Journal
ORGANIC LETTERS
Volume 20, Issue 7, Pages 1798-1801Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.8b00246
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Funding
- NSFC [21672033, 21372041]
- Jilin Province Natural Science Foundation [20160520140JH, 20160519003JH]
- Fundamental Research Funds for the Central Universities [2412017ZD001]
- Changbai Mountain Scholarship Program
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The development of an efficient, straightforward approach for access to a wide range of enantioenriched boron-containing 2,3-disubstituted indolines via highly chemo-, diastereo-, and enantioselective copper-catalyzed intramolecular boraylative cyclization of readily available 2-styrylimines is reported. This reaction proceeds under very mild conditions and displays a high degree of functional group compatibility. The practicability of this approach is demonstrated by a gram-scale reaction and further transformations of the chiral borylated indolines.
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