☆ 4.7 Article

ERβ ligands.: Part 1:: The discovery of ERβ selective ligands which embrace the 4-hydroxy-biphenyl template

BIOORGANIC & MEDICINAL CHEMISTRY (2003)

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Journal

BIOORGANIC & MEDICINAL CHEMISTRY
Volume 11, Issue 16, Pages 3457-3474

Publisher

PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/S0968-0896(03)00303-1

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Categories

Biochemistry & Molecular Biology Chemistry, Medicinal Chemistry, Organic

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The synthesis and structure-activity relationships of a series of simple biphenyls is described. Optimization of the 4-hydroxy-biphenyl template led to compounds with ERP selectivity on the order of 20-70-fold. (C) 2003 Elsevier Ltd. All rights reserved.

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