4.7 Article

Palladium-Catalyzed Annulation of 2-(1-Alkynyl)benzenamines with Disulfides: Synthesis of 3-Sulfenylindoles

Journal

ADVANCED SYNTHESIS & CATALYSIS
Volume 351, Issue 16, Pages 2615-2618

Publisher

WILEY-V C H VERLAG GMBH
DOI: 10.1002/adsc.200900055

Keywords

2-(1-alkynyl)benzenamines; annulation; disulfides; palladium; 3-sulfenylindoles

Funding

  1. National Natural Science Foundation of China [20872112]
  2. Zhejiang Provincial Natural Science Foundation of China [Y407116, Y407079, Y4080027]
  3. Program for New Century Excellent Talents in University [NCET-06-0711]

Ask authors/readers for more resources

3-Sulfenylindoles can be efficiently prepared in moderate to good yields from 2-(1-alkynyl)benzenamines and disulfides using the palladium/air catalytic systems. The study also provides a useful route to the synthesis of fipronil analogues.

Authors

I am an author on this paper
Click your name to claim this paper and add it to your profile.

Reviews

Primary Rating

4.7
Not enough ratings

Secondary Ratings

Novelty
-
Significance
-
Scientific rigor
-
Rate this paper

Recommended

No Data Available
No Data Available