Journal
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
Volume 57, Issue 32, Pages 10338-10342Publisher
WILEY-V C H VERLAG GMBH
DOI: 10.1002/anie.201805258
Keywords
annulation; diaziridines; donor-acceptor cyclopropanes; nitrogen heterocycles; small ring systems
Categories
Funding
- Russian Science Foundation [17-73-10404]
- Russian Science Foundation [17-73-10404] Funding Source: Russian Science Foundation
Ask authors/readers for more resources
The first example of (3+3)-annulation of two different three-membered rings is reported herein. Donor-acceptor cyclopropanes in reaction with diaziridines were found to afford perhydropyridazine derivatives in high yields and diastereoselectivity under mild Lewis acid catalysis. The disclosed reaction is applicable for the broad substrate scope and exhibits an excellent functional group tolerance.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available
Share Paper
