Journal
ORGANIC LETTERS
Volume 20, Issue 10, Pages 2880-2883Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.8b00905
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Funding
- NSFC [21372256, 21572264]
- Program for Changjiang Scholars and Innovative Research Team Project [IRT1042]
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A palladium-catalyzed enantioselective [4 + 2] cycloaddition reaction of vinyl benzoxazinones with sulfamate-derived cyclic imines is described, affording the tetrahydro-quinazolines bearing several functional rings in high yields (up to 99% yield) with good to excellent diastereoselectivities and excellent enantioselectivities (up to 96% ee). This reaction represents the first Pd-catalyzed asymmetric decarboxylative cycloaddition of vinyl benzoxazinones with imines.
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