Related references
Note: Only part of the references are listed.An overview of the key routes to the best selling 5-membered ring heterocyclic pharmaceuticals
Marcus Baumann et al.
BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY (2011)
Imidazo[1,2-a]pyridin-3-amines as potential HIV-1 non-nucleoside reverse transcriptase inhibitors
Moira L. Bode et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2011)
Evidence for in Situ Catalyst Modification during the Pd-Catalyzed Conversion of Aryl Triflates to Aryl Fluorides
Thomas J. Maimone et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2011)
Palladium-catalyzed coupling of functionalized primary and secondary amines with aryl and heteroaryl halides: two ligands suffice in most cases
Debabrata Maiti et al.
CHEMICAL SCIENCE (2011)
Discovery of imidazo[1,2-a]pyrazine-based Aurora kinase inhibitors
David B. Belanger et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Discovery of a Potent, Injectable Inhibitor of Aurora Kinases Based on the Imidazo-[1,2-a]-Pyrazine Core
Tao Yu et al.
ACS MEDICINAL CHEMISTRY LETTERS (2010)
Pyrazole NNRTIs 4: Selection of UK-453,061 (lersivirine) as a Development Candidate
Charles E. Mowbray et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
Pd-Catalyzed N-Arylation of Secondary Acyclic Amides: Catalyst Development, Scope, and Computational Study
Jacqueline D. Hicks et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2009)
An efficient system for the Pd-catalyzed cross-coupling of amides and aryl chlorides
Brett P. Fors et al.
TETRAHEDRON (2009)
A highly active catalyst for Pd-catalyzed amination reactions: Cross-coupling reactions using aryl mesylates and the highly selective monoarylation of primary amines using aryl chlorides
Brett P. Fors et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2008)
Highly reactive, general and long-lived catalysts for palladium-catalyzed amination of heteroaryl and aryl chlorides, bromides, and iodides: Scope and structure-activity relationships
Qilong Shen et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2008)
Pd-catalyzed amidations of aryl chlorides using monodentate biaryl phosphine ligands: A kinetic, computational, and synthetic investigation
Takashi Ikawa et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2007)
Lewis acid acceleration of C-N bond-forming reductive elimination from heteroarylpalladium complexes and catalytic amidation of heteroaryl bromides
Qilong Shen et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2007)
Recent progress in the pharmacology of imidazo[1,2-a]pyridines
Cecile Enguehard-Gueiffier et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2007)
Significantly improved method for the Pd-catalyzed coupling of phenols with aryl halides: Understanding ligand effects
Carlos H. Burgos et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2006)
The histamine H3 receptor:: From gene cloning to H3 receptor drugs
R Leurs et al.
NATURE REVIEWS DRUG DISCOVERY (2005)
Highly reactive, general, and long-lived catalysts for coupling heteroaryl and aryl chlorides with primary nitrogen nucleophiles
QL Shen et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2005)
Efficient Pd-catalyzed amination of heteroaryl halides
MD Charles et al.
ORGANIC LETTERS (2005)
Imidazo[1,2-α]pyridines.: Part 2:: SAR and optimisation of a potent and selective class of cyclin-dependent kinase inhibitors
KF Byth et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)
Imidazo[1,2-b]pyridazines:: a potent and selective class of cyclin-dependent kinase inhibitors
KF Byth et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)
Understanding the coupling of heteroaromatic substrates: Synthesis, structures, and reductive eliminations of heteroarylpalladium amido complexes
MW Hooper et al.
ORGANOMETALLICS (2003)
Scope and mechanism of palladium-catalyzed amination of five-membered heterocyclic halides
MW Hooper et al.
JOURNAL OF ORGANIC CHEMISTRY (2003)
Pd-catalyzed intermolecular amidation of aryl halides: The discovery that xantphos can be trans-chelating in a palladium complex
JJ Yin et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2002)
Palladium-catalyzed intermolecular coupling of aryl halides and amides
JJ Yin et al.
ORGANIC LETTERS (2000)