4.3 Article

A ring expansion strategy in antiviral synthesis: A novel approach to TAK-779

Journal

SYNTHETIC COMMUNICATIONS
Volume 34, Issue 11, Pages 1973-1980

Publisher

MARCEL DEKKER INC
DOI: 10.1081/SCC-120037909

Keywords

ring transformations; amines; suzuki reactions; coupling reaction

Ask authors/readers for more resources

A synthesis of TAK-779 that relies on construction of a key carboxylic acid intermediate by a ring expansion with TMSCHN2 is described.

Authors

I am an author on this paper
Click your name to claim this paper and add it to your profile.

Reviews

Primary Rating

4.3
Not enough ratings

Secondary Ratings

Novelty
-
Significance
-
Scientific rigor
-
Rate this paper

Recommended

No Data Available
No Data Available