Journal
TETRAHEDRON LETTERS
Volume 59, Issue 21, Pages 2054-2056Publisher
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tetlet.2018.04.038
Keywords
C-H activation; Copper-catalyzed; Benzothiadiazine 1,1-dioxide; Benzenesulfonyl chloride; Trichloroacetonitrile; Primary amine
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Funding
- Research Council of Shahid Beheshti University of Medical Sciences
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The synthesis of functionalized benzothiadiazine 1,1-dioxide derivatives was achieved through a novel three-component intramolecular C-H activation reaction of trichloroacetonitrile, benzenesulfonyl chloride, and various primary amines. This reaction was performed in the presence of catalytic copper(I) and L-proline as the ligand in tetrahydrofuran at room temperature. (C) 2018 Elsevier Ltd. All rights reserved.
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