Related references
Note: Only part of the references are listed.Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode
Lisa M. Miller et al.
JOURNAL OF MEDICINAL CHEMISTRY (2017)
Redox-Neutral α-Arylation of Alkyl Nitriles with Aryl Sulfoxides: A Rapid Electrophilic Rearrangement
Li Shang et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2017)
Recent progress in transition-metal-catalyzed enantioselective indole functionalizations
Jing-Biao Chen et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2017)
Metal-free O-H/C-H difunctionalization of phenols by o-hydroxyarylsulfonium salts in water
Dengfeng Chen et al.
CHEMICAL SCIENCE (2017)
Regioselective synthesis of C3 alkylated and arylated benzothiophenes
Harry J. Shrives et al.
NATURE COMMUNICATIONS (2017)
Recent Advances in Catalytic C(sp2)-H Allylation Reactions
Neeraj Kumar Mishra et al.
ACS CATALYSIS (2017)
Cascades of Interrupted Pummerer Reaction-Sigmatropic Rearrangement
Hideki Yorimitsu
CHEMICAL RECORD (2017)
Transition metal-catalyzed site- and regio-divergent C-H bond functionalization
Lucy Ping et al.
CHEMICAL SOCIETY REVIEWS (2017)
A conjugate Lewis base-Bronsted acid catalyst for the sulfenylation of nitrogen containing heterocycles under mild conditions
Christopher J. Nalbandian et al.
CHEMICAL COMMUNICATIONS (2017)
Cs2CO3-Catalyzed Aerobic Oxidative Cross-Dehydrogenative Coupling of Thiols with Phosphonates and Arenes
Song Song et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2017)
An Asymmetric Redox Arylation: Chirality Transfer from Sulfur to Carbon through a Sulfonium [3,3]-Sigmatropic Rearrangement
Dainis Kaldre et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2017)
Desulfination as an Emerging Strategy in Palladium-Catalyzed C-C Coupling Reactions
Dirk H. Ortgies et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2016)
Manganese(I)-Catalyzed Substitutive C-H Allylation
Weiping Liu et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2016)
Azulenesulfonium Salts: Accessible, Stable, and Versatile Reagents for Cross-Coupling
Paul Cowper et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2016)
C-H Coupling Reactions Directed by Sulfoxides: Teaching an Old Functional Group New Tricks
Alexander P. Pulis et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2016)
Metal-free C-H thioarylation of arenes using sulfoxides: a direct, general diaryl sulfide synthesis
Jose A. Fernandez-Salas et al.
CHEMICAL COMMUNICATIONS (2016)
Radical-promoted site-specific cross dehydrogenative coupling of heterocycles with nitriles
Zhong-Quan Liu et al.
CHEMICAL COMMUNICATIONS (2016)
Synthesis and preliminary evaluation of 3-thiocyanato-1H-indoles as potential anticancer agents
Margiani P. Fortes et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
Catalytic Synthesis of 3-Thioindoles Using Bunte Salts as Sulfur Sources under Metal-Free Conditions
Hong Qi et al.
JOURNAL OF ORGANIC CHEMISTRY (2016)
Cross-coupling of Aryl Sulfides Powered by N-Heterocyclic Carbene Ligands
Ke Gao et al.
JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN (2016)
Metal-Free Approach to Biaryls from Phenols and Aryl Sulfoxides by Temporarily Sulfur-Tethered Regioselective C-H/C-H Coupling
Tomoyuki Yanagi et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2016)
Metal-Free CH-CH-Type Cross-Coupling of Arenes and Alkynes Directed by a Multifunctional Sulfoxide Group
Jose A. Fernandez-Salas et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2016)
Cobalt(III)-Catalyzed C-C Coupling of Arenes with 7-Oxabenzonorbornadiene and 2-Vinyloxirane via C-H Activation
Lingheng Kong et al.
ORGANIC LETTERS (2016)
Ruthenium-Catalyzed, Site-Selective C-H Allylation of Indoles with Allyl Alcohols as Coupling Partners
Gangam Srikanth Kumar et al.
ORGANIC LETTERS (2016)
The emergence of sulfoxide and iodonio-based redox arylation as a synthetic tool
Alexandr Shafir
TETRAHEDRON LETTERS (2016)
Regioselectivity in palladium-catalysed direct arylation of 5-membered ring heteroaromatics
Charles Beromeo Bheeter et al.
CATALYSIS SCIENCE & TECHNOLOGY (2016)
Heterogeneously Catalyzed Direct C-H Thiolation of Heteroarenes
Suhelen Vasquez-Cespedes et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2015)
Dehydrative Direct C-H Allylation with Allylic Alcohols under [Cp*CoIII] Catalysis
Yudai Suzuki et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2015)
TFA-promoted direct C-H sulfenylation at the C2 position of non-protected indoles
Thomas Hostier et al.
CHEMICAL COMMUNICATIONS (2015)
Sulfoxide-Directed Metal-Free ortho-Propargylation of Aromatics and Heteroaromatics
Andrew J. Eberhart et al.
CHEMISTRY-A EUROPEAN JOURNAL (2015)
Iodine-Catalyzed Regioselective Sulfenylation of Indoles with Sodium Sulfinates
Fuhong Xiao et al.
ADVANCED SYNTHESIS & CATALYSIS (2014)
A Bronsted Acid Catalyzed Redox Arylation
Bo Peng et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2014)
Chemoselective Intermolecular a-Arylation of Amides**
Bo Peng et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2014)
Synthesis and evaluation of benzimidazole carbamates bearing indole moieties for antiproliferative and antitubulin activities
Qi Guan et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Indolylarylsulfones Carrying a Heterocyclic Tail as Very Potent and Broad Spectrum HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors
Valeria Famiglini et al.
JOURNAL OF MEDICINAL CHEMISTRY (2014)
Co(III)-Catalyzed C-H Activation/Formal SN-Type Reactions: Selective and Efficient Cyanation, Halogenation, and Allylation
Da-Gang Yu et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)
Sulfur Mediated Allylic C-H Alkylation of Tri- and Disubstituted Olefins
Gang Hu et al.
ORGANIC LETTERS (2014)
Recent Advances in Transition-Metal-Catalyzed C-S Activation: From Thioester to (Hetero)aryl Thioether
Fei Pan et al.
ACS CATALYSIS (2014)
Nucleophilic ortho-Propargylation of Aryl Sulfoxides: An Interrupted Pummerer/Allenyl Thio-Claisen Rearrangement Sequence
Andrew J. Eberhart et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2013)
Iodine-Catalyzed Regioselective Sulfenylation of Indoles with Sulfonyl Hydrazides
Fu-Lai Yang et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2013)
Transition-metal mediated carbon-sulfur bond activation and transformations
Liandi Wang et al.
CHEMICAL SOCIETY REVIEWS (2013)
Toward Highly Potent Cancer Agents by Modulating the C-2 Group of the Arylthioindole Class of Tubulin Polymerization Inhibitors
Giuseppe La Regina et al.
JOURNAL OF MEDICINAL CHEMISTRY (2013)
Design of Potent Poxvirus Inhibitors of the Heterodimeric Processivity Factor Required for Viral Replication
Manunya Nuth et al.
JOURNAL OF MEDICINAL CHEMISTRY (2013)
Iridium-Catalyzed Intermolecular Asymmetric Hydroheteroarylation of Bicycloalkenes
Christo S. Sevov et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
Sulfur(IV)-Mediated Transformations: From Ylide Transfer to Metal-Free Arylation of Carbonyl Compounds
Xueliang Huang et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
Chemistry and Biology of Indoles and Indazoles: A Mini-Review
Nasir Shafakat Ali et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2013)
Nucleophilic ortho-Allylation of Pyrroles and Pyrazoles: An Accelerated Pummerer/Thio-Claisen Rearrangement Sequence
Andrew J. Eberhart et al.
ORGANIC LETTERS (2013)
Synthesis and antioxidant activity of new C-3 sulfenyl indoles
Claudio C. Silveira et al.
TETRAHEDRON LETTERS (2013)
A Metal-Free Sulfenylation and Bromosulfenylation of Indoles: Controllable Synthesis of 3-Arylthioindoles and 2-Bromo-3-arylthioindoles
Dayun Huang et al.
ADVANCED SYNTHESIS & CATALYSIS (2012)
Unprecedented C-2 arylation of indole with diazonium salts: Syntheses of 2,3-disubstituted indoles and their antimicrobial activity
Seth Daly et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Substituted indole-1-acetic acids as potent and selective CRTh2 antagonists-discovery of AZD1981
Tim Luker et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Design and Synthesis of 2-Heterocyclyl-3-arylthio-1H-indoles as Potent Tubulin Polymerization and Cell Growth Inhibitors with Improved Metabolic Stability
Giuseppe La Regina et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Sulfoxide-Mediated α-Arylation of Carbonyl Compounds
Xueliang Huang et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2011)
Palladium-Catalyzed Direct 2-Alkylation of Indoles by Norbornene-Mediated Regioselective Cascade C-H Activation
Lei Jiao et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2011)
Nucleophilic Ortho Allylation of Aryl and Heteroaryl Sulfoxides
Andrew J. Eberhart et al.
ORGANIC LETTERS (2011)
Selective Catalytic C-H Alkylation of Alkenes with Alcohols
Dong-Hwan Lee et al.
SCIENCE (2011)
A Direct Ylide Transfer to Carbonyl Derivatives and Heteroaromatic Compounds
Xueliang Huang et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2010)
Beyond the Pummerer Reaction: Recent Developments in Thionium Ion Chemistry
Laura H. S. Smith et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2010)
Reaction of 2-(2,2,2-Trifluoroethylidene)-1,3-dithiane 1-Oxide with Ketones under Pummerer Conditions and Its Application to the Synthesis of 3-Trifluoromethyl-Substituted Five-Membered Heteroarenes
Takayuki Kobatake et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2010)
Inhibition of soluble epoxide hydrolase enhances the anti-inflammatory effects of aspirin and 5-lipoxygenase activation protein inhibitor in a murine model
Jun-Yan Liu et al.
BIOCHEMICAL PHARMACOLOGY (2010)
Synthesis and biological activities of novel indole derivatives as potent and selective PPARγ modulators
Yann Lamotte et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
The matricellular protein CCN1 induces fibroblast senescence and restricts fibrosis in cutaneous wound healing
Joon-Il Jun et al.
NATURE CELL BIOLOGY (2010)
Ruthenium Catalyzed Directing Group-Free C2-Selective Carbenoid Functionalization of Indoles by α-Aryldiazoesters
Wai-Wing Chan et al.
ORGANIC LETTERS (2010)
Visible Light-Mediated Intermolecular C-H Functionalization of Electron-Rich Heterocycles with Malonates
Laura Furst et al.
ORGANIC LETTERS (2010)
2-(2,2,2-Trifluoroethylidene)-1,3-dithiane Monoxide as a Trifluoromethylketene Equivalent
Suguru Yoshida et al.
ORGANIC LETTERS (2009)
Direct functionalization of nitrogen heterocycles via Rh-catalyzed C-H bond activation
Jared C. Lewis et al.
ACCOUNTS OF CHEMICAL RESEARCH (2008)
Novel indole-3-sulfonamides as potent HIV non-nucleoside reverse transcriptase inhibitors (NNRTIs)
Zhijian Zhao et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)
Gene family encoding the major toxins of lethal Amanita mushrooms
Heather E. Hallen et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2007)
Direct transition metal-catalyzed functionalization of heteroaromatic compounds
Ilya V. Seregin et al.
CHEMICAL SOCIETY REVIEWS (2007)
Arylthiopyrrole (AThP) derivatives as non-nucleoside HIV-1 reverse transcriptase inhibitors: Synthesis, structure-activity relationships, and docking studies (Part 1)
Roberto Di Santo et al.
CHEMMEDCHEM (2006)
Inhibition of five lipoxygenase activating protein (FLAP) by MK-886 decreases atherosclerosis in apoE/LDLR-double knockout mice
J Jawien et al.
EUROPEAN JOURNAL OF CLINICAL INVESTIGATION (2006)
Development of a novel, highly efficient halide-catalyzed sulfenylation of Indoles
M Tudge et al.
ORGANIC LETTERS (2006)
New arylthioindoles: Potent inhibitors of tubulin polymerization. 2. Structure-activity relationships and molecular modeling studies
G De Martino et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Design, molecular modeling, synthesis, and anti-HIV-1 activity of new indolyl aryl sulfones. Novel derivatives of the indole-2-carboxamide
Rino Ragno et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Docking and 3-D QSAR studies on indolyl aryl sulfones.: Binding mode exploration at the HIV-1 reverse transcriptase non-nucleoside binding site and design of highly active N-(2-hydroxyethyl)carboxamide and N-(2-hydroxyethyl)carbohydrazide derivatives
R Ragno et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
Rational design of 6-methylsulfonylindoles as selective cyclooxygenase-2 inhibitors
JA Campbell et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2004)
The Pummerer reaction: Methodology and strategy for the synthesis of heterocyclic compounds
SK Bur et al.
CHEMICAL REVIEWS (2004)
Novel indolyl aryl sulfones active against HIV-1 carrying NNRTI resistance mutations: Synthesis and SAR studies
R Silvestri et al.
JOURNAL OF MEDICINAL CHEMISTRY (2003)
New synthetic capabilities of sulfonium salts
VG Nenaidenko et al.
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY (2003)
Mechanism of the second sulfenylation of indole
P Hamel
JOURNAL OF ORGANIC CHEMISTRY (2002)
Pyrrolo[1,2-f]phenanthridines and related non-rigid analogues as antiviral agents
AM Almerico et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2002)
Structure-based design, synthesis and SAR of a novel series of thiopheneamidine urokinase plasminogen activator inhibitors
NL Subasinghe et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2001)
Share Paper
