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Flexible strategy for differentially 3,5-disubstituted 4-oxypyridin-2(1H)-ones based on site-selective Pd-catalyzed cross-coupling reactions
David Conreaux et al.
ORGANIC LETTERS (2007)
An epoxidation approach to a chiral lactone: Application of the Shi epoxidation
David J. Ager et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2007)
Aryl-aryl bond formation by transition-metal-catalyzed direct arylation
Dino Alberico et al.
CHEMICAL REVIEWS (2007)
A new family of biisoquinoline chelates
Fabien Durola et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2007)
3,4,5-Triarylisothiazoles via C-C coupling chemistry
Irene C. Christoforou et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2007)
Direct transition metal-catalyzed functionalization of heteroaromatic compounds
Ilya V. Seregin et al.
CHEMICAL SOCIETY REVIEWS (2007)
Regioselective (site-selective) functionalisation of unsaturated halogenated nitrogen, oxygen and sulfur heterocycles by Pd-catalysed cross-couplings and direct arylation processes
Ian J. S. Fairlamb
CHEMICAL SOCIETY REVIEWS (2007)
Organotrifluoroborates: Protected boronic acids that expand the versatility of the Suzuki coupling reaction
Gary A. Molander et al.
ACCOUNTS OF CHEMICAL RESEARCH (2007)
Continuous-flow Suzuki-Miyaura reaction in supercritical carbon dioxide
Gary A. Leeke et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2007)
Synthesis of 2,2 '-bipyridyl-type compounds via the Suzuki-Miyaura cross-coupling reaction
Nicholas A. Jones et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2007)
Macroporous monolith supports for continuous flow capillary microreactors
Katrina F. Bolton et al.
TETRAHEDRON LETTERS (2006)
Regioselective cross-coupling reactions and nucleophilic aromatic substitutions on a 5,7-dichloro-pyrido[4,3-d]pyrimidine scaffold
Mi-Yeon Jang et al.
TETRAHEDRON LETTERS (2006)
3-(Indol-2-yl)indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6
Mark E. Fraley et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2006)
Regioselectivity in alkenyl(aryl)-heteroaryl Suzuki cross-coupling reactions of 2,4-dibromopyridine.: A synthetic and mechanistic study
Cristina Sicre et al.
TETRAHEDRON (2006)
Regioselective couplings of dibromopyrrole esters
Scott T. Handy et al.
SYNTHESIS-STUTTGART (2006)
Synthesis of a naphthyridone p38 MAP kinase inhibitor
John Y. L. Chung et al.
JOURNAL OF ORGANIC CHEMISTRY (2006)
Regioselective suzuki coupling on pyridinium N-(3,5-dibromoheteroar-2-yl)aminides
M. Jose Reyes et al.
TETRAHEDRON LETTERS (2006)
Total synthesis of (R)-telomestatin
Takayuki Doi et al.
ORGANIC LETTERS (2006)
Tandem Diels-Alder cycloadditions of 2-pyrone-5-acrylates for the efficient synthesis of novel tetracyclolactones
Soo-Im Chung et al.
JOURNAL OF ORGANIC CHEMISTRY (2006)
Six-step synthesis of (S)-brevicolline from (S)-nicotine
Florence F. Wagner et al.
ORGANIC LETTERS (2006)
Cross-coupling reactions on azoles with two and more heteroatoms
Michael Schnurch et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2006)
Efficient synthesis of a highly selective NPY-5 receptor antagonist: A drug candidate for the treatment of obesity
Takahiro Itoh et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2006)
Selected patented cross-coupling reaction technologies
Jean-Pierre Corbet et al.
CHEMICAL REVIEWS (2006)
Microwave-assisted, efficient and regioselective Pd-catalyzed C-phenylation of halopyrimidines
Susana Conde Ceide et al.
TETRAHEDRON LETTERS (2006)
Microwave-assisted Suzuki coupling reactions with an encapsulated palladium catalyst for batch and continuous-flow transformations
Ian R. Baxendale et al.
CHEMISTRY-A EUROPEAN JOURNAL (2006)
Halogenated 2′-chlorobithiazoles via Pd-catalyzed cross-coupling reactions
P Stanetty et al.
JOURNAL OF ORGANIC CHEMISTRY (2006)
An efficient multikilogram synthesis of ABT-963: A selective COX-2 inhibitor
FAJ Kerdesky et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2006)
A highly regioselective synthesis of 2-aryl-6-chlorobenzothiazoles employing microwave-promoted Suzuki-Miyaura coupling reaction
Y Heo et al.
TETRAHEDRON LETTERS (2006)
Regioselective dicouplings: Application to differentially substituted pyrroles
ST Handy et al.
ORGANIC LETTERS (2006)
First cross-coupling reactions on halogenated 1H-1,2,4-triazole nucleosides
S Wille et al.
TETRAHEDRON (2006)
On the nature of the active species in palladium catalyzed Mizoroki-Heck and Suzuki-Miyaura couplings - Homogeneous or heterogeneous catalysis, a critical review
NTS Phan et al.
ADVANCED SYNTHESIS & CATALYSIS (2006)
Imidazo[1,2-a]pyrimidines as functionally selective GABAA ligands
WP Blackaby et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2006)
Mild aerobic oxidative palladium (II) catalyzed C-H bond functionalization: Regioselective and switchable C-H alkenylation and annulation of pyrroles
EM Beck et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
A highly regioselective amination of 6-aryl-2,4-dichloropyrimidine
ZH Peng et al.
ORGANIC LETTERS (2006)
New chiral tridentate ligands for asymmetric catalysis
K Murtagh et al.
PURE AND APPLIED CHEMISTRY (2006)
Total synthesis of lamellarins D, L, and N
N Fujikawa et al.
TETRAHEDRON (2006)
A simple guide for predicting regioselectivity in the coupling of polyhaloheteroaromatics
ST Handy et al.
CHEMICAL COMMUNICATIONS (2006)
Palladium-catalyzed alkylation of aryl C-H bonds with sp3 organotin reagents using benzoquinone as a crucial promoter
X Chen et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
The regioselective synthesis of aryl pyrroles
Jason A. Smith et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2006)
Insights into the mechanism of the site-selective sequential palladium-catalyzed cross-coupling reactions of dibromothiophenes/dibromothiazoles and arylboronic acids. Synthesis of PPAR beta/delta agonists
Raquel Pereira et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2006)
Synthesis of the PPAR beta/delta-selective agonist GW501516 and C4-thiazole-substituted analogs
R Pereira et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2006)
Sterically non-hindering endocyclic ligands of the bi-isoquinoline family
F Durola et al.
CHEMICAL COMMUNICATIONS (2006)
A versatile method for Suzuki cross-coupling reactions of nitrogen heterocycles
N Kudo et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2006)
Process development and large-scale synthesis of a PDE4 inhibitor
DA Conlon et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2006)
The synthesis of substituted phenylpyrimidines via Suzuki coupling reactions
TJ Delia et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2006)
Effective methods for introducing some aryl and heteroaryl substituent onto 1-azaazulene nuclei
N Abe et al.
HETEROCYCLES (2005)
Polymer-supported palladium catalysed Suzuki-Miyaura reactions in batch and a mini-continuous flow reactor system
NTS Phan et al.
TETRAHEDRON (2005)
Non-conventional methodologies for transition-metal catalysed carbon-carbon coupling: a critical overview. Part 1: The Heck reaction
F Alonso et al.
TETRAHEDRON (2005)
Efficient synthesis of a trisubstituted 1,6-naphthyridone from acetonedicarboxylate and regioselective Suzuki arylation
JYL Chung et al.
JOURNAL OF ORGANIC CHEMISTRY (2005)
Convergent stereoselective synthesis of the visual pigment A2E
C Sicre et al.
ORGANIC LETTERS (2005)
Regioselective lithium-halogen exchange and palladium-catalyzed cross-coupling reactions of 2,4-dihaloquinolines
DL Comins et al.
TETRAHEDRON LETTERS (2005)
Controlled monoarylation of dibromoarenes in water with a polymeric palladium catalyst
Y Uozumi et al.
SYNLETT (2005)
Synthesis, resolution and racemisation studies of new tridentate ligands for asymmetric catalysis
BA Sweetman et al.
TETRAHEDRON LETTERS (2005)
Expanding the substitution pattern of 2(1H)-pyrazinones via Suzuki and Heck reactions
R Azzam et al.
TETRAHEDRON (2005)
Application of cross-coupling and metalation chemistry of 3(2H)-pyridazinones to fungicide and herbicide discovery
TM Stevenson et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2005)
Synthesis of pyrazine alealoids from Botryllus leachi.: Diazines 43
F Buron et al.
JOURNAL OF ORGANIC CHEMISTRY (2005)
Regioselective cross-coupling reactions of multiple halogenated nitrogen-, oxygen-, and sulfur-containing heterocycles
S Schröter et al.
TETRAHEDRON (2005)
Carbon-carbon bonding made easy
A Suzuki
CHEMICAL COMMUNICATIONS (2005)
In vivo optical Imaging of amyloid aggregates in brain: Design of fluorescent markers
EE Nesterov et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2005)
Palladium-catalyzed cross-coupling reactions in total synthesis
KC Nicolaou et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2005)
Efficient batch and continuous flow Suzuki cross-coupling reactions under mild conditions, catalysed by polyurea-encapsulated palladium (II) acetate and tetra-n-butylammonium salts
CKY Lee et al.
CHEMICAL COMMUNICATIONS (2005)
Palladium-catalyzed intermolecular alkenylation of indoles by solvent-controlled regioselective C-H functionalization
NP Grimster et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2005)
Directed palladation: fine tuning permits the catalytic 2-alkenylation of indoles
E Capito et al.
CHEMICAL COMMUNICATIONS (2005)
Comparison of the Suzuki cross-coupling reactions of 4,7-dichloroquinoline and 7-chloro-4-iodoquinoline with arylboronic acids using phosphine-free palladium catalysis in water
RW Friesen et al.
CANADIAN JOURNAL OF CHEMISTRY (2004)
Regioselectivity in cross-coupling reactions of 2,6,8-trichloro-9-(tetrahydropyran-2-yl)purine: Synthesis of 2,6,8-trisubstituted purine bases
M Hocek et al.
SYNTHESIS-STUTTGART (2004)
5-Pyrimidylboronic acid and 2-methoxy-5-pyrimidylboronic acid: new heteroarylpyrimidine derivatives via Suzuki cross-coupling reactions
N Saygili et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2004)
The synthesis and properties of solution processable red-emitting phosphorescent dendrimers
MJ Frampton et al.
JOURNAL OF MATERIALS CHEMISTRY (2004)
Isolation and structure of antagonists of chemokine receptor (CCR5)
H Jayasuriya et al.
JOURNAL OF NATURAL PRODUCTS (2004)
Microwave-assisted Suzuki reactions in a continuous flow capillary reactor
H Ping et al.
APPLIED CATALYSIS A-GENERAL (2004)
A novel antimicrobial indolizinium alkaloid from Aniba panurensis
P Klausmeyer et al.
JOURNAL OF NATURAL PRODUCTS (2004)
Large-scale synthesis of the anti-cancer marine natural product (+)-discodermolide. Part 4: Preparation of fragment C7-24
SJ Mickel et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2004)
An efficient two-step total synthesis of the quaterpyridine nemertelline
A Bouillon et al.
JOURNAL OF ORGANIC CHEMISTRY (2003)
Bioactive marine metabolites, Part 124.: Ageladine A:: An antiangiogenic matrixmetalloproteinase inhibitor from the marine sponge Agelas nakamurai
M Fujita et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2003)
Successive replacement of halogen atoms in 4,6-dihaloquinolines in cross-coupling reactions with arylboronic acids catalyzed by palladium and nickel complexes
IP Beletskaya et al.
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY (2003)
Regiospecific Suzuki coupling of 3,5-dichloroisothiazole-4-carbonitrile
IC Christoforou et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2003)
Efficient synthesis of 2-aryl-6-chloronicotinamides via PXPd2-catalyzed regioselective Suzuki coupling
W Yang et al.
ORGANIC LETTERS (2003)
14C-labeled and large-scale synthesis of the angiotensin-(1-7)-receptor agonist AVE 0991 by cross-coupling reactions
V Derdau et al.
JOURNAL OF ORGANIC CHEMISTRY (2003)
Short and flexible route to 3,4-diarylpyrrole marine alkaloids: syntheses of permethyl storniamide A, ningalin B, and lamellarin G trimethyl ether
M Iwao et al.
TETRAHEDRON LETTERS (2003)
The synthesis of OSU 6162: Efficient, large-scale implementation of a Suzuki coupling
MF Lipton et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2003)
Practical asymmetric synthesis of a potent cathepsin K inhibitor. Efficient palladium removal following Suzuki coupling
CY Chen et al.
JOURNAL OF ORGANIC CHEMISTRY (2003)
A convenient synthesis of unsymmetrically substituted terphenyls of biologically active stilbenes via a double Suzuki cross-coupling protocol
D Simoni et al.
TETRAHEDRON LETTERS (2003)
An unusual dehalogenation in the Suzuki coupling of 4-bromopyrrole-2-carboxylates
ST Handy et al.
TETRAHEDRON LETTERS (2003)
The palladium-catalyzed cross-coupling reactions of 3-chloro-4-halogeno-1,2,5-thiadiazoles
A Merschaert et al.
HETEROCYCLES (2003)
Chemistry and biology of khafrefungin. Large-scale synthesis, design, and structure-activity relationship of khafrefungin, an antifungal agent
M Nakamura et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2003)
Preparing functional bis(indole) pyrazine by stepwise cross-coupling reactions: An efficient method to construct the skeleton of dragmacidin D
CG Yang et al.
JOURNAL OF ORGANIC CHEMISTRY (2002)
Regioselective Stille coupling reactions of 3,5-dibromo-2-pyrone with various aryl and vinyl stannanes
WS Kim et al.
TETRAHEDRON LETTERS (2002)
Suzuki-miyaura cross-coupling reactions of potassium alkenyltrifluoroborates
GA Molander et al.
JOURNAL OF ORGANIC CHEMISTRY (2002)
Recent applications of the Suzuki-Miyaura cross-coupling reaction in organic synthesis
S Kotha et al.
TETRAHEDRON (2002)
Synthesis of 4-aryl-5-hydroxy- and 5-aryl-4-hydroxypyridazin-3(2H)-ones and their use in the preparation of 4,5-diarylpyridazin-3(2H)-ones and hitherto unknown isochromeno[3,4-d]pyridazinediones
BUW Maes et al.
TETRAHEDRON (2002)
The successive substitution of halogens in 4-chloro-6-iodoquinoline by aryl groups in cross-coupling reactions with arylboronic acids
AV Tsvetkov et al.
TETRAHEDRON LETTERS (2002)
Ru-, Rh-, and Pd-catalyzed C-C bond formation involving C-H activation and addition on unsaturated substrates: Reactions and mechanistic aspects
V Ritleng et al.
CHEMICAL REVIEWS (2002)
A study for palladium-catalyzed chemoselective vinylation at C-3 position of 4-bromo-1-tosylindole
Y Yokoyama et al.
HETEROCYCLES (2002)
Arylated pyridines: Suzuki reactions of O-substituted 2,6-dihalogenated-3-hydroxypyridines
GM Chapman et al.
JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 (2002)
Ring fluorinated thiophenes: applications to liquid crystal synthesis
AA Kiryanov et al.
TETRAHEDRON LETTERS (2001)
Arylation of halogenated pyrimidines via a Suzuki coupling reaction
JM Schomaker et al.
JOURNAL OF ORGANIC CHEMISTRY (2001)
Regioselective palladium-catalyzed cross-coupling reactions in the synthesis of novel 2,3-disubstituted thiophene derivatives
R Pereira et al.
TETRAHEDRON (2001)
Palladium-catalyzed carbonylative cross-coupling reactions of pyridine halides and aryl boronic acids:: a convenient access to α-pyridyl ketones
S Couve-Bonnaire et al.
TETRAHEDRON LETTERS (2001)
Concise formation of 4-benzyl piperidines and related derivatives using a Suzuki protocol
S Vice et al.
JOURNAL OF ORGANIC CHEMISTRY (2001)
Suzuki reactions on chloropyridazinones:: an easy approach towards arylated 3(2H)-pyridazinones
BUW Maes et al.
TETRAHEDRON (2001)
Bis-Suzuki reactions of 2,3-dihaloindoles. A convenient synthesis of 2,3-diarylindoles
YB Liu et al.
TETRAHEDRON LETTERS (2000)
Reversible diastereoselective photocyclization of a diarylethene in a single-crystalline phase
T Kodani et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2000)
Total synthesis of ningalin B utilizing a heterocyclic azadiene Diels-Alder reaction and discovery of a new class of potent multidrug resistant (MDR) reversal agents
DL Boger et al.
JOURNAL OF ORGANIC CHEMISTRY (2000)
Biosynthesis of pyrrolnitrin and other phenylpyrrole derivatives by bacteria
KH van Pee et al.
NATURAL PRODUCT REPORTS (2000)