Journal
ORGANIC LETTERS
Volume 3, Issue 17, Pages 2673-2676Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol016254m
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- NIGMS NIH HHS [F31GM20439] Funding Source: Medline
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[GRAPHICS] A new method to produce benzimidazolium salts based on a successive Buchwald-Hartwig amination and ring closure is reported. A variety of different benzimidazolium salts can be prepared using this procedure. Amines that bear an alpha -chiral group undergo the reaction to furnish chiral benzimidazolium salts. The salts that lack a C2 substituent on the heterocycle are readily deprotonated to give nucleophilic carbenes.
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