecular Biology

β2 subunit propeptides influence cooperative proteasome assembly

M De et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2003)

Article Biochemistry & Molecular Biology

Transcriptome analysis of human autosomal trisomy

DR FitzPatrick et al.

HUMAN MOLECULAR GENETICS (2002)

Article Multidisciplinary Sciences

Microarray analysis reveals a major direct role of DNA copy number alteration in the transcriptional program of human breast tumors

JR Pollack et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2002)

Article Biochemistry & Molecular Biology

NF-κB as a therapeutic target in multiple myeloma

T Hideshima et al.

JOURNAL OF BIOLOGICAL CHEMISTRY (2002)

Article Chemistry, Analytical

Validation of immunoassays for bioanalysis: a pharmaceutical industry perspective

JWA Findlay et al.

JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS (2000)