4.8 Article

Copper-Catalyzed Domino Cycloaddition/C-N Coupling/Cyclization/(C-H Arylation): An Efficient Three-Component Synthesis of Nitrogen Polyheterocycles

Journal

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
Volume 52, Issue 42, Pages 10992-10996

Publisher

WILEY-V C H VERLAG GMBH
DOI: 10.1002/anie.201305970

Keywords

amidation; CH arylation; copper catalysis; heterocycles; multicomponent reactions

Funding

  1. Amgen Therapeutic Discovery

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