Related references
Note: Only part of the references are listed.Beta blockers and cancer prognosis - The role of immortal time bias: A systematic review and meta-analysis
Janick Weberpals et al.
CANCER TREATMENT REVIEWS (2016)
Chemical Space of DNA-Encoded Libraries
Raphael M. Franzini et al.
JOURNAL OF MEDICINAL CHEMISTRY (2016)
Allosteric nanobodies reveal the dynamic range and diverse mechanisms of G-protein-coupled receptor activation
Dean P. Staus et al.
NATURE (2016)
Conformationally selective RNA aptamers allosterically modulate the β2-adrenoceptor
Alem W. Kahsai et al.
NATURE CHEMICAL BIOLOGY (2016)
Emerging Approaches to GPCR Ligand Screening for Drug Discovery
Punita Kumari et al.
TRENDS IN MOLECULAR MEDICINE (2015)
Cell-Based Selection Expands the Utility of DNA-Encoded Small-Molecule Library Technology to Cell Surface Drug Targets: Identification of Novel Antagonists of the NK3 Tachykinin Receptor
Zining Wu et al.
ACS COMBINATORIAL SCIENCE (2015)
Ligand bias prevents class equality among beta-blockers
Vaidehi J. Thanawala et al.
CURRENT OPINION IN PHARMACOLOGY (2014)
Divergent Transducer-specific Molecular Efficacies Generate Biased Agonism at a G Protein-coupled Receptor ( GPCR)
Ryan T. Strachan et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2014)
Visualization of arrestin recruitment by a G-protein-coupled receptor
Arun K. Shukla et al.
NATURE (2014)
Beta-Blockers in the Management of Hypertension and/or Chronic Kidney Disease
Hirofumi Tomiyama et al.
INTERNATIONAL JOURNAL OF HYPERTENSION (2014)
Advances in G Protein-Coupled Receptor Allostery: From Function to Structure
Arthur Christopoulos
MOLECULAR PHARMACOLOGY (2014)
International Union of Basic and Clinical Pharmacology. XC. Multisite Pharmacology: Recommendations for the Nomenclature of Receptor Allosterism and Allosteric Ligands
Arthur Christopoulos et al.
PHARMACOLOGICAL REVIEWS (2014)
Regulation of β2-Adrenergic Receptor Function by Conformationally Selective Single-Domain Intrabodies
Dean P. Staus et al.
MOLECULAR PHARMACOLOGY (2014)
Structure of active β-arrestin-1 bound to a G-protein-coupled receptor phosphopeptide
Arun K. Shukla et al.
NATURE (2013)
Emerging paradigms in GPCR allostery: implications for drug discovery
Denise Wootten et al.
NATURE REVIEWS DRUG DISCOVERY (2013)
Thermodynamics and Docking of Agonists to the β2-Adrenoceptor Determined Using [3H](R,R′)-4-Methoxyfenoterol as the Marker Ligand
Lawrence Toll et al.
MOLECULAR PHARMACOLOGY (2012)
20 years of DNA-encoded chemical libraries
Luca Mannocci et al.
CHEMICAL COMMUNICATIONS (2011)
Quantifying Ligand Bias at Seven-Transmembrane Receptors
Sudarshan Rajagopal et al.
MOLECULAR PHARMACOLOGY (2011)
Structure of a nanobody-stabilized active state of the β2 adrenoceptor
Soren G. F. Rasmussen et al.
NATURE (2011)
Crystal structure of the β2 adrenergic receptor-Gs protein complex
Soren G. F. Rasmussen et al.
NATURE (2011)
Distinct Phosphorylation Sites on the β2-Adrenergic Receptor Establish a Barcode That Encodes Differential Functions of β-Arrestin
Kelly N. Nobles et al.
SCIENCE SIGNALING (2011)
Therapeutic potential of β-arrestin- and G protein-biased agonists
Erin J. Whalen et al.
TRENDS IN MOLECULAR MEDICINE (2011)
Structural insights into adrenergic receptor function and pharmacology
Brian K. Kobilka
TRENDS IN PHARMACOLOGICAL SCIENCES (2011)
In Vitro Selection of a DNA-Templated Small-Molecule Library Reveals a Class of Macrocyclic Kinase Inhibitors
Ralph E. Kleiner et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2010)
Design, synthesis and selection of DNA-encoded small-molecule libraries
Matthew A. Clark et al.
NATURE CHEMICAL BIOLOGY (2009)
β2-adrenergic receptor signaling and desensitization elucidated by quantitative modeling of real time cAMP dynamics
Jonathan D. Violin et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2008)
National asthma education and prevention program - Expert panel report 3 (EPR-3): Guidelines for the diagnosis and management of asthma - Summary report 2007
[Anonymous]
JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY (2007)
A monoclonal antibody for G protein-coupled receptor crystallography
Peter W. Day et al.
NATURE METHODS (2007)
A monomeric G protein-coupled receptor isolated in a high-density lipoprotein particle efficiently activates its G protein
Matthew R. Whorton et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2007)
Seven transmembrane receptors: something old, something new
R. J. Lefkowitz
ACTA PHYSIOLOGICA (2007)
G-protein-coupled receptor kinase specificity for β-arrestin recruitment to the β2-adrenergic receptor revealed by fluorescence resonance energy transfer
Jonathan D. Violin et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2006)
Maraviroc (UK-427,857), a potent, orally bioavailable, and selective small-molecule inhibitor of chemokine receptor CCR5 with broad-spectrum anti-human immunodeficiency virus type 1 activity
P Dorr et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2005)
Functional G protein-coupled receptor assays for primary and secondary screening
RM Eglen
COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING (2005)
Cinacalcet HCl, an oral calcimimetic agent for the treatment of secondary hyperparathyroidism in Hemodialysis and peritoneal dialysis: A randomized, double-blind, multicenter study
JS Lindberg et al.
JOURNAL OF THE AMERICAN SOCIETY OF NEPHROLOGY (2005)
The stability of the G protein-coupled receptor-β-arrestin interaction determines the mechanism and functional consequence of ERK activation
A Tohgo et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2003)
Differential affinities of visual arrestin, βarrestin1, and βarrestin2 for G protein-coupled receptors delineate two major classes of receptors
RH Oakley et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2000)