Journal
TETRAHEDRON LETTERS
Volume 59, Issue 23, Pages 2243-2247Publisher
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tetlet.2018.04.036
Keywords
8-Aminoquinolines; Catalyzed-free; C-H functionalization; Halogenation; Hydrogen halide (HX)
Categories
Funding
- Major Scientific and Technological Innovation Projects of Hangzhou City - China [20162011A036]
- Natural Science Foundation of China - China [21376058]
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Simple and halide-atom economical HX reagents (X = Cl, Br and I) were applied to the remote C-H bond halogenation reaction of 8-aminoquinoline amides. This strategy features a broad substrate scope and good functional group tolerance. A series of CS-halogenated 8-aminoquinolines were obtained in moderate to good yields under mild conditions. (C) 2018 Elsevier Ltd. All rights reserved.
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