Journal
ORGANIC PROCESS RESEARCH & DEVELOPMENT
Volume 22, Issue 1, Pages 97-102Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.oprd.7b00370
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We report a five-step synthesis of 2-cyano-5-formyl-4-methyl-1H-indole through sequential functionalization of readily available 4-methyl-1H-indole. Cyano and aldehyde functionalities are regioselectively installed at the 2 and 5 position, respectively. The sequence is concise and high-yielding, amenable for kilogram scale production.
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