4.8 Article

1,2,3-Triazoles as Amide Bond Mimics: Triazole Scan Yields Protease-Resistant Peptidomimetics for Tumor Targeting

Journal

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
Volume 52, Issue 34, Pages 8957-8960

Publisher

WILEY-V C H VERLAG GMBH
DOI: 10.1002/anie.201303108

Keywords

click chemistry; drug delivery; metabolic stabilization; peptidomimetics; radiopharmaceuticals

Funding

  1. Swiss National Science Foundation [132280]
  2. Nora van Meeuwen-Hfliger Foundation

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