Journal
ORGANIC LETTERS
Volume 19, Issue 20, Pages 5665-5668Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.7b02824
Keywords
-
Categories
Funding
- SERB [EMR/2014/385]
- CSIR
- T.R.G. (N-PDF
- DST), India
Ask authors/readers for more resources
The methylphenyl sulfoximine (MPS) directing group (DG) successfully promotes the one-pot double annulation of acrylic acids with alkynes under Ru catalysis, which is unprecedented. Diverse arrays of pyrido-fused-isoquinolinone skeletons are fabricated from acrylamides, creating two C-C and two C-N bonds in a single operation. The unsymmetrical annulation with two distinct alkynes is presented. The recovery of methylphenyl sulfoxide, a precursor of MPS, validates the synthetic adaptability of transformable-DG (T(f)DG) in C-H activation
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available